Search Results - "Perdona', Elisabetta" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Novel morpholine scaffolds as selective dopamine (DA) D3 receptor antagonists

Novel morpholine scaffolds as selective dopamine (DA) D3 receptor antagonists

by Micheli, Fabrizio, Cremonesi, Susanna, Semeraro, Teresa, Tarsi, Luca, Tomelleri, Silvia, Cavanni, Paolo, Oliosi, Beatrice, Perdonà, Elisabetta, Sava, Anna, Zonzini, Laura, Feriani, Aldo, Braggio, Simone, Heidbreder, Christian
Published in Bioorganic & medicinal chemistry letters (15.02.2016)

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Affinity, potency, efficacy, and selectivity of neurokinin A analogs at human recombinant NK2 and NK1 receptors

Affinity, potency, efficacy, and selectivity of neurokinin A analogs at human recombinant NK2 and NK1 receptors

by Rupniak, Nadia M J, Perdona, Elisabetta, Griffante, Cristiana, Cavallini, Palmina, Sava, Anna, Ricca, Daniel J, Thor, Karl B, Burgard, Edward C, Corsi, Mauro
Published in PloS one (25.10.2018)

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Distinct receptor subtypes mediate arginine vasopressin-dependent ACTH release and intracellular calcium mobilization in rat pituitary cells

Distinct receptor subtypes mediate arginine vasopressin-dependent ACTH release and intracellular calcium mobilization in rat pituitary cells

by Perdonà, Elisabetta, Arban, Roberto, Griffante, Cristiana
Published in European journal of pharmacology (15.03.2012)

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Functional and binding kinetic studies make a distinction between OX1 and OX2 orexin receptor antagonists

Functional and binding kinetic studies make a distinction between OX1 and OX2 orexin receptor antagonists

by Faedo, Stefania, Perdonà, Elisabetta, Antolini, Marinella, di Fabio, Romano, Merlo Pich, Emilio, Corsi, Mauro
Published in European journal of pharmacology (05.10.2012)

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In vitro and in vivo characterization of the novel GABA B receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)

In vitro and in vivo characterization of the novel GABA B receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)

by Perdona’, Elisabetta, Costantini, Vivian J.A., Tessari, Michela, Martinelli, Prisca, Carignani, Corrado, Valerio, Enzo, Mok, M.H. Selina, Zonzini, Laura, Visentini, Filippo, Gianotti, Massimo, Gordon, Laurie, Rocheville, Magalie, Corsi, Mauro, Capelli, Anna Maria
Published in Neuropharmacology (01.10.2011)

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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK1 receptor antagonists

Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK1 receptor antagonists

by SABBATINI, Fabio M, DI FABIO, Romano, DENIS, Yves St, COSTA, Silvano, CORSI, Mauro, GRIFFANTE, Cristiana, PENTASSUGLIA, Giorgio, ZONZINI, Laura, MELOTTO, Sergio, ALVARO, Giuseppe, CAPELLI, Anna M, PIPPO, Lara, PERDONA, Elisabetta
Published in Bioorganic & medicinal chemistry letters (15.01.2010)

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In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)

In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)

by Perdona', Elisabetta, Costantini, Vivian J A, Tessari, Michela, Martinelli, Prisca, Carignani, Corrado, Valerio, Enzo, Mok, M H Selina, Zonzini, Laura, Visentini, Filippo, Gianotti, Massimo, Gordon, Laurie, Rocheville, Magalie, Corsi, Mauro, Capelli, Anna Maria
Published in Neuropharmacology (01.10.2011)

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Azabicyclo[3.1.0]hexane-1-carbohydrazides as Potent and Selective GHSR1a Ligands Presenting a Specific in vivo Behavior

Azabicyclo[3.1.0]hexane-1-carbohydrazides as Potent and Selective GHSR1a Ligands Presenting a Specific in vivo Behavior

by Sabbatini, Fabio Maria, Melotto, Sergio, Bernasconi, Giovanni, Bromidge, Steve M., D'Adamo, Lucilla, Rinaldi, Marilisa, Savoia, Chiara, Mundi, Claudia, Di Francesco, Carla, Zonzini, Laura, Costantini, Vivian J. A., Perini, Benedetta, Valerio, Enzo, Pozzan, Alfonso, Perdonà, Elisabetta, Visentini, Filippo, Corsi, Mauro, Di Fabio, Romano
Published in ChemMedChem (04.11.2011)

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Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists

Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists

by Sabbatini, Fabio Maria, Di Fabio, Romano, Corsi, Mauro, Cavanni, Paolo, Bromidge, Steve M., St-Denis, Yves, D'Adamo, Lucilla, Contini, Stefania, Rinaldi, Marilisa, Guery, Sebastien, Savoia, Chiara, Mundi, Claudia, Perini, Benedetta, Carpenter, Andrew J., Dal Forno, Giovanna, Faggioni, Federico, Tessari, Michela, Pavone, Francesca, Di Francesco, Carla, Buson, Alberto, Mattioli, Mario, Perdona', Elisabetta, Melotto, Sergio
Published in ChemMedChem (03.09.2010)

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Pharmacological characterization of the ghrelin receptor antagonist, GSK1614343 in rat RC-4B/C cells natively expressing GHS type 1a receptors

Pharmacological characterization of the ghrelin receptor antagonist, GSK1614343 in rat RC-4B/C cells natively expressing GHS type 1a receptors

by Perdonà, Elisabetta, Faggioni, Federico, Buson, Alberto, Sabbatini, Fabio Maria, Corti, Corrado, Corsi, Mauro
Published in European journal of pharmacology (10.01.2011)

