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Published in Journal of medicinal chemistry (26.10.2017)
Published in Journal of medicinal chemistry (26.10.2017)
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Discovery and optimization of novel pyridines as highly potent and selective glycogen synthase kinase 3 inhibitors
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Published in ACS medicinal chemistry letters (13.10.2011)
Published in ACS medicinal chemistry letters (13.10.2011)
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Inhibition of prenylated KRAS in a lipid environment
Jansen, Johanna M, Wartchow, Charles, Jahnke, Wolfgang, Fong, Susan, Tsang, Tiffany, Pfister, Keith, Zavorotinskaya, Tatiana, Bussiere, Dirksen, Cheng, Jan Marie, Crawford, Kenneth, Dai, Yumin, Dove, Jeffrey, Fang, Eric, Feng, Yun, Florent, Jean-Michel, Fuller, John, Gossert, Alvar D, Hekmat-Nejad, Mohammad, Henry, Chrystèle, Klopp, Julia, Lenahan, William P, Lingel, Andreas, Ma, Sylvia, Meyer, Arndt, Mishina, Yuji, Narberes, Jamie, Pardee, Gwynn, Ramurthy, Savithri, Rieffel, Sebastien, Stuart, Darrin, Subramanian, Sharadha, Tandeske, Laura, Widger, Stephania, Widmer, Armin, Winterhalter, Aurelie, Zaror, Isabel, Hardy, Stephen
Published in PloS one (06.04.2017)
Published in PloS one (06.04.2017)
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Synthesis and in Vitro and in Vivo Evaluation of Phosphoinositide-3-kinase Inhibitors
Burger, Matthew T, Knapp, Mark, Wagman, Allan, Ni, Zhi-Jie, Hendrickson, Thomas, Atallah, Gordana, Zhang, Yanchen, Frazier, Kelly, Verhagen, Joelle, Pfister, Keith, Ng, Simon, Smith, Aaron, Bartulis, Sarah, Merrit, Hanne, Weismann, Marion, Xin, Xiaohua, Haznedar, Joshua, Voliva, Charles F, Iwanowicz, Ed, Pecchi, Sabina
Published in ACS medicinal chemistry letters (13.01.2011)
Published in ACS medicinal chemistry letters (13.01.2011)
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Synthesis of cyclic and acyclic enol ethers (vinyl ethers)
Gassman, Paul G, Burns, Stephen J, Pfister, Keith B
Published in Journal of organic chemistry (01.03.1993)
Published in Journal of organic chemistry (01.03.1993)
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Biased Complement Diversity Selection for Effective Exploration of Chemical Space in Hit-Finding Campaigns
Jansen, Johanna M, De Pascale, Gianfranco, Fong, Susan, Lindvall, Mika, Moser, Heinz E, Pfister, Keith, Warne, Bob, Wartchow, Charles
Published in Journal of chemical information and modeling (28.05.2019)
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Azaindoles as Zinc‐Binding Small‐Molecule Inhibitors of the JAMM Protease CSN5
Altmann, Eva, Erbel, Paul, Renatus, Martin, Schaefer, Michael, Schlierf, Anita, Druet, Adelaide, Kieffer, Laurence, Sorge, Mickael, Pfister, Keith, Hassiepen, Ulrich, Jones, Matthew, Ruedisser, Simon, Ostermeier, Daniela, Martoglio, Bruno, Jefferson, Anne B., Quancard, Jean
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Discovery of a Selective and Potent Inhibitor of Mitogen-Activated Protein Kinase-Interacting Kinases 1 and 2 (MNK1/2) Utilizing Structure-Based Drug Design
Han, Wooseok, Ding, Yu, Xu, Yongjin, Pfister, Keith, Zhu, Shejin, Warne, Bob, Doyle, Mike, Aikawa, Mina, Amiri, Payman, Appleton, Brent, Stuart, Darrin D, Fanidi, Abdallah, Shafer, Cynthia M
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SHIN JIN SOO, NEYTS JOHAN, LEE SANG HO, LEE CHONG KYO, KIM HAE SOO, POON DANIEL, PFISTER KEITH BRUCE, CHAKRASALI PRASHANT, KIM CHONSAENG, MALPANI YASHWARDHAN R, JUNG YOUNG SIK, HAN SOO BONG
Year of Publication 21.02.2023
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Year of Publication 21.02.2023
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Year of Publication 21.02.2023
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Year of Publication 21.02.2023
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4-(Aminoalkylamino)-3-benzimidazole-quinolinones as potent CHK-1 inhibitors
Ni, Zhi-Jie, Barsanti, Paul, Brammeier, Nathan, Diebes, Anthony, Poon, Daniel J., Ng, Simon, Pecchi, Sabina, Pfister, Keith, Renhowe, Paul A., Ramurthy, Savithri, Wagman, Allan S., Bussiere, Dirksen E., Le, Vincent, Zhou, Yasheen, Jansen, Johanna M., Ma, Sylvia, Gesner, Thomas G.
