Identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by Diketo acid derivatives
Corona, Angela, Di Leva, Francesco Saverio, Thierry, Sylvain, Pescatori, Luca, Cuzzucoli Crucitti, Giuliana, Subra, Frederic, Delelis, Olivier, Esposito, Francesca, Rigogliuso, Giuseppe, Costi, Roberta, Cosconati, Sandro, Novellino, Ettore, Di Santo, Roberto, Tramontano, Enzo
Published in Antimicrobial agents and chemotherapy (01.10.2014)
Published in Antimicrobial agents and chemotherapy (01.10.2014)
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Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives
Saccoliti, Francesco, Angiulli, Gabriella, Pupo, Giovanni, Pescatori, Luca, Madia, Valentina Noemi, Messore, Antonella, Colotti, Gianni, Fiorillo, Annarita, Scipione, Luigi, Gramiccia, Marina, Di Muccio, Trentina, Di Santo, Roberto, Costi, Roberta, Ilari, Andrea
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
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Diaryl Disulfides as Novel Stabilizers of Tumor Suppressor Pdcd4
Schmid, Tobias, Blees, Johanna S, Bajer, Magdalena M, Wild, Janine, Pescatori, Luca, Cuzzucoli Crucitti, Giuliana, Scipione, Luigi, Costi, Roberta, Henrich, Curtis J, Brüne, Bernhard, Colburn, Nancy H, Di Santo, Roberto
Published in PloS one (16.03.2016)
Published in PloS one (16.03.2016)
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Discovery and Pharmacological Profile of New 1H‑Indazole-3-carboxamide and 2H‑Pyrrolo[3,4‑c]quinoline Derivatives as Selective Serotonin 4 Receptor Ligands
Furlotti, Guido, Alisi, Maria Alessandra, Apicella, Claudia, Capezzone de Joannon, Alessandra, Cazzolla, Nicola, Costi, Roberta, Cuzzucoli Crucitti, Giuliana, Garrone, Beatrice, Iacovo, Alberto, Magarò, Gabriele, Mangano, Giorgina, Miele, Gaetano, Ombrato, Rosella, Pescatori, Luca, Polenzani, Lorenzo, Rosi, Federica, Vitiello, Marco, Di Santo, Roberto
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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Salmonella enterica serovar Typhimurium growth is inhibited by the concomitant binding of Zn(II) and a pyrrolyl-hydroxamate to ZnuA, the soluble component of the ZnuABC transporter
Ilari, Andrea, Pescatori, Luca, Di Santo, Roberto, Battistoni, Andrea, Ammendola, Serena, Falconi, Mattia, Berlutti, Francesca, Valenti, Piera, Chiancone, Emilia
Published in Biochimica et biophysica acta (01.03.2016)
Published in Biochimica et biophysica acta (01.03.2016)
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Structure–Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV‑1 Integrase and Reverse Transcriptase Ribonuclease H Domain
Cuzzucoli Crucitti, Giuliana, Métifiot, Mathieu, Pescatori, Luca, Messore, Antonella, Madia, Valentina Noemi, Pupo, Giovanni, Saccoliti, Francesco, Scipione, Luigi, Tortorella, Silvano, Esposito, Francesca, Corona, Angela, Cadeddu, Marta, Marchand, Christophe, Pommier, Yves, Tramontano, Enzo, Costi, Roberta, Di Santo, Roberto
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
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Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1H-pyrrolyl)(phenyl)methyl-1H-innidazole Derivatives as Antiprotozoal Agents
Saccoliti, Francesco, Madia, Valentina Noemi, Tudino, Valeria, De Leo, Alessandro, Pescatori, Luca, Messore, Antonella, De Vita, Daniela, Scipione, Luigi, Brun, Reto, Kaiser, Marcel, Maser, Pascal, Calvet, Claudia M., Jennings, Gareth K., Podust, Larissa M., Pepe, Giacomo, Cirilli, Roberto, Faggi, Cristina, Di Marco, Annalise, Battista, Maria Rosaria, Summa, Vincenzo, Costi, Roberta, Di Santo, Roberto
Published in Journal of medicinal chemistry (14.02.2019)
Published in Journal of medicinal chemistry (14.02.2019)
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Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity
Madia, Valentina Noemi, Messore, Antonella, Pescatori, Luca, Saccoliti, Francesco, Tudino, Valeria, De Leo, Alessandro, Bortolami, Martina, Scipione, Luigi, Costi, Roberta, Rivara, Silvia, Scalvini, Laura, Mor, Marco, Ferrara, Fabiana Fosca, Pavoni, Emiliano, Roscilli, Giuseppe, Cassinelli, Giuliana, Milazzo, Ferdinando M, Battistuzzi, Gianfranco, Di Santo, Roberto, Giannini, Giuseppe
Published in Journal of medicinal chemistry (09.08.2018)
Published in Journal of medicinal chemistry (09.08.2018)
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6‑(1-Benzyl‑1H‑pyrrol-2-yl)-2,4-dioxo-5-hexenoic Acids as Dual Inhibitors of Recombinant HIV‑1 Integrase and Ribonuclease H, Synthesized by a Parallel Synthesis Approach
Costi, Roberta, Métifiot, Mathieu, Esposito, Francesca, Cuzzucoli Crucitti, Giuliana, Pescatori, Luca, Messore, Antonella, Scipione, Luigi, Tortorella, Silvano, Zinzula, Luca, Novellino, Ettore, Pommier, Yves, Tramontano, Enzo, Marchand, Christophe, Di Santo, Roberto
Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H
Corona, Angela, di Leva, Francesco Saverio, Rigogliuso, Giuseppe, Pescatori, Luca, Madia, Valentina Noemi, Subra, Frederic, Delelis, Olivier, Esposito, Francesca, Cadeddu, Marta, Costi, Roberta, Cosconati, Sandro, Novellino, Ettore, di Santo, Roberto, Tramontano, Enzo
