Targeting the APP-Mint2 Protein–Protein Interaction with a Peptide-Based Inhibitor Reduces Amyloid‑β Formation
Bartling, Christian R. O, Jensen, Thomas M. T, Henry, Shawna M, Colliander, Anna L, Sereikaite, Vita, Wenzler, Marcella, Jain, Palash, Maric, Hans M, Harpsøe, Kasper, Pedersen, Søren W, Clemmensen, Louise S, Haugaard-Kedström, Linda M, Gloriam, David E, Ho, Angela, Strømgaard, Kristian
Published in Journal of the American Chemical Society (20.01.2021)
Published in Journal of the American Chemical Society (20.01.2021)
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Biochemical investigations of the mechanism of action of small molecules ZL006 and IC87201 as potential inhibitors of the nNOS-PDZ/PSD-95-PDZ interactions
Bach, Anders, Pedersen, Søren W, Dorr, Liam A, Vallon, Gary, Ripoche, Isabelle, Ducki, Sylvie, Lian, Lu-Yun
Published in Scientific reports (16.07.2015)
Published in Scientific reports (16.07.2015)
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Probing backbone hydrogen bonding in PDZ/ligand interactions by protein amide-to-ester mutations
Pedersen, Søren W, Pedersen, Stine B, Anker, Louise, Hultqvist, Greta, Kristensen, Anders S, Jemth, Per, Strømgaard, Kristian
Published in Nature communications (01.01.2014)
Published in Nature communications (01.01.2014)
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Development of a Potent Cyclic Peptide Inhibitor of the nNOS/PSD-95 Interaction
Balboa, Javier R., Essig, Dominik J., Ma, Sana, Karer, Nichlas, Clemmensen, Louise S., Pedersen, Søren W., Joerger, Andreas C., Knapp, Stefan, Østergaard, Søren, Strømgaard, Kristian
Published in Journal of medicinal chemistry (12.01.2023)
Published in Journal of medicinal chemistry (12.01.2023)
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Cell-Permeable and Plasma-Stable Peptidomimetic Inhibitors of the Postsynaptic Density-95/N-Methyl-d-Aspartate Receptor Interaction
Bach, Anders, Eildal, Jonas N. N, Stuhr-Hansen, Nicolai, Deeskamp, Rasmus, Gottschalk, Marie, Pedersen, Søren W, Kristensen, Anders S, Strømgaard, Kristian
Published in Journal of medicinal chemistry (10.03.2011)
Published in Journal of medicinal chemistry (10.03.2011)
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The role of backbone hydrogen bonds in the transition state for protein folding of a PDZ domain
Pedersen, Søren W, Hultqvist, Greta, Strømgaard, Kristian, Jemth, Per
Published in PloS one (01.04.2014)
Published in PloS one (01.04.2014)
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Site-Specific Phosphorylation of PSD-95 PDZ Domains Reveals Fine-Tuned Regulation of Protein–Protein Interactions
Pedersen, Søren W, Albertsen, Louise, Moran, Griffin E, Levesque, Brié, Pedersen, Stine B, Bartels, Lina, Wapenaar, Hannah, Ye, Fei, Zhang, Mingjie, Bowen, Mark E, Strømgaard, Kristian
Published in ACS chemical biology (15.09.2017)
Published in ACS chemical biology (15.09.2017)
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Importance of a Conserved Lys/Arg Residue for Ligand/PDZ Domain Interactions as Examined by Protein Semisynthesis
Pedersen, Søren W., Moran, Griffin E., Sereikaitė, Vita, Haugaard-Kedström, Linda M., Strømgaard, Kristian
Published in Chembiochem : a European journal of chemical biology (17.10.2016)
Published in Chembiochem : a European journal of chemical biology (17.10.2016)
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Ligand binding to the PDZ domains of postsynaptic density protein 95
Toto, Angelo, Pedersen, Søren W., Karlsson, O. Andreas, Moran, Griffin E., Andersson, Eva, Chi, Celestine N., Strømgaard, Kristian, Gianni, Stefano, Jemth, Per
Published in Protein engineering, design and selection (01.05.2016)
Published in Protein engineering, design and selection (01.05.2016)
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Modified Peptides as Potent Inhibitors of the Postsynaptic Density-95/N-Methyl-d-Aspartate Receptor Interaction
Bach, Anders, Chi, Celestine N, Olsen, Thomas B, Pedersen, Søren W, Røder, Martin U, Pang, Gar F, Clausen, Rasmus P, Jemth, Per, Strømgaard, Kristian
Published in Journal of medicinal chemistry (23.10.2008)
Published in Journal of medicinal chemistry (23.10.2008)
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The role of backbone hydrogen bonds in the transition state for protein folding of a PDZ domain
Søren W Pedersen, Greta Hultqvist, Kristian Strømgaard, Per Jemth
Published in PloS one (01.01.2014)
Published in PloS one (01.01.2014)
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