P2-339: Development of a screening platform for the identification of new Rac1/Rac1b inhibitors active in the prevention of amyloid-beta production
Lambeng, Nathalie, Coutadeur, Séverine, Peillon, Hélène, Loiseau, Nadia, Bachelot, Florence, De Oliveira, Catherine, Carton, Rachel, Leblond, Bertr, Beausoleil, Eric, Chauvignac, Cédric, Taverne, Thierry, Schweighoffer, Fabien, Desire, Laurent
Published in Alzheimer's & dementia (01.07.2008)
Published in Alzheimer's & dementia (01.07.2008)
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Journal Article
RAC1 Inhibition Targets Amyloid Precursor Protein Processing by γ-Secretase and Decreases Aβ Production in Vitro and in Vivo
Désiré, Laurent, Bourdin, Jérôme, Loiseau, Nadia, Peillon, Hélène, Picard, Virginie, De Oliveira, Catherine, Bachelot, Florence, Leblond, Bertrand, Taverne, Thierry, Beausoleil, Eric, Lacombe, Sandrine, Drouin, Dominique, Schweighoffer, Fabien
Published in The Journal of biological chemistry (11.11.2005)
Published in The Journal of biological chemistry (11.11.2005)
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Journal Article
Etazolate, a neuroprotective drug linking GABAA receptor pharmacology to amyloid precursor protein processing
Marcade, Maryline, Bourdin, Jérôme, Loiseau, Nadia, Peillon, Hélène, Rayer, Aurélie, Drouin, Dominique, Schweighoffer, Fabien, Désiré, Laurent
Published in Journal of neurochemistry (01.07.2008)
Published in Journal of neurochemistry (01.07.2008)
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Journal Article
Etazolate, a neuroprotective drug linking GABA(A) receptor pharmacology to amyloid precursor protein processing
Marcade, Maryline, Bourdin, Jérôme, Loiseau, Nadia, Peillon, Hélène, Rayer, Aurélie, Drouin, Dominique, Schweighoffer, Fabien, Désiré, Laurent
Published in Journal of neurochemistry (01.07.2008)
Published in Journal of neurochemistry (01.07.2008)
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Journal Article
Structure–activity relationship of isoform selective inhibitors of Rac1/1b GTPase nucleotide binding
Beausoleil, Eric, Chauvignac, Cédric, Taverne, Thierry, Lacombe, Sandrine, Pognante, Laure, Leblond, Bertrand, Pallares, Diego, Oliveira, Catherine De, Bachelot, Florence, Carton, Rachel, Peillon, Hélène, Coutadeur, Séverine, Picard, Virginie, Lambeng, Nathalie, Désiré, Laurent, Schweighoffer, Fabien
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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Journal Article
RAC1 inhibition targets amyloid precursor protein processing by gamma-secretase and decreases Abeta production in vitro and in vivo
Désiré, Laurent, Bourdin, Jérôme, Loiseau, Nadia, Peillon, Hélène, Picard, Virginie, De Oliveira, Catherine, Bachelot, Florence, Leblond, Bertrand, Taverne, Thierry, Beausoleil, Eric, Lacombe, Sandrine, Drouin, Dominique, Schweighoffer, Fabien
Published in The Journal of biological chemistry (11.11.2005)
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Published in The Journal of biological chemistry (11.11.2005)
Journal Article
Rac1b Increases with Progressive Tau Pathology within Cholinergic Nucleus Basalis Neurons in Alzheimer's Disease
Perez, Sylvia E, Getova, Damianka P, He, Bin, Counts, Scott E, Geula, Changiz, Desire, Laurent, Coutadeur, Severine, Peillon, Helene, Ginsberg, Stephen D, Mufson, Elliott J
Published in The American journal of pathology (01.02.2012)
Published in The American journal of pathology (01.02.2012)
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Journal Article
P2-325: EHT0202, an alpha-secretase stimulator active against amyloid-beta accumulation and neurotoxicity that improves attention and cognition
Desire, Laurent, Lambeng, Nathalie, Marcade, Maryline, Peillon, Helene, Rayer, Aurelie, Drouin, Dominique, Schweighoffer, Fabien
Published in Alzheimer's & dementia (01.07.2008)
Published in Alzheimer's & dementia (01.07.2008)
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Journal Article
Etazolate, a neuroprotective drug linking GABAAreceptor pharmacology to amyloid precursor protein processing
Marcade, Maryline, Bourdin, Jerome, Loiseau, Nadia, Peillon, Helene, Rayer, Aurelie, Drouin, Dominique, Schweighoffer, Fabien, Desire, Laurent
Published in Journal of neurochemistry (01.07.2008)
Published in Journal of neurochemistry (01.07.2008)
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Journal Article