Resorcinol-based hemiindigoid derivatives as human tyrosinase inhibitors and melanogenesis suppressors in human melanoma cells
Roulier, Brayan, Rush, Inbal, Lazinski, Leticia M., Pérès, Basile, Olleik, Hamza, Royal, Guy, Fishman, Ayelet, Maresca, Marc, Haudecoeur, Romain
Published in European journal of medicinal chemistry (15.01.2023)
Published in European journal of medicinal chemistry (15.01.2023)
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Journal Article
Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review
Haudecoeur, Romain, Peuchmaur, Marine, Pérès, Basile, Rome, Maxime, Taïwe, Germain Sotoing, Boumendjel, Ahcène, Boucherle, Benjamin
Published in Journal of ethnopharmacology (15.02.2018)
Published in Journal of ethnopharmacology (15.02.2018)
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Journal Article
Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design
Goracci, Laura, Nurisso, Alessandra, Roussel, Emile, Pérès, Basile, Chaptal, Vincent, Falson, Pierre, Marminon, Christelle, Jose, Joachim, Le Borgne, Marc, Boumendjel, Ahcène
Published in European journal of medicinal chemistry (15.02.2023)
Published in European journal of medicinal chemistry (15.02.2023)
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Journal Article
Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2
Roussel, Emile, Moréno, Alexis, Altounian, Nicolas, Philouze, Christian, Pérès, Basile, Thomas, Aline, Renaudet, Olivier, Falson, Pierre, Boumendjel, Ahcène
Published in European journal of medicinal chemistry (15.09.2020)
Published in European journal of medicinal chemistry (15.09.2020)
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Journal Article
Ferrocene-embedded flavonoids targeting the Achilles heel of multidrug-resistant cancer cells through collateral sensitivity
Pérès, Basile, Nasr, Rachad, Zarioh, Malik, Lecerf-Schmidt, Florine, Di Pietro, Attilio, Baubichon-Cortay, Hélène, Boumendjel, Ahcène
Published in European journal of medicinal chemistry (21.04.2017)
Published in European journal of medicinal chemistry (21.04.2017)
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Journal Article
Substituted Chromones as Highly Potent Nontoxic Inhibitors, Specific for the Breast Cancer Resistance Protein
Valdameri, Glaucio, Genoux-Bastide, Estelle, Peres, Basile, Gauthier, Charlotte, Guitton, Jérôme, Terreux, Raphaël, Winnischofer, Sheila M. B, Rocha, Maria E. M, Boumendjel, Ahcène, Di Pietro, Attilio
Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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Journal Article
Molecular analysis of the massive GSH transport mechanism mediated by the human Multidrug Resistant Protein 1/ABCC1
Nasr, Rachad, Lorendeau, Doriane, Khonkarn, Ruttiros, Dury, Lauriane, Pérès, Basile, Boumendjel, Ahcène, Cortay, Jean-Claude, Falson, Pierre, Chaptal, Vincent, Baubichon-Cortay, Hélène
Published in Scientific reports (06.05.2020)
Published in Scientific reports (06.05.2020)
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Journal Article
Crossing of the Cystic Barriers of Toxoplasma gondii by the Fluorescent Coumarin Tetra-Cyclopeptide
Dard, Céline, Leforestier, Baptiste, Francisco Hilário, Flaviane, Traoré, Mohamed Dit Mady, Lespinasse, Marie-Ange, Pérès, Basile, Molina, Marie-Carmen, Pereira de Freitas, Rossimiriam, Milet, Anne, Maubon, Danièle, Wong, Yung-Sing
Published in Molecules (Basel, Switzerland) (11.12.2021)
Published in Molecules (Basel, Switzerland) (11.12.2021)
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Journal Article
New, highly potent and non-toxic, chromone inhibitors of the human breast cancer resistance protein ABCG2
Pires, Amanda do Rocio Andrade, Lecerf-Schmidt, Florine, Guragossian, Nathalie, Pazinato, Jaqueline, Gozzi, Gustavo Jabor, Winter, Evelyn, Valdameri, Glaucio, Veale, Alexander, Boumendjel, Ahcène, Di Pietro, Attilio, Pérès, Basile
Published in European journal of medicinal chemistry (21.10.2016)
Published in European journal of medicinal chemistry (21.10.2016)
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Journal Article
Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II)
Ettaoussi, Mohamed, Pérès, Basile, Errazani, Aïcha, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (27.01.2015)
Published in European journal of medicinal chemistry (27.01.2015)
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Journal Article
