Development of a pharmacophore model for histamine H-3 receptor antagonists, using the newly developed molecular modeling program SLATE
De Esch, IJP, Mills, JEJ, Perkins, TDJ, Romeo, G, Hoffmann, M, Wieland, K, Leurs, R, Menge, WMPB, Nederkoorn, PHJ, Dean, PM, Timmerman, H
Published in Journal of medicinal chemistry (24.05.2001)
Published in Journal of medicinal chemistry (24.05.2001)
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Analysis and optimization of structure-based virtual screening protocols: 2. Examination of docked ligand orientation sampling methodology: mapping a pharmacophore for success
Good, Andrew C., Cheney, Daniel L., Sitkoff, Doree F., Tokarski, John S., Stouch, Terry R., Bassolino, Donna A., Krystek, Stanley R., Li, Yi, Mason, Jonathan S., Perkins, Timothy D.J.
Published in Journal of molecular graphics & modelling (01.09.2003)
Published in Journal of molecular graphics & modelling (01.09.2003)
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Molecular surface-volume and property matching to superpose flexible dissimilar molecules
Perkins, T D, Mills, J E, Dean, P M
Published in Journal of computer-aided molecular design (01.12.1995)
Published in Journal of computer-aided molecular design (01.12.1995)
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New Approach to Molecular Docking and Its Application to Virtual Screening of Chemical Databases
Baxter, Carol A, Murray, Christopher W, Waszkowycz, Bohdan, Li, Jin, Sykes, Richard A, Bone, Richard G. A, Perkins, Tim D. J, Wylie, William
Published in Journal of Chemical Information and Computer Sciences (01.03.2000)
Published in Journal of Chemical Information and Computer Sciences (01.03.2000)
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An automated method for predicting the positions of hydrogen-bonding atoms in binding sites
Mills, J E, Perkins, T D, Dean, P M
Published in Journal of computer-aided molecular design (01.05.1997)
Published in Journal of computer-aided molecular design (01.05.1997)
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Journal Article
Proposed solution structure of endothelin
Perkins, T D, Hider, R C, Barlow, D J
Published in International journal of peptide and protein research (01.08.1990)
Published in International journal of peptide and protein research (01.08.1990)
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