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Published in Clinical and translational science (01.01.2020)
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First-in-Class Pan Caspase Inhibitor Developed for the Treatment of Liver Disease
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Published in Biomedical chromatography (01.02.2007)
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Published in Vaccine (03.09.2014)
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Wang, Haishan, Yu, Niefang, Chen, Dizhong, Lee, Ken Chi Lik, Lye, Pek Ling, Chang, Joyce Wei Wei, Deng, Weiping, Ng, Melvin Chi Yeh, Lu, Ting, Khoo, Mui Ling, Poulsen, Anders, Sangthongpitag, Kanda, Wu, Xiaofeng, Hu, Changyong, Goh, Kee Chuan, Wang, Xukun, Fang, Lijuan, Goh, Kay Lin, Khng, Hwee Hoon, Goh, Siok Kun, Yeo, Pauline, Liu, Xin, Bonday, Zahid, Wood, Jeanette M, Dymock, Brian W, Kantharaj, Ethirajulu, Sun, Eric T
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Published in Journal of medicinal chemistry (14.07.2011)
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SB939, a novel potent and orally active histone deacetylase inhibitor with high tumor exposure and efficacy in mouse models of colorectal cancer
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Published in Molecular cancer therapeutics (01.03.2010)
Published in Molecular cancer therapeutics (01.03.2010)
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First-in-human phase 1 study of ETC-159 an oral PORCN inhbitor in patients with advanced solid tumours
Ng, Matthew, Tan, David SP, Subbiah, Vivek, Weekes, Colin D., Teneggi, Vincenzo, Diermayr, Veronica, Ethirajulu, Kantharaj, Yeo, Pauline, Chen, Deborah, Blanchard, Stephanie, Nellore, Ranjani, Gan, Bong Hwa, Yasin, Maryam, Lee, Lay Hoon, Lee, May Ann, Hill, Jeffrey, Madan, Babita, Virshup, David, Matter, Alex
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Preclinical Metabolism and Disposition of SB939 (Pracinostat), an Orally Active Histone Deacetylase Inhibitor, and Prediction of Human Pharmacokinetics
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Published in Drug metabolism and disposition (01.12.2011)
Published in Drug metabolism and disposition (01.12.2011)
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Yeo, Pauline, Venkatesh, P., Goh, Evelyn, Zeng, Peizi, New, Lee S., Hu, Changyong, Sangthongpitag, Kanda, William, Anthony D., Goh, Kee C., Wood, Jeanette M., Kantharaj, Ethirajulu
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Published in Blood (16.11.2007)
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Preclinical metabolism and pharmacokinetics of SB1317 (TG02), a potent CDK/JAK2/FLT3 inhibitor
Pasha, Mohammed Khalid, Jayaraman, Ramesh, Reddy, Venkatesh Pilla, Yeo, Pauline, Goh, Evelyn, Williams, Anthony, Goh, Kee Chuan, Kantharaj, Ethirajulu
Published in Drug metabolism letters (01.03.2012)
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Published in Drug metabolism letters (01.03.2012)
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Pharmacodynamic evaluation of AUM001/tinodasertib, an oral inhibitor of mitogen-activated protein kinase (MAPK)-interacting protein kinase 1, 2 (MNK1/2) in preclinical models and tissues from a Phase 1 clinical study
Gan, Bong Hwa, Lee, Lay Hoon, Takeda, Reika, Yasin, Maryam, Teneggi, Vincenzo, Ethirajulu, Kantharaj, Yeo, Pauline, Umrani, Dhananjay, Pendharkar, Vishal, Darren Wen Teck Lim, Li, Greg, Lu, Qingshu, Cao, Yang, Nellore, Ranjani, Blanchard, Stephanie, Hentze, Hannes, Novotny-Diermayr, Veronica
Published in bioRxiv (29.02.2024)
Published in bioRxiv (29.02.2024)
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Oxidation/reduction chemistry of thiol groups in biological molecules
Rabenstein, Dallas L., Yeo, Pauline, Millis, Kevin K., Keire, David A.
Published in Journal of inorganic biochemistry (01.07.1993)
Published in Journal of inorganic biochemistry (01.07.1993)
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