Advances in high‐throughput mass spectrometry in drug discovery
Dueñas, Maria Emilia, Peltier‐Heap, Rachel E, Leveridge, Melanie, Annan, Roland S, Büttner, Frank H, Trost, Matthias
Published in EMBO molecular medicine (11.01.2023)
Published in EMBO molecular medicine (11.01.2023)
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Journal Article
A high-throughput MALDI-TOF MS biochemical screen for small molecule inhibitors of the antigen aminopeptidase ERAP1
Müller, Leonie, Burton, Amy K, Tayler, Chloe L, Rowedder, James E, Hutchinson, Jonathan P, Peace, Simon, Quayle, Julie M, Leveridge, Melanie V, Annan, Roland S, Trost, Matthias, Peltier-Heap, Rachel E, Dueñas, Maria Emilia
Published in SLAS discovery (01.01.2023)
Published in SLAS discovery (01.01.2023)
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Journal Article
A Matrix-Assisted Laser Desorption/Ionization Time-of-Flight Assay Identifies Nilotinib as an Inhibitor of Inflammation in Acute Myeloid Leukemia
Marín-Rubio, José Luis, Peltier-Heap, Rachel E., Dueñas, Maria Emilia, Heunis, Tiaan, Dannoura, Abeer, Inns, Joseph, Scott, Jonathan, Simpson, A. John, Blair, Helen J., Heidenreich, Olaf, Allan, James M., Watt, Jessica E., Martin, Mathew P., Saxty, Barbara, Trost, Matthias
Published in Journal of medicinal chemistry (22.09.2022)
Published in Journal of medicinal chemistry (22.09.2022)
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Journal Article
A chemoproteomic platform for selective deubiquitinase inhibitor discovery
Cookson, Rosa, Vuorinen, Aini, Pettinger, Jonathan, Kennedy, Cassandra R., Kirkpatrick, Joanna M., Peltier-Heap, Rachel E., Powell, Andrew, Snijders, Ambrosius P., Skehel, Mark, House, David, Rittinger, Katrin, Bush, Jacob T.
Published in Cell reports physical science (18.10.2023)
Published in Cell reports physical science (18.10.2023)
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Journal Article
A chemoproteomic platform for reactive fragment profiling against the deubiquitinases
Cookson, Rosa, Vuorinen, Aini, Pettinger, Jonathan, Kennedy, Cassandra R, Kirkpatrick, Joanna M, Peltier-Heap, Rachel E, Powell, Andrew, Snijders, Ambrosius P, Skehel, Mark, House, David, Rittinger, Katrin, Bush, Jacob T
Published in bioRxiv (03.02.2023)
Published in bioRxiv (03.02.2023)
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