Structure–Activity Relationships of Bis-Intercalating Peptides and Their Application as Antibody–Drug Conjugate Payloads
Petersen, Mark E., Brant, Michael G., Lasalle, Manuel, Fung, Vincent K. C., Rojas, Andrea Hernandez, Wong, Jodi, Das, Samir, Barnscher, Stuart D., Rich, Jamie R., Winters, Geoffrey C.
Published in Journal of medicinal chemistry (22.06.2023)
Published in Journal of medicinal chemistry (22.06.2023)
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Journal Article
Chemical synthesis of Shiga toxin subunit B using a next-generation traceless "helping hand" solubilizing tag
Fulcher, James M, Petersen, Mark E, Giesler, Riley J, Cruz, Zachary S, Eckert, Debra M, Francis, J. Nicholas, Kawamoto, Eric M, Jacobsen, Michael T, Kay, Michael S
Published in Organic & biomolecular chemistry (28.12.2019)
Published in Organic & biomolecular chemistry (28.12.2019)
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The Integrated Probabilistic Data Association Filter Adapted to Lie Groups
Petersen, Mark E., Beard, Randal W.
Published in IEEE transactions on aerospace and electronic systems (01.06.2023)
Published in IEEE transactions on aerospace and electronic systems (01.06.2023)
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Generation and structure-activity relationships of novel imidazo-thienopyridine based TLR7 agonists: application as payloads for immunostimulatory antibody drug-conjugates
Brant, Michael G., Garnett, Graham A.E., Guedia, Joy, Lasalle, Manuel, Lawn, Samuel, Petersen, Mark E., Duan, Renee, Mendez-Campos, José, Hirkala-Schaefer, Truman, Winters, Geoffrey C., Barnscher, Stuart D.
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
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Journal Article
Design and Evaluation of ZD06519, a Novel Camptothecin Payload for Antibody Drug Conjugates
Petersen, Mark E, Brant, Michael G, Lasalle, Manuel, Das, Samir, Duan, Renee, Wong, Jodi, Ding, Tong, Wu, Kaylee J, Siddappa, Dayananda, Fang, Chen, Zhang, Wen, Wu, Alex M L, Hirkala-Schaefer, Truman, Garnett, Graham A E, Fung, Vincent, Yang, Luying, Hernandez Rojas, Andrea, Lawn, Samuel O, Barnscher, Stuart D, Rich, Jamie R, Colombo, Raffaele
Published in Molecular cancer therapeutics (02.05.2024)
Published in Molecular cancer therapeutics (02.05.2024)
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Journal Article
Synthesis of hydrophobic insulin-based peptides using a helping hand strategy
Disotuar, Maria M, Petersen, Mark E, Nogueira, Jason M, Kay, Michael S, Chou, Danny Hung-Chieh
Published in Organic & biomolecular chemistry (13.02.2019)
Published in Organic & biomolecular chemistry (13.02.2019)
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Journal Article
Synthesis of tumor necrosis factor α for use as a mirror-image phage display target
Petersen, Mark E, Jacobsen, Michael T, Kay, Michael S
Published in Organic & biomolecular chemistry (21.06.2016)
Published in Organic & biomolecular chemistry (21.06.2016)
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Journal Article
Synthesis and Biological Evaluation of Fluorescent Bryostatin Analogues
Cummins, Thomas J., Kedei, Noemi, Czikora, Agnes, Lewin, Nancy E., Kirk, Sharon, Petersen, Mark E., McGowan, Kevin M., Chen, Jin‐Qiu, Luo, Xiaoling, Johnson, Randall C., Ravichandran, Sarangan, Blumberg, Peter M., Keck, Gary E.
Published in Chembiochem : a European journal of chemical biology (16.04.2018)
Published in Chembiochem : a European journal of chemical biology (16.04.2018)
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Biological activity of the bryostatin analog Merle 23 on mouse epidermal cells and mouse skin
Kelsey, Jessica S., Cataisson, Christophe, Chen, Jinqiu, Herrmann, Michelle A., Petersen, Mark E., Baumann, David O., McGowan, Kevin M., Yuspa, Stuart H., Keck, Gary E., Blumberg, Peter M.