Characterization of Potent ABCG2 Inhibitor Derived from Chromone: From the Mechanism of Inhibition to Human Extracellular Vesicles for Drug Delivery
Valdameri, Glaucio, Kita, Diogo Henrique, Dutra, Julia de Paula, Gomes, Diego Lima, Tonduru, Arun Kumar, Kronenberger, Thales, Gavinho, Bruno, Rossi, Izadora Volpato, Carvalho, Mariana Mazetto de, Pérès, Basile, Zattoni, Ingrid Fatima, Rego, Fabiane Gomes de Moraes, Picheth, Geraldo, Freitas, Rilton Alves de, Poso, Antti, Ambudkar, Suresh V, Ramirez, Marcel I, Boumendjel, Ahcène, Moure, Vivian Rotuno
Published in Pharmaceutics (01.04.2023)
Published in Pharmaceutics (01.04.2023)
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Journal Article
Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens
Olleik, Hamza, Yahiaoui, Samir, Roulier, Brayan, Courvoisier-Dezord, Elise, Perrier, Josette, Pérès, Basile, Hijazi, Akram, Baydoun, Elias, Raymond, Josette, Boumendjel, Ahcène, Maresca, Marc, Haudecoeur, Romain
Published in European journal of medicinal chemistry (01.03.2019)
Published in European journal of medicinal chemistry (01.03.2019)
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Journal Article
Piperidinyl-embeded chalcones possessing anti PI3Kδ inhibitory properties exhibit anti-atopic properties in preclinical models
Dumontet, Charles, Beck, Guillaume, Gardebien, Fabrice, Haudecoeur, Romain, Mathé, Doriane, Matera, Eva-Laure, Tourette, Anne, Mattei, Eve, Esmenjaud, Justine, Boyère, Cédric, Nurisso, Alessandra, Peuchmaur, Marine, Pérès, Basile, Bouchaud, Grégory, Magnan, Antoine, Monneret, Guillaume, Boumendjel, Ahcène
Published in European journal of medicinal chemistry (05.10.2018)
Published in European journal of medicinal chemistry (05.10.2018)
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Journal Article
Design, synthesis and biological evaluation of novel ring-opened cromakalim analogues with relaxant effects on vascular and respiratory smooth muscles and as stimulators of elastin synthesis
Bouhedja, Mourad, Peres, Basile, Fhayli, Wassim, Ghandour, Zeinab, Boumendjel, Ahcène, Faury, Gilles, Khelili, Smail
Published in European journal of medicinal chemistry (20.01.2018)
Published in European journal of medicinal chemistry (20.01.2018)
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Journal Article
Synthesis and Pharmacological Evaluation of a series of the Agomelatine Analogues as Melatonin MT1/MT2 Agonist and 5-HT2C Antagonist
Ettaoussi, Mohamed, Sabaouni, Ahmed, Pérès, Basile, Landagaray, Elodie, Nosjean, Olivier, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in ChemMedChem (01.11.2013)
Published in ChemMedChem (01.11.2013)
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Journal Article
Two Independent Ways of Preparing Hypercharged Hydrolyzable Polyaminorotaxane
Pérès, Basile, Richardeau, Nicolas, Jarroux, Nathalie, Guégan, Philippe, Auvray, Loïc
Published in Biomacromolecules (01.07.2008)
Published in Biomacromolecules (01.07.2008)
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Journal Article
Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT1 melatoninergic ligands
Mésangeau, Christophe, Pérès, Basile, Descamps-François, Carole, Chavatte, Philippe, Audinot, Valérie, Coumailleau, Sophie, Boutin, Jean A., Delagrange, Philippe, Bennejean, Caroline, Renard, Pierre, Caignard, Daniel H., Berthelot, Pascal, Yous, Saïd
Published in Bioorganic & medicinal chemistry (15.05.2010)
Published in Bioorganic & medicinal chemistry (15.05.2010)
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Journal Article
Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2
Roussel, Emile, Tran-Nguyen, Viet-Khoa, Bouhedjar, Khalid, Dems, Mohamed Abdesselem, Belaidi, Amine, Matougui, Brahim, Peres, Basile, Azioune, Ammar, Renaudet, Olivier, Falson, Pierre, Boumendjel, Ahcène
Published in European journal of medicinal chemistry (15.12.2019)
Published in European journal of medicinal chemistry (15.12.2019)
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Journal Article
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT2 melatoninergic ligands
POISSONNIER-DURIEUX, Sophie, ETTAOUSSI, Mohamed, LESIEUR, Daniel, YOUS, Saïd, PERES, Basile, BOUTIN, Jean A, AUDINOT, Valérie, BENNEJEAN, Caroline, DELAGRANGE, Philippe, HENRI CAIGNARD, Daniel, RENARD, Pierre, BERTHELOT, Pascal
Published in Bioorganic & medicinal chemistry (15.09.2008)
Published in Bioorganic & medicinal chemistry (15.09.2008)
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Journal Article