Synthesis of Cytotoxic Indenoisoquinoline Topoisomerase I Poisons
Strumberg, Dirk, Pommier, Yves, Paull, Kenneth, Jayaraman, Muthusamy, Nagafuji, Pamela, Cushman, Mark
Published in Journal of medicinal chemistry (11.02.1999)
Published in Journal of medicinal chemistry (11.02.1999)
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Evaluation of a soluble tetrazolium/formazan assay for cell growth and drug sensitivity in culture using human and other tumor cell lines
SCUDIERO, D. A, SHOEMAKER, R. H, PAULL, K. D, MONKS, A, TIERNEY, S, NOFZIGER, T. H, CURRENS, M. J, SENIFF, D, BOYD, M. R
Published in Cancer research (Chicago, Ill.) (01.09.1988)
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Published in Cancer research (Chicago, Ill.) (01.09.1988)
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Identification of Epidermal Growth Factor Receptor and c-erbB2 Pathway Inhibitors by Correlation With Gene Expression Patterns
Wosikowski, Katja, Schuurhuis, Danita, Johnson, Kathryn, Bates, Susan E., Paull, Kenneth D., Myers, Timothy G., Weinstein, John N.
Published in JNCI : Journal of the National Cancer Institute (15.10.1997)
Published in JNCI : Journal of the National Cancer Institute (15.10.1997)
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Journal Article
Neural Computing in Cancer Drug Development: Predicting Mechanism of Action
Weinstein, John N., Kohn, Kurt W., Grever, Michael R., Viswanadhan, Vellarkad N., Rubinstein, Lawrence V., Monks, Anne P., Scudiero, Dominic A., Welch, Lester, Koutsoukos, Antonis D., Chiausa, August J., Paull, Kenneth D.
Published in Science (American Association for the Advancement of Science) (16.10.1992)
Published in Science (American Association for the Advancement of Science) (16.10.1992)
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Protein-Linked DNA Strand Breaks Induced by NSC 314622, a Novel Noncamptothecin Topoisomerase I Poison
Kohlhagen, G, Paull, K D, Cushman, M, Nagafuji, P, Pommier, Y
Published in Molecular pharmacology (01.07.1998)
Published in Molecular pharmacology (01.07.1998)
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Synthesis and cytotoxicity of 1,6,7,8-substituted 2-(4'-substituted phenyl)-4-quinolones and related compounds: identification as antimitotic agents interacting with tubulin
Kuo, Sheng Chu, Lee, Hong Zin, Juang, Jung Pin, Lin, Yih Tyng, Wu, Tian Shung, Chang, Jer Jang, Lednicer, Dan, Paull, Kenneth D, Lin, Chii M
Published in Journal of medicinal chemistry (30.04.1993)
Published in Journal of medicinal chemistry (30.04.1993)
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Multidrug-resistant phenotype of disease-oriented panels of human tumor cell lines used for anticancer drug screening
LIN WU, SMYTHE, A. M, SHOEMAKER, R. H, STINSON, S. F, MULLENDORE, L. A, MONKS, A, SCUDIERO, D. A, PAULL, K. D, KOUTSOUKOS, A. D, RUBINSTEIN, L. V, BOYD, M. R
Published in Cancer research (Chicago, Ill.) (01.06.1992)
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Published in Cancer research (Chicago, Ill.) (01.06.1992)
Journal Article
Mining and Visualizing Large Anticancer Drug Discovery Databases
Shi, Leming M, Fan, Yi, Lee, Jae K, Waltham, Mark, Andrews, Darren T, Scherf, Uwe, Paull, Kenneth D, Weinstein, John N
Published in Journal of Chemical Information and Computer Sciences (01.03.2000)
Published in Journal of Chemical Information and Computer Sciences (01.03.2000)
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Mining the NCI Anticancer Drug Discovery Databases: Genetic Function Approximation for the QSAR Study of Anticancer Ellipticine Analogues
Shi, Leming M, Fan, Yi, Myers, Timothy G, O'Connor, Patrick M, Paull, Kenneth D, Friend, Stephen H, Weinstein, John N
Published in Journal of Chemical Information and Computer Sciences (01.03.1998)
Published in Journal of Chemical Information and Computer Sciences (01.03.1998)
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Mining the National Cancer Institute Anticancer Drug Discovery Database: Cluster Analysis of Ellipticine Analogs with p53-Inverse and Central Nervous System-Selective Patterns of Activity
Shi, L M, Myers, T G, Fan, Y, O'Connor, P M, Paull, K D, Friend, S H, Weinstein, J N
Published in Molecular pharmacology (01.02.1998)
Published in Molecular pharmacology (01.02.1998)
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Journal Article
Site of action of two novel pyrimidine biosynthesis inhibitors accurately predicted by the COMPARE program
Cleaveland, Emily S., Monks, Anne, Vaigro-Wolff, Anne, Zaharevitz, Daniel W., Paull, Kenneth, Ardalan, Katherine, Cooney, David A., Ford, Harry
Published in Biochemical pharmacology (30.03.1995)
Published in Biochemical pharmacology (30.03.1995)
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Design and Synthesis of Ellipticinium Salts and 1,2-Dihydroellipticines with High Selectivities against Human CNS Cancers in vitro
Jurayj, Jurjus, Haugwitz, Rudiger D, Varma, Ravi K, Paull, Kenneth D, Barrett, John F, Cushman, Mark
Published in Journal of medicinal chemistry (01.07.1994)
Published in Journal of medicinal chemistry (01.07.1994)
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Journal Article
Cytotoxicity of a new IMP dehydrogenase inhibitor, benzamide riboside, to human myelogenous leukemia K562 cells
Jayaram, Hiremagalur N., Gharehbaghi, Kamran, Jayaram, Nagesh H., Rieser, Jason, Krohn, Karsten, Paull, Kenneth D.
Published in Biochemical and biophysical research communications (14.08.1992)
Published in Biochemical and biophysical research communications (14.08.1992)
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Journal Article
Cytotoxicity and characterization of an active metabolite of benzamide riboside, a novel inhibitor of IMP dehydrogenase
Gharehbaghi, K, Paull, K D, Kelley, J A, Barchi, Jr, J J, Marquez, V E, Cooney, D A, Monks, A, Scudiero, D, Krohn, K, Jayaram, H N
Published in International journal of cancer (15.03.1994)
Published in International journal of cancer (15.03.1994)
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Reductase Enzyme Expression Across the National Cancer Institute Tumor Cell Line Panel: Correlation With Sensitivity to Mitomycin C and EO9
Fitzsimmons, Sara A., Workman, Paul, Grever, Michael, Paull, Kenneth, Camalier, Richard, Lewis, Alexander D.
Published in JNCI : Journal of the National Cancer Institute (06.03.1996)
Published in JNCI : Journal of the National Cancer Institute (06.03.1996)
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Feasibility of a high-flux anticancer drug screen using a diverse panel of cultured human tumor cell lines
Monks, A, Scudiero, D, Skehan, P, Shoemaker, R, Paull, K, Vistica, D, Hose, C, Langley, J, Cronise, P, Vaigro-Wolff, A
Published in JNCI : Journal of the National Cancer Institute (05.06.1991)
Published in JNCI : Journal of the National Cancer Institute (05.06.1991)
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