Published in Antiviral research (01.10.2016)
Published in Antiviral research (01.10.2016)
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In Vitro Antiviral Activity of New Oxazoline Derivatives as Potent Poliovirus Inhibitors
Madia, Valentina Noemi, Messore, Antonella, Pescatori, Luca, Saccoliti, Francesco, Tudino, Valeria, De Leo, Alessandro, Scipione, Luigi, Fiore, Lucia, Rhoden, Eric, Manetti, Fabrizio, Oberste, M. Steven, Di Santo, Roberto, Costi, Roberta
Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
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Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity
Messore, Antonella, Madia, Valentina Noemi, Pescatori, Luca, Saccoliti, Francesco, Tudino, Valeria, De Leo, Alessandro, Bortolami, Martina, De Vita, Daniela, Scipione, Luigi, Pepi, Federico, Costi, Roberta, Rivara, Silvia, Scalvini, Laura, Mor, Marco, Ferrara, Fabiana Fosca, Pavoni, Emiliano, Roscilli, Giuseppe, Cassinelli, Giuliana, Milazzo, Ferdinando M, Battistuzzi, Gianfranco, Di Santo, Roberto, Giannini, Giuseppe
Published in Journal of medicinal chemistry (13.12.2018)
Published in Journal of medicinal chemistry (13.12.2018)
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Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents
Saccoliti, Francesco, Madia, Valentina Noemi, Tudino, Valeria, De Leo, Alessandro, Pescatori, Luca, Messore, Antonella, De Vita, Daniela, Scipione, Luigi, Brun, Reto, Kaiser, Marcel, Mäser, Pascal, Calvet, Claudia M, Jennings, Gareth K, Podust, Larissa M, Pepe, Giacomo, Cirilli, Roberto, Faggi, Cristina, Di Marco, Annalise, Battista, Maria Rosaria, Summa, Vincenzo, Costi, Roberta, Di Santo, Roberto
Published in Journal of medicinal chemistry (14.02.2019)
Published in Journal of medicinal chemistry (14.02.2019)
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Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents
Saccoliti, Francesco, Madia, Valentina Noemi, Tudino, Valeria, De Leo, Alessandro, Pescatori, Luca, Messore, Antonella, De Vita, Daniela, Scipione, Luigi, Brun, Reto, Kaiser, Marcel, Mäser, Pascal, Calvet, Claudia Magalhaes, Jennings, Gareth K., Podust, Larissa M., Costi, Roberta, Di Santo, Roberto
Published in European journal of medicinal chemistry (05.08.2018)
Published in European journal of medicinal chemistry (05.08.2018)
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Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
Costi, Roberta, Métifiot, Mathieu, Chung, Suhman, Cuzzucoli Crucitti, Giuliana, Maddali, Kasthuraiah, Pescatori, Luca, Messore, Antonella, Madia, Valentina Noemi, Pupo, Giovanni, Scipione, Luigi, Tortorella, Silvano, Di Leva, Francesco Saverio, Cosconati, Sandro, Marinelli, Luciana, Novellino, Ettore, Le Grice, Stuart F. J, Corona, Angela, Pommier, Yves, Marchand, Christophe, Di Santo, Roberto
Published in Journal of medicinal chemistry (24.04.2014)
Published in Journal of medicinal chemistry (24.04.2014)
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Journal Article
N‑Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase
Pescatori, Luca, Métifiot, Mathieu, Chung, Suhman, Masoaka, Takashi, Cuzzucoli Crucitti, Giuliana, Messore, Antonella, Pupo, Giovanni, Madia, Valentina Noemi, Saccoliti, Francesco, Scipione, Luigi, Tortorella, Silvano, Di Leva, Francesco Saverio, Cosconati, Sandro, Marinelli, Luciana, Novellino, Ettore, Le Grice, Stuart F. J, Pommier, Yves, Marchand, Christophe, Costi, Roberta, Di Santo, Roberto
Published in Journal of medicinal chemistry (11.06.2015)
Published in Journal of medicinal chemistry (11.06.2015)
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Monotopic and heteroditopic calix[4]arene receptors as hosts for pyridinium and viologen ion pairs: a solution and solid-state study
Pescatori, Luca, Arduini, Arturo, Pochini, Andrea, Secchi, Andrea, Massera, Chiara, Ugozzoli, Franco
Published in Organic & biomolecular chemistry (01.01.2009)
Published in Organic & biomolecular chemistry (01.01.2009)
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Journal Article
Guest Controlled Assembly of Gold Nanoparticles Coated with Calix[4]arene Hosts
Ciesa, Flavio, Plech, Anton, Mattioli, Cristina, Pescatori, Luca, Arduini, Arturo, Pochini, Andrea, Rossi, Francesca, Secchi, Andrea
Published in Journal of physical chemistry. C (19.08.2010)
Published in Journal of physical chemistry. C (19.08.2010)
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Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75
Cuzzucoli Crucitti, Giuliana, Pescatori, Luca, Messore, Antonella, Madia, Valentina Noemi, Pupo, Giovanni, Saccoliti, Francesco, Scipione, Luigi, Tortorella, Silvano, Di Leva, Francesco Saverio, Cosconati, Sandro, Novellino, Ettore, Debyser, Zeger, Christ, Frauke, Costi, Roberta, Di Santo, Roberto
Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
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