New compound sets identified from high throughput phenotypic screening against three kinetoplastid parasites: an open resource
Peña, Imanol, Pilar Manzano, M, Cantizani, Juan, Kessler, Albane, Alonso-Padilla, Julio, Bardera, Ana I, Alvarez, Emilio, Colmenarejo, Gonzalo, Cotillo, Ignacio, Roquero, Irene, de Dios-Anton, Francisco, Barroso, Vanessa, Rodriguez, Ana, Gray, David W, Navarro, Miguel, Kumar, Vinod, Sherstnev, Alexander, Drewry, David H, Brown, James R, Fiandor, Jose M, Julio Martin, J
Published in Scientific reports (05.03.2015)
Published in Scientific reports (05.03.2015)
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Identification of novel bromodomain inhibitors of Trypanosoma cruzi bromodomain factor 2 (TcBDF2) using a fluorescence polarization-based high-throughput assay
Tavernelli, Luis E., Alonso, Victoria L., Peña, Imanol, Rodríguez Araya, Elvio, Manarin, Romina, Cantizani, Juan, Martin, Julio, Salamanca, Juan, Bamborough, Paul, Calderón, Felix, Gabarro, Raquel, Serra, Esteban
Published in Antimicrobial agents and chemotherapy (07.08.2024)
Published in Antimicrobial agents and chemotherapy (07.08.2024)
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Structure-Guided Design and Synthesis of a Pyridazinone Series of Trypanosoma cruzi Proteasome Inhibitors
Thomas, Michael G., McGonagle, Kate, Rowland, Paul, Robinson, David A., Dodd, Peter G., Camino-Díaz, Isabel, Campbell, Lorna, Cantizani, Juan, Castañeda, Pablo, Conn, Daniel, Craggs, Peter D., Edwards, Darren, Ferguson, Liam, Fosberry, Andrew, Frame, Laura, Goswami, Panchali, Hu, Xiao, Korczynska, Justyna, MacLean, Lorna, Martin, Julio, Mutter, Nicole, Osuna-Cabello, Maria, Paterson, Christy, Peña, Imanol, Pinto, Erika G., Pont, Caterina, Riley, Jennifer, Shishikura, Yoko, Simeons, Frederick R. C., Stojanovski, Laste, Thomas, John, Wrobel, Karolina, Young, Robert J., Zmuda, Filip, Zuccotto, Fabio, Read, Kevin D., Gilbert, Ian H., Marco, Maria, Miles, Timothy J., Manzano, Pilar, De Rycker, Manu
Published in Journal of medicinal chemistry (10.08.2023)
Published in Journal of medicinal chemistry (10.08.2023)
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Importance of secondary screening with clinical isolates for anti-leishmania drug discovery
Hefnawy, Aya, Cantizani, Juan, Peña, Imanol, Manzano, Pilar, Rijal, Suman, Dujardin, Jean-Claude, De Muylder, Geraldine, Martin, Julio
Published in Scientific reports (06.08.2018)
Published in Scientific reports (06.08.2018)
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Automated high-content assay for compounds selectively toxic to Trypanosoma cruzi in a myoblastic cell line
Alonso-Padilla, Julio, Cotillo, Ignacio, Presa, Jesús L, Cantizani, Juan, Peña, Imanol, Bardera, Ana I, Martín, Jose J, Rodriguez, Ana
Published in PLoS neglected tropical diseases (01.01.2015)
Published in PLoS neglected tropical diseases (01.01.2015)
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Complex Interplay between Sphingolipid and Sterol Metabolism Revealed by Perturbations to the Leishmania Metabolome Caused by Miltefosine
Armitage, Emily G, Alqaisi, Amjed Q I, Godzien, Joanna, Peña, Imanol, Mbekeani, Alison J, Alonso-Herranz, Vanesa, López-Gonzálvez, Ángeles, Martín, Julio, Gabarro, Raquel, Denny, Paul W, Barrett, Michael P, Barbas, Coral
Published in Antimicrobial agents and chemotherapy (01.05.2018)
Published in Antimicrobial agents and chemotherapy (01.05.2018)
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A Replicative In Vitro Assay for Drug Discovery against Leishmania donovani
Tegazzini, Diana, Díaz, Rosario, Aguilar, Fernando, Peña, Imanol, Presa, Jesús L, Yardley, Vanessa, Martin, Julio J, Coteron, Jose M, Croft, Simon L, Cantizani, Juan
Published in Antimicrobial agents and chemotherapy (01.06.2016)
Published in Antimicrobial agents and chemotherapy (01.06.2016)
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Journal Article
Metabolic Clustering Analysis as a Strategy for Compound Selection in the Drug Discovery Pipeline for Leishmaniasis
Armitage, Emily G, Godzien, Joanna, Peña, Imanol, López-Gonzálvez, Ángeles, Angulo, Santiago, Gradillas, Ana, Alonso-Herranz, Vanesa, Martín, Julio, Fiandor, Jose M, Barrett, Michael P, Gabarro, Raquel, Barbas, Coral
Published in ACS chemical biology (18.05.2018)
Published in ACS chemical biology (18.05.2018)
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Journal Article
Automated High-Content Assay for Compounds Selectively Toxic to Trypanosoma cruzi in a Myoblastic Cell Line: e0003493
Alonso-Padilla, Julio, Cotillo, Ignacio, Presa, Jesús L, Cantizani, Juan, Peña, Imanol, Bardera, Ana I, Martín, Jose J, Rodriguez, Ana
Published in PLoS neglected tropical diseases (01.01.2015)
Published in PLoS neglected tropical diseases (01.01.2015)
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Journal Article
Identification of novel Bromodomain inhibitors of Trypanosoma cruzi Bromodomain Factor 2 (TcBDF2) using a fluorescence polarization-base high-throughput assay
Serra, Esteban Carlos, Tavernelli, Luis, Alonso, Victoria Lucia, Peña, Imanol, Elvio Rodríguez Araya, Manarin, Romina, Cantizani, Juan, Martin, Julio, Salamanca, Juan, Bamborough, Paul, Calderón, Felix, Gabarro, Raquel
Published in bioRxiv (18.02.2024)
Published in bioRxiv (18.02.2024)
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Paper
COMPUESTO DERIVADO DE PIRAZOL PARA TRATAMIENTO O PREVENCIÓN DE LA ENFERMEDAD DE CHAGAS
IGNACIO COTILLO TORREJON, IMANOL PEÑA URQUIZA, RODRIGUEZ ANA, ELBAN MARK, JOSE JULIO MARTIN, JULIO ALONSO PADILLA, ADAM KENNETH CHARNLEY, BETH ANNE KNAPP-REED, ALBANE MARIE KESSLER, TERRY VINCENT HUGHES, LIAN YIQIAN
Year of Publication 01.06.2016
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Year of Publication 01.06.2016
Patent
BENZOTHIAZOLE DERIVATIVE USEFUL IN THE TREATMENT OF CHAGAS DISEASE
MARTIN, JOSE JULIO, CHARNLEY, ADAM KENNETH, COTILLO TORREJON, IGNACIO, KESSLER, ALBANE MARIE, KNAPP-REED, BETH ANNE, PENA URQUIZA, IMANOL, ELBAN, MARK, RODRIGUEZ FERNANDEZ, ANA, LIAN, YIQIAN, HUGHES, TERRY VINCENT, ALONSO PADILLA, JULIO
Year of Publication 14.04.2016
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Year of Publication 14.04.2016
Patent