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1,2,4-Triazolyl 5‑Azaspiro[2.4]heptanes: Lead Identification and Early Lead Optimization of a New Series of Potent and Selective Dopamine D3 Receptor Antagonists

1,2,4-Triazolyl 5‑Azaspiro[2.4]heptanes: Lead Identification and Early Lead Optimization of a New Series of Potent and Selective Dopamine D3 Receptor Antagonists

by Micheli, Fabrizio, Bacchi, Alessia, Braggio, Simone, Castelletti, Laura, Cavallini, Palmina, Cavanni, Paolo, Cremonesi, Susanna, Dal Cin, Michele, Feriani, Aldo, Gehanne, Sylvie, Kajbaf, Mahmud, Marchió, Luciano, Nola, Selena, Oliosi, Beatrice, Pellacani, Annalisa, Perdonà, Elisabetta, Sava, Anna, Semeraro, Teresa, Tarsi, Luca, Tomelleri, Silvia, Wong, Andrea, Visentini, Filippo, Zonzini, Laura, Heidbreder, Christian
Published in Journal of medicinal chemistry (22.09.2016)

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Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systems

Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systems

by Grillo, Alessandro, Chemi, Giulia, Brogi, Simone, Brindisi, Margherita, Relitti, Nicola, Fezza, Filomena, Fazio, Domenico, Castelletti, Laura, Perdona, Elisabetta, Wong, Andrea, Lamponi, Stefania, Pecorelli, Alessandra, Benedusi, Mascia, Fantacci, Manuela, Valoti, Massimo, Valacchi, Giuseppe, Micheli, Fabrizio, Novellino, Ettore, Campiani, Giuseppe, Butini, Stefania, Maccarrone, Mauro, Gemma, Sandra
Published in European journal of medicinal chemistry (01.12.2019)

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Potency, efficacy, and selectivity of GR64349 at human recombinant neurokinin NK2 and NK1 receptors

Potency, efficacy, and selectivity of GR64349 at human recombinant neurokinin NK2 and NK1 receptors

by Perdona, Elisabetta, Cavallini, Palmina, Sava, Anna, Griffante, Cristiana, Ricca, Daniel J., Thor, Karl B., Rupniak, Nadia M.J., Corsi, Mauro
Published in Neuroscience letters (15.10.2019)

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In vitro and in vivo characterization of the novel GABA sub(B receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2- p iperidinyl}ethanol (CMPPE))

In vitro and in vivo characterization of the novel GABA sub(B receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2- p iperidinyl}ethanol (CMPPE))

by Perdona', Elisabetta, Costantini, Vivian JA, Tessari, Michela, Martinelli, Prisca, Carignani, Corrado, Valerio, Enzo, Mok, MHSelina, Zonzini, Laura, Visentini, Filippo, Gianotti, Massimo, Gordon, Laurie, Rocheville, Magalie, Corsi, Mauro, Capelli, Anna Maria
Published in Neuropharmacology (01.11.2011)

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Evidence that the metabotropic glutamate receptor 5 antagonist MPEP may act as an inhibitor of the norepinephrine transporter in vitro and in vivo

Evidence that the metabotropic glutamate receptor 5 antagonist MPEP may act as an inhibitor of the norepinephrine transporter in vitro and in vivo

by Heidbreder, Christian A., Bianchi, Massimiliano, Lacroix, Laurent P., Faedo, Stefania, Perdona, Elisabetta, Remelli, Rosaria, Cavanni, Paolo, Crespi, Francesco
Published in Synapse (New York, N.Y.) (15.12.2003)

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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK sub(1) receptor antagonists

Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK sub(1) receptor antagonists

by Sabbatini, Fabio M, Di Fabio, Romano, Griffante, Cristiana, Pentassuglia, Giorgio, Zonzini, Laura, Melotto, Sergio, Alvaro, Giuseppe, Capelli, Anna M, Pippo, Lara, Perdona', Elisabetta, St Denis, Yves, Costa, Silvano, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (15.01.2010)

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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK 1 receptor antagonists

Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK 1 receptor antagonists

by Sabbatini, Fabio M., Fabio, Romano Di, Griffante, Cristiana, Pentassuglia, Giorgio, Zonzini, Laura, Melotto, Sergio, Alvaro, Giuseppe, Capelli, Anna M., Pippo, Lara, Perdona’, Elisabetta, Denis, Yves St, Costa, Silvano, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (2010)

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Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK(1) receptor antagonists

Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK(1) receptor antagonists

by Sabbatini, Fabio M, Di Fabio, Romano, Griffante, Cristiana, Pentassuglia, Giorgio, Zonzini, Laura, Melotto, Sergio, Alvaro, Giuseppe, Capelli, Anna M, Pippo, Lara, Perdona', Elisabetta, St Denis, Yves, Costa, Silvano, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (15.01.2010)

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Backbone 1H, 13C and 15N resonance assignment of the N-terminal 24 kDa fragment of the gyrase B subunit from E. coli

Backbone 1H, 13C and 15N resonance assignment of the N-terminal 24 kDa fragment of the gyrase B subunit from E. coli

by Bellanda, Massimo, Peggion, Evaristo, Otting, Gottfried, Weigelt, Johan, Perdona, Elisabetta, Domenici, Enrico, Marchioro, Carla, Mammi, Stefano
Published in Journal of biomolecular NMR (01.04.2002)

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Ciprofloxacin affects conformational equilibria of DNA gyrase A in the presence of magnesium ions

Ciprofloxacin affects conformational equilibria of DNA gyrase A in the presence of magnesium ions

by Sissi, Claudia, Perdonà, Elisabetta, Domenici, Enrico, Feriani, Aldo, Howells, Alison J, Maxwell, Anthony, Palumbo, Manlio
Published in Journal of molecular biology (03.08.2001)

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