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Published in European journal of pharmacology (10.01.2011)
Published in European journal of pharmacology (10.01.2011)
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Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Affinity, potency, efficacy, and selectivity of neurokinin A analogs at human recombinant NK2 and NK1 receptors
Rupniak, Nadia M J, Perdona, Elisabetta, Griffante, Cristiana, Cavallini, Palmina, Sava, Anna, Ricca, Daniel J, Thor, Karl B, Burgard, Edward C, Corsi, Mauro
Published in PloS one (25.10.2018)
Published in PloS one (25.10.2018)
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Functional and binding kinetic studies make a distinction between OX1 and OX2 orexin receptor antagonists
Faedo, Stefania, Perdonà, Elisabetta, Antolini, Marinella, di Fabio, Romano, Merlo Pich, Emilio, Corsi, Mauro
Published in European journal of pharmacology (05.10.2012)
Published in European journal of pharmacology (05.10.2012)
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In vitro and in vivo characterization of the novel GABA B receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)
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Published in Neuropharmacology (01.10.2011)
Published in Neuropharmacology (01.10.2011)
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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK1 receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)
Perdona', Elisabetta, Costantini, Vivian J A, Tessari, Michela, Martinelli, Prisca, Carignani, Corrado, Valerio, Enzo, Mok, M H Selina, Zonzini, Laura, Visentini, Filippo, Gianotti, Massimo, Gordon, Laurie, Rocheville, Magalie, Corsi, Mauro, Capelli, Anna Maria
Published in Neuropharmacology (01.10.2011)
Published in Neuropharmacology (01.10.2011)
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Azabicyclo[3.1.0]hexane-1-carbohydrazides as Potent and Selective GHSR1a Ligands Presenting a Specific in vivo Behavior
Sabbatini, Fabio Maria, Melotto, Sergio, Bernasconi, Giovanni, Bromidge, Steve M., D'Adamo, Lucilla, Rinaldi, Marilisa, Savoia, Chiara, Mundi, Claudia, Di Francesco, Carla, Zonzini, Laura, Costantini, Vivian J. A., Perini, Benedetta, Valerio, Enzo, Pozzan, Alfonso, Perdonà, Elisabetta, Visentini, Filippo, Corsi, Mauro, Di Fabio, Romano
Published in ChemMedChem (04.11.2011)
Published in ChemMedChem (04.11.2011)
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Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists
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Published in ChemMedChem (03.09.2010)
Published in ChemMedChem (03.09.2010)
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Ciprofloxacin affects conformational equilibria of DNA gyrase A in the presence of magnesium ions
Sissi, Claudia, Perdonà, Elisabetta, Domenici, Enrico, Feriani, Aldo, Howells, Alison J, Maxwell, Anthony, Palumbo, Manlio
Published in Journal of molecular biology (03.08.2001)
Published in Journal of molecular biology (03.08.2001)
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Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systems
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Published in European journal of medicinal chemistry (01.12.2019)
Published in European journal of medicinal chemistry (01.12.2019)
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Potency, efficacy, and selectivity of GR64349 at human recombinant neurokinin NK2 and NK1 receptors
Perdona, Elisabetta, Cavallini, Palmina, Sava, Anna, Griffante, Cristiana, Ricca, Daniel J., Thor, Karl B., Rupniak, Nadia M.J., Corsi, Mauro
Published in Neuroscience letters (15.10.2019)
Published in Neuroscience letters (15.10.2019)
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Letter to the Editor: Backbone 1H, 13C and 15N resonance assignment of the N-terminal 24 kDa fragment of the gyrase B subunit from E. coli
Bellanda, Massimo, Peggion, Evaristo, Otting, Gottfried, Weigelt, Johan, Perdonà, Elisabetta, Domenici, Enrico, Marchioro, Carla, Mammi, Stefano
Published in Journal of biomolecular NMR (01.04.2002)
Published in Journal of biomolecular NMR (01.04.2002)
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In vitro and in vivo characterization of the novel GABA sub(B receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2- p iperidinyl}ethanol (CMPPE))
Perdona', Elisabetta, Costantini, Vivian JA, Tessari, Michela, Martinelli, Prisca, Carignani, Corrado, Valerio, Enzo, Mok, MHSelina, Zonzini, Laura, Visentini, Filippo, Gianotti, Massimo, Gordon, Laurie, Rocheville, Magalie, Corsi, Mauro, Capelli, Anna Maria
Published in Neuropharmacology (01.11.2011)
Published in Neuropharmacology (01.11.2011)
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Evidence that the metabotropic glutamate receptor 5 antagonist MPEP may act as an inhibitor of the norepinephrine transporter in vitro and in vivo
Heidbreder, Christian A., Bianchi, Massimiliano, Lacroix, Laurent P., Faedo, Stefania, Perdona, Elisabetta, Remelli, Rosaria, Cavanni, Paolo, Crespi, Francesco
Published in Synapse (New York, N.Y.) (15.12.2003)
Published in Synapse (New York, N.Y.) (15.12.2003)
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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK sub(1) receptor antagonists
Sabbatini, Fabio M, Di Fabio, Romano, Griffante, Cristiana, Pentassuglia, Giorgio, Zonzini, Laura, Melotto, Sergio, Alvaro, Giuseppe, Capelli, Anna M, Pippo, Lara, Perdona', Elisabetta, St Denis, Yves, Costa, Silvano, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK 1 receptor antagonists
Sabbatini, Fabio M., Fabio, Romano Di, Griffante, Cristiana, Pentassuglia, Giorgio, Zonzini, Laura, Melotto, Sergio, Alvaro, Giuseppe, Capelli, Anna M., Pippo, Lara, Perdona’, Elisabetta, Denis, Yves St, Costa, Silvano, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK(1) receptor antagonists
Sabbatini, Fabio M, Di Fabio, Romano, Griffante, Cristiana, Pentassuglia, Giorgio, Zonzini, Laura, Melotto, Sergio, Alvaro, Giuseppe, Capelli, Anna M, Pippo, Lara, Perdona', Elisabetta, St Denis, Yves, Costa, Silvano, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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