Details Matter in Structure-based Drug Design
Kuhn, Bernd, Peters, Jens-Uwe, Rudolph, Markus G, Mohr, Peter, Stahl, Martin, Tosstorff, Andreas
Published in Chimia (01.08.2023)
Published in Chimia (01.08.2023)
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Journal Article
Fenobam: A Clinically Validated Nonbenzodiazepine Anxiolytic Is a Potent, Selective, and Noncompetitive mGlu5 Receptor Antagonist with Inverse Agonist Activity
Porter, Richard H P, Jaeschke, Georg, Spooren, Will, Ballard, Theresa M, Büttelmann, Bernd, Kolczewski, Sabine, Peters, Jens-Uwe, Prinssen, Eric, Wichmann, Jürgen, Vieira, Eric, Mühlemann, Andreas, Gatti, Silvia, Mutel, Vincent, Malherbe, Pari
Published in The Journal of pharmacology and experimental therapeutics (01.11.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2005)
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Metabotropic Glutamate Receptor 5 Negative Allosteric Modulators: Discovery of 2‑Chloro-4-[1-(4-fluorophenyl)-2,5-dimethyl‑1H‑imidazol-4-ylethynyl]pyridine (Basimglurant, RO4917523), a Promising Novel Medicine for Psychiatric Diseases
Jaeschke, Georg, Kolczewski, Sabine, Spooren, Will, Vieira, Eric, Bitter-Stoll, Nadia, Boissin, Patrick, Borroni, Edilio, Büttelmann, Bernd, Ceccarelli, Simona, Clemann, Nicole, David, Beatrice, Funk, Christoph, Guba, Wolfgang, Harrison, Anthony, Hartung, Thomas, Honer, Michael, Huwyler, Jörg, Kuratli, Martin, Niederhauser, Urs, Pähler, Axel, Peters, Jens-Uwe, Petersen, Ann, Prinssen, Eric, Ricci, Antonio, Rueher, Daniel, Rueher, Marianne, Schneider, Manfred, Spurr, Paul, Stoll, Theodor, Tännler, Daniel, Wichmann, Jürgen, Porter, Richard H, Wettstein, Joseph G, Lindemann, Lothar
Published in Journal of medicinal chemistry (12.02.2015)
Published in Journal of medicinal chemistry (12.02.2015)
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Journal Article
Inhibitors of dipeptidyl peptidase IV--recent advances and structural views
Hunziker, Daniel, Hennig, Michael, Peters, Jens-Uwe
Published in Current topics in medicinal chemistry (01.12.2005)
Published in Current topics in medicinal chemistry (01.12.2005)
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Journal Article
Safety screening in early drug discovery: An optimized assay panel
Bendels, Stefanie, Bissantz, Caterina, Fasching, Bernhard, Gerebtzoff, Grégori, Guba, Wolfgang, Kansy, Manfred, Migeon, Jacques, Mohr, Susanne, Peters, Jens-Uwe, Tillier, Fabien, Wyler, René, Lerner, Christian, Kramer, Christian, Richter, Hans, Roberts, Sonia
Published in Journal of pharmacological and toxicological methods (01.09.2019)
Published in Journal of pharmacological and toxicological methods (01.09.2019)
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Journal Article
Can we discover pharmacological promiscuity early in the drug discovery process?
Peters, Jens-Uwe, Hert, Jérôme, Bissantz, Caterina, Hillebrecht, Alexander, Gerebtzoff, Grégori, Bendels, Stefanie, Tillier, Fabien, Migeon, Jacques, Fischer, Holger, Guba, Wolfgang, Kansy, Manfred
Published in Drug discovery today (01.04.2012)
Published in Drug discovery today (01.04.2012)
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Journal Article
Metabolite Identification via LC-SPE-NMR-MS of the In vitro Biooxidation Products of a Lead mGlu5 Allosteric Antagonist and Impact on the Improvement of Metabolic Stability in the Series
Ceccarelli, Simona M., Schlotterbeck, Götz, Boissin, Patrick, Binder, Martin, Buettelmann, Bernd, Hanlon, Steven, Jaeschke, Georg, Kolczewski, Sabine, Kupfer, Ernst, Peters, Jens-Uwe, Porter, Richard H. P., Prinssen, Eric P., Rueher, Marianne, Ruf, Iris, Spooren, Will, Stämpfli, Andreas, Vieira, Eric
Published in ChemMedChem (11.01.2008)
Published in ChemMedChem (11.01.2008)
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Journal Article
Tyramine fragment binding to BACE-1
Kuglstatter, Andreas, Stahl, Martin, Peters, Jens-Uwe, Huber, Walter, Stihle, Martine, Schlatter, Daniel, Benz, Jörg, Ruf, Armin, Roth, Doris, Enderle, Thilo, Hennig, Michael
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Journal Article
Synthesis of potential drug metabolites by a modified Udenfriend reaction
Slavik, Roger, Peters, Jens-Uwe, Giger, Rudolf, Bürkler, Markus, Bald, Eric
Published in Tetrahedron letters (16.02.2011)
Published in Tetrahedron letters (16.02.2011)
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Journal Article
Lead Generation: Sowing the Seeds for Future Success
Konrad H. Bleicher, Matthias Nettekoven, Jens-Uwe Peters, René Wyler
Published in Chimia (01.09.2004)
Published in Chimia (01.09.2004)
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Journal Article
1,3-Disubstituted 4-aminopiperidines as useful tools in the optimization of the 2-aminobenzo[a]quinolizine dipeptidyl peptidase IV inhibitors
Lübbers, Thomas, Böhringer, Markus, Gobbi, Luca, Hennig, Michael, Hunziker, Daniel, Kuhn, Bernd, Löffler, Bernd, Mattei, Patrizio, Narquizian, Robert, Peters, Jens-Uwe, Ruff, Yves, Wessel, Hans Peter, Wyss, Pierre
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
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Journal Article
A facile Horner–Wadsworth–Emmons route to 2-quinolones
Peters, Jens-Uwe, Capuano, Tony, Weber, Silja, Kritter, Stéphane, Sägesser, Matthias
Published in Tetrahedron letters (16.06.2008)
Published in Tetrahedron letters (16.06.2008)
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Journal Article
Discovery of potent, balanced and orally active dual NK1/NK3 receptor ligands
Peters, Jens-Uwe, Hoffmann, Torsten, Schnider, Patrick, Stadler, Heinz, Koblet, Andreas, Alker, André, Poli, Sonia Maria, Ballard, Theresa M., Spooren, Will, Steward, Lucinda, Sleight, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
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Journal Article
Cyclic guanidines as dual 5-HT5A/5-HT7 receptor ligands : Structure-activity relationship elucidation
PETERS, Jens-Uwe, LÜBBERS, Thomas, ALANINE, Alexander, KOLCZEWSKI, Sabine, BLASCO, Francesca, STEWARD, Lucinda
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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