Published in Molecular carcinogenesis (01.12.2016)
Published in Molecular carcinogenesis (01.12.2016)
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Molecular Systems Pharmacology: Isoelectric Focusing Signature of Protein Kinase Cδ Provides an Integrated Measure of Its Modulation in Response to Ligands
Kedei, Noemi, Chen, Jin-Qiu, Herrmann, Michelle A, Telek, Andrea, Goldsmith, Paul K, Petersen, Mark E, Keck, Gary E, Blumberg, Peter M
Published in Journal of medicinal chemistry (26.06.2014)
Published in Journal of medicinal chemistry (26.06.2014)
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Journal Article
Synthesis of hydrophobic insulin-based peptides using a helping hand strategyElectronic supplementary information (ESI) available: Detailed synthesis procedure and mass spectrometry data; along with cell assay protocol. See DOI: 10.1039/c8ob01212a
Disotuar, Maria M, Petersen, Mark E, Nogueira, Jason M, Kay, Michael S, Chou, Danny Hung-Chieh
Year of Publication 13.02.2019
Year of Publication 13.02.2019
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Abstract 3127: Development of three-dimensional cancer cell line spheroid models for the in vitro functional characterization of cytotoxic antibody-drug conjugates
Wong, Jodi, Rojas, Andrea Hernández, Bissessur, Allysha, Degefie, Lemlem T., Sagoe-Wagner, Araba P., Das, Samir, Fung, Vincent, Yin, Kevin, Duan, Renee, Lawn, Sam, Madera, Laurence, Kim, Catrina Mi Jung, Wu, Alex, Petersen, Mark E., Colombo, Raffaele, Rich, Jamie R., Barnscher, Stuart D.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract 1862: ZW191 - a FRα-targeting antibody drug conjugate with strong preclinical activity across multiple FRα-expressing indications
Lawn, Sam, Rojas, Andrea Hernandez, Colombo, Raffaele, Wong, Jodi, Wu, Kaylee, Fung, Vincent, Lasalle, Manuel, Petersen, Mark E., Degefie, Lemlem, Sagoe-Wagner, Araba, Urosev, Dunja, Yang, Luying, Wu, Ambroise, Kim, Catrina, Chua, Amos, Stahl, Kurt, Winters, Geoffrey C., Fann, John C., Rich, Jamie, Barnscher, Stuart
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Journal Article
Abstract 2101: Comparison of transcriptional response to phorbol ester, bryostatin 1, and bryostatin analogue in LNCaP and U937 cells provides insight into their differential mechanism
Kedei, Noemi, Michalowski, Aleksandra M., Petersen, Mark E., Keck, Gary E., Blumberg, Peter M.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Abstract 2658: ZW251, a novel glypican-3-targeting antibody drug conjugate bearing a topoisomerase 1 inhibitor payload
Madera, Laurence, Rojas, Andrea Hernández, Colombo, Raffaele, Wu, Alex, Piscitelli, Chayne L., Urosev, Dunja, Bissessur, Allysha, Cheng, Chi Wing, Duan, Renee, Kim, Catrina, Yin, Kevin, Fung, Vincent, Wu, Kaylee, Cheung, Winnie, Alonzo, Diego A., Petersen, Mark E., Barnscher, Stuart D., Rich, Jamie R.
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Abstract 3815: Comparison of transcriptional response to phorbol ester, bryostatin 1, and bryostatin analogues in LNCaP and U937 cancer cell lines provides insight into their differential mechanism of action
Kedei, Noemi, Telek, Andrea, Michalowski, Aleksandra M., Kraft, Matthew B., Li, Wei, Poudel, Yam B., Rudra, Arnab, Petersen, Mark E., Keck, Gary E., Blumberg, Peter M.
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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