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
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Abstract B38: Inhibiting mutated KRAS, a broken switch of effector pathways
Jansen, Johanna, Jahnke, Wolfgang, Fong, Susan, Tandeske, Laura, Wartchow, Charles, Pfister, Keith, Zavorotinskaya, Tatiana, Blechschmidt, Anke, Bussiere, Dirksen, Dai, Yumin, Dove, Jeff, Fang, Eric, Farley, David, Florent, Jean-Michel, Fuller, John, Gokhin, Simona, Gossert, Alvar, Hekmat-Nejad, Mohammad, Henry, Chrystèle, Klopp, Julia, Lenahan, Bill, Lingel, Andreas, Meyer, Arndt, Narberes, Jamie, Pardee, Gwynn, Paris, C Gregory, Ramurthy, Savithri, Renhowe, Paul, Rieffel, Sebastien, Shoemaker, Kevin, Subramanian, Sharadha, Tsang, Tiffany, Widger, Stephania, Widmer, Armin, Zaror, Isabel, Hardy, Stephen
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Azaindoles as Zinc‐Binding Small‐Molecule Inhibitors of the JAMM Protease CSN5
Altmann, Eva, Erbel, Paul, Renatus, Martin, Schaefer, Michael, Schlierf, Anita, Druet, Adelaide, Kieffer, Laurence, Sorge, Mickael, Pfister, Keith, Hassiepen, Ulrich, Jones, Matthew, Ruedisser, Simon, Ostermeier, Daniela, Martoglio, Bruno, Jefferson, Anne B., Quancard, Jean
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PYRAZINYLPYRIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES
HU CHENG, BARSANTI PAUL A, SENDZIK MARTIN, PFISTER KEITH B, SUTTON JAMES
Year of Publication 09.07.2012
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Year of Publication 09.07.2012
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HAN WOOSEOK, MIN ZHONGCHENG, ZHANG QIONG, LEE PATRICK, LINDVALL MIKA, POON DANIEL, HUANG ZILIN, JIANG QUN, PAN YUE, ZHOU JIANGUANG, BAGDANOFF JEFFREY T, JIN JEFF XIANMING, KOU XIANG, RAUNIYAR VIVEK, DING YU, ZHU SHEJIN, PFISTER KEITH BRUCE, WANG XIAOJING MICHAEL, PECCHI SABINA
Year of Publication 05.07.2016
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Year of Publication 05.07.2016
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3-(AMINOARYL)-PYRIDINE COMPOUNDS
HU CHENG, BARSANTI PAUL A, SENDZIK MARTIN, ANTONIOS MCCREA WILLIAM R, MARTIN ERIC J, WAN LIFENG, PAN YUE, JIN XIANMING, PFISTER KEITH B, SUTTON JAMES
Year of Publication 23.10.2013
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Year of Publication 23.10.2013
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