On the intrinsic reactivity of highly potent trypanocidal cruzain inhibitors
Bonatto, Vinicius, Batista, Pedro Henrique Jatai, Cianni, Lorenzo, De Vita, Daniela, Silva, Daniel G, Cedron, Rodrigo, Tezuka, Daiane Y, de Albuquerque, Sérgio, Moraes, Carolina Borsoi, Franco, Caio Haddad, Lameira, Jerônimo, Leitão, Andrei, Montanari, Carlos A
Published in MedChemComm (18.11.2020)
Published in MedChemComm (18.11.2020)
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Journal Article
Assessment of the Cruzain Cysteine Protease Reversible and Irreversible Covalent Inhibition Mechanism
Silva, José Rogério A, Cianni, Lorenzo, Araujo, Deborah, Batista, Pedro Henrique Jatai, de Vita, Daniela, Rosini, Fabiana, Leitão, Andrei, Lameira, Jerônimo, Montanari, Carlos A
Published in Journal of chemical information and modeling (23.03.2020)
Published in Journal of chemical information and modeling (23.03.2020)
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Journal Article
Novel selective proline-based peptidomimetics for human cathepsin K inhibition
Cardoso Prado Martins, Felipe, dos Reis Rocho, Fernanda, Bonatto, Vinícius, Jatai Batista, Pedro Henrique, Lameira, Jerônimo, Leitão, Andrei, Montanari, Carlos A.
Published in Bioorganic & medicinal chemistry letters (15.09.2024)
Published in Bioorganic & medicinal chemistry letters (15.09.2024)
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Journal Article
Synthesis and matched molecular pair analysis of covalent reversible inhibitors of the cysteine protease CPB
Matos, Thiago Kelvin Brito, Batista, Pedro Henrique Jatai, dos Reis Rocho, Fernanda, de Vita, Daniela, Pearce, Nicholas, Kellam, Barrie, Montanari, Carlos Alberto, Leitão, Andrei
Published in Bioorganic & medicinal chemistry letters (15.09.2020)
Published in Bioorganic & medicinal chemistry letters (15.09.2020)
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Journal Article
Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement
Gomes, Juliana C., Cianni, Lorenzo, Ribeiro, Jean, dos Reis Rocho, Fernanda, da Costa Martins Silva, Samelyn, Batista, Pedro Henrique Jatai, Moraes, Carolina Borsoi, Franco, Caio Haddad, Freitas-Junior, Lucio H.G., Kenny, Peter W., Leitão, Andrei, Burtoloso, Antonio C.B., de Vita, Daniela, Montanari, Carlos A.
Published in Bioorganic & medicinal chemistry (15.11.2019)
Published in Bioorganic & medicinal chemistry (15.11.2019)
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Journal Article
Synthesis, biochemical evaluation and molecular modeling studies of nonpeptidic nitrile-based fluorinated compounds
Fonseca Lameiro, Rafael da, Shamim, Anwar, Rosini, Fabiana, Cendron, Rodrigo, Jatai Batista, Pedro Henrique, Montanari, Carlos Alberto
Published in Future medicinal chemistry (01.01.2021)
Published in Future medicinal chemistry (01.01.2021)
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Journal Article
TERPENOIDS AND COUMARINS FROM Jatropha ribifolia (Pohl) Baill
Batista, Pedro Henrique Jataí, Andrade, José Roberto M. de, Matos, Taynara Simão, Sousa, Thiciana da Silva, Pinto, Francisco das Chagas L., Silveira, Edilberto Rocha, Loiola, Maria Iracema B., Pessoa, Otilia D. Loiola
Published in Química nova (2014)
Published in Química nova (2014)
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Journal Article
Terpenoides e cumarinas de Jatropha ribifolia (Pohl) Baill
Pedro Henrique Jataí Batista, José Roberto M. de Andrade, Taynara Simão Matos, Thiciana da Silva Sousa, Francisco das Chagas L. Pinto, Edilberto Rocha Silveira, Maria Iracema B. Loiola, Otilia D. Loiola Pessoa
Published in Química Nova (01.07.2014)
Published in Química Nova (01.07.2014)
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Journal Article