The Lactol Route to Fesoterodine: An Amine-Promoted Friedel–Crafts Alkylation on Commercial Scale
Dirat, Olivier, Bibb, Andrew J, Burns, Colin M, Checksfield, Graham D, Dillon, Barry R, Field, Stuart E, Fussell, Steven J, Green, Stuart P, Mason, Clive, Mathew, Jinu, Mathew, Suju, Moses, Ian B, Nikiforov, Petar I, Pettman, Alan J, Susanne, Flavien
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Published in Organic process research & development (16.09.2011)
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Development of a Scaleable Process for the Synthesis of the A2a Agonist, UK-371,104
Challenger, Stephen, Dessi, Yann, Fox, Darrell E, Hesmondhalgh, Lynsey C, Pascal, Pierre, Pettman, Alan J, Smith, Julian D
Published in Organic process research & development (01.07.2008)
Published in Organic process research & development (01.07.2008)
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Enzymatic Desymmetrization Route to Ethyl [3-(2-Amino-2-methylpropyl)phenyl]acetate
de Koning, Pieter D, Gladwell, Iain R, Morrison, Natalie A, Moses, Ian B, Panesar, Maninder S, Pettman, Alan J, Thomson, Nicholas M, Yazbeck, Daniel R
Published in Organic process research & development (15.07.2011)
Published in Organic process research & development (15.07.2011)
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Accelerated Process Development of Pharmaceuticals: Selective Catalytic Hydrogenations of Nitro Compounds Containing Other Functionalities
Hoogenraad, Marcel, van der Linden, Johannes B., Smith, Alan A., Hughes, Bob, Derrick, Andrew M., Harris, Laurence J., Higginson, Paul D., Pettman, Alan J.
Published in Organic process research & development (01.05.2004)
Published in Organic process research & development (01.05.2004)
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Commercial Route Development Toward PF-07265807, an AXL-MER Inhibitor Oncology Candidate
Critcher, Douglas J., Ashcroft, Christopher Paul, Pettman, Alan J., Badland, Matthew, Szpera, Robert, Waddington, William
Published in Organic process research & development (19.07.2024)
Published in Organic process research & development (19.07.2024)
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Real-time monitoring of nitrile biotransformations by mid-infrared spectroscopy
Dadd, Michael R., Sharp, David C.A., Pettman, Alan J., Knowles, Christopher J.
Published in Journal of microbiological methods (01.06.2000)
Published in Journal of microbiological methods (01.06.2000)
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Regioselective biotransformation of the dinitrile compounds 2-, 3- and 4-(cyanomethyl) benzonitrile by the soil bacterium Rhodococcus rhodochrous LL100-21
DADD, Michael R, CLARIDGE, Timothy D. W, WALTON, Robert, PETTMAN, Alan J, KNOWLES, Christopher J
Published in Enzyme and microbial technology (05.07.2001)
Published in Enzyme and microbial technology (05.07.2001)
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A robust method to heterogenise and recycle group 9 catalystsElectronic supplementary information (ESI) available: Complete experimental data for novel compounds, catalytic experiments and crystal structure determination described. CCDC 913126. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c3cc42550a
Lucas, Stephanie J, Crossley, Benjamin D, Pettman, Alan J, Vassileiou, Antony D, Screen, Thomas E. O, Blacker, A. John, McGowan, Patrick C
Year of Publication 23.05.2013
Year of Publication 23.05.2013
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Development of an Enabling Route to PF-00610355: A Novel Inhaled β2-Adrenoreceptor Agonist
de Koning, Pieter D., Gladwell, Iain R., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)
Published in Organic process research & development (18.11.2011)
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Development of an Enabling Route to PF-00610355: A Novel Inhaled beta(2)-Adrenoreceptor Agonist
de Koning, Pieter D., Gladwell, Iain R., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (01.11.2011)
Published in Organic process research & development (01.11.2011)
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Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled beta(2)-Adrenoreceptor Agonist
de Koning, Pieter D., Castro, Nieves, Gladwell, Iain R., Morrison, Natalie A., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (01.11.2011)
Published in Organic process research & development (01.11.2011)
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Journal Article
Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled β2-Adrenoreceptor Agonist
de Koning, Pieter D., Castro, Nieves, Gladwell, Iain R., Morrison, Natalie A., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)
Published in Organic process research & development (18.11.2011)
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Journal Article
Development of an Enabling Route to PF-00610355: A Novel Inhaled β 2 -Adrenoreceptor Agonist
de Koning, Pieter D., Gladwell, Iain R., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)
Published in Organic process research & development (18.11.2011)
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Journal Article
Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled β 2 -Adrenoreceptor Agonist
de Koning, Pieter D., Castro, Nieves, Gladwell, Iain R., Morrison, Natalie A., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)
Published in Organic process research & development (18.11.2011)
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