Structure-based design, synthesis, and study of pyrazolo[1,5-a][1,3,5]triazine derivatives as potent inhibitors of protein kinase CK2
Nie, Zhe, Perretta, Carin, Erickson, Philip, Margosiak, Stephen, Almassy, Robert, Lu, Jia, Averill, April, Yager, Kraig M., Chu, Shaosong
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
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Identification of (3R)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a Novel Potent and Selective Opioid κ Receptor Antagonist
Thomas, James B, Atkinson, Robert N, Vinson, N. Ariane, Catanzaro, Jennifer L, Perretta, Carin L, Fix, Scott E, Mascarella, S. Wayne, Rothman, Richard B, Xu, Heng, Dersch, Christina M, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F. Ivy
Published in Journal of medicinal chemistry (03.07.2003)
Published in Journal of medicinal chemistry (03.07.2003)
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Structure-based design and synthesis of novel macrocyclic pyrazolo[1,5- a] [1,3,5]triazine compounds as potent inhibitors of protein kinase CK2 and their anticancer activities
Nie, Zhe, Perretta, Carin, Erickson, Philip, Margosiak, Stephen, Lu, Jia, Averill, April, Almassy, Robert, Chu, Shaosong
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Structure-Based Design, Synthesis, and Study of Potent Inhibitors of β-Ketoacyl-acyl Carrier Protein Synthase III as Potential Antimicrobial Agents
Nie, Zhe, Perretta, Carin, Lu, Jia, Su, Ying, Margosiak, Stephen, Gajiwala, Ketan S, Cortez, Joseph, Nikulin, Victor, Yager, Kraig M, Appelt, Krzysztof, Chu, Shaosong
Published in Journal of medicinal chemistry (10.03.2005)
Published in Journal of medicinal chemistry (10.03.2005)
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Synthesis and resolution of the benzomorphan-based kappa opioid agonist bremazocine
Thomas, James B., Brieaddy, Lawrence E., Boldt, Karl G., Perretta, Carin, Carroll, F. Ivy
Published in Synthesis (Stuttgart) (16.05.2007)
Published in Synthesis (Stuttgart) (16.05.2007)
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Identification of (3R)-7-hydroxy-N-((1S)-1-[[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a novel potent and selective opioid kappa receptor antagonist
Thomas, James B, Atkinson, Robert N, Vinson, N Ariane, Catanzaro, Jennifer L, Perretta, Carin L, Fix, Scott E, Mascarella, S Wayne, Rothman, Richard B, Xu, Heng, Dersch, Christina M, Cantrell, Buddy E, Zimmerman, Dennis M, Carroll, F Ivy
Published in Journal of medicinal chemistry (03.07.2003)
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Published in Journal of medicinal chemistry (03.07.2003)
Journal Article
Identification of (3R)-7-hydroxy-N-((1S)-1-{[(3R, 4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidiny l]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide as a novel potent and selective opioid K receptor antagonist
THOMAS, James B, ATKINSON, Robert N, CANTRELL, Buddy E, ZIMMERMAN, Dennis M, CARROLL, F. Ivy, VINSON, N. Ariane, CATANZARO, Jennifer L, PERRETTA, Carin L, FIX, Scott E, MASCARELLA, S. Wayne, ROTHMAN, Richard B, HENG XU, DERSCH, Christina M
Published in Journal of medicinal chemistry (2003)
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Published in Journal of medicinal chemistry (2003)
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