Thermal Stability Assessment of Peptide Coupling Reagents Commonly Used in Pharmaceutical Manufacturing
Sperry, Jeffrey B, Minteer, Christopher J, Tao, JingYa, Johnson, Rebecca, Duzguner, Remzi, Hawksworth, Michael, Oke, Samantha, Richardson, Paul F, Barnhart, Richard, Bill, David R, Giusto, Robert A
Published in Organic process research & development (21.09.2018)
Published in Organic process research & development (21.09.2018)
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Journal Article
Design of Potent and Selective Inhibitors to Overcome Clinical Anaplastic Lymphoma Kinase Mutations Resistant to Crizotinib
Huang, Qinhua, Johnson, Ted W, Bailey, Simon, Brooun, Alexei, Bunker, Kevin D, Burke, Benjamin J, Collins, Michael R, Cook, Andrew S, Cui, J. Jean, Dack, Kevin N, Deal, Judith G, Deng, Ya-Li, Dinh, Dac, Engstrom, Lars D, He, Mingying, Hoffman, Jacqui, Hoffman, Robert L, Johnson, Patrick S, Kania, Robert S, Lam, Hieu, Lam, Justine L, Le, Phuong T, Li, Qiuhua, Lingardo, Laura, Liu, Wei, Lu, Melissa West, McTigue, Michele, Palmer, Cynthia L, Richardson, Paul F, Sach, Neal W, Shen, Hong, Smeal, Tod, Smith, Graham L, Stewart, Albert E, Timofeevski, Sergei, Tsaparikos, Konstantinos, Wang, Hui, Zhu, Huichun, Zhu, Jinjiang, Zou, Helen Y, Edwards, Martin P
Published in Journal of medicinal chemistry (27.02.2014)
Published in Journal of medicinal chemistry (27.02.2014)
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Journal Article
Scalable Synthesis of 1-Bicyclo[1.1.1]pentylamine via a Hydrohydrazination Reaction
Bunker, Kevin D, Sach, Neal W, Huang, Qinhua, Richardson, Paul F
Published in Organic letters (02.09.2011)
Published in Organic letters (02.09.2011)
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Discovery of (10R)-7-Amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2H-8,4-(metheno)pyrazolo[4,3-h][2,5,11]-benzoxadiazacyclotetradecine-3-carbonitrile (PF-06463922), a Macrocyclic Inhibitor of Anaplastic Lymphoma Kinase (ALK) and c-ros Oncogene 1 (ROS1) with Preclinical Brain Exposure and Broad-Spectrum Potency against ALK-Resistant Mutations
Johnson, Ted W., Richardson, Paul F., Bailey, Simon, Brooun, Alexei, Burke, Benjamin J., Collins, Michael R., Cui, J. Jean, Deal, Judith G., Deng, Ya-Li, Dinh, Dac, Engstrom, Lars D., He, Mingying, Hoffman, Jacqui, Hoffman, Robert L., Huang, Qinhua, Kania, Robert S., Kath, John C., Lam, Hieu, Lam, Justine L., Le, Phuong T., Lingardo, Laura, Liu, Wei, McTigue, Michele, Palmer, Cynthia L., Sach, Neal W., Smeal, Tod, Smith, Graham L., Stewart, Albert E., Timofeevski, Sergei, Zhu, Huichun, Zhu, Jinjiang, Zou, Helen Y., Edwards, Martin P.
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
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Journal Article
Practical Singly and Doubly Electrophilic Aminating Agents: A New, More Sustainable Platform for Carbon–Nitrogen Bond Formation
Kattamuri, Padmanabha V, Yin, Jun, Siriwongsup, Surached, Kwon, Doo-Hyun, Ess, Daniel H, Li, Qun, Li, Guigen, Yousufuddin, Muhammed, Richardson, Paul F, Sutton, Scott C, Kürti, László
Published in Journal of the American Chemical Society (16.08.2017)
Published in Journal of the American Chemical Society (16.08.2017)
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Journal Article
Conformational Studies and Atropisomerism Kinetics of the ALK Clinical Candidate Lorlatinib (PF-06463922) and Desmethyl Congeners
Elleraas, Jeff, Ewanicki, Jason, Johnson, Ted W., Sach, Neal W., Collins, Michael R., Richardson, Paul F.
Published in Angewandte Chemie (International ed.) (07.03.2016)
Published in Angewandte Chemie (International ed.) (07.03.2016)
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Journal Article
Discovery of N-X anomeric amides as electrophilic halogenation reagents
Wang, Yu, Bi, Cheng, Kawamata, Yu, Grant, Lauren N, Samp, Lacey, Richardson, Paul F, Zhang, Shasha, Harper, Kaid C, Palkowitz, Maximilian D, Vasilopoulos, Aristidis, Collins, Michael R, Oderinde, Martins S, Tyrol, Chet C, Chen, Doris, LaChapelle, Erik A, Bailey, Jake B, Qiao, Jennifer X, Baran, Phil S
Published in Nature chemistry (01.09.2024)
Published in Nature chemistry (01.09.2024)
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Mechanistic Study of Enantioselective Pd-Catalyzed C(sp3)–H Activation of Thioethers Involving Two Distinct Stereomodels
Saint-Denis, Tyler G, Lam, Nelson Y. S, Chekshin, Nikita, Richardson, Paul F, Chen, Jason S, Elleraas, Jeff, Hesp, Kevin D, Schmitt, Daniel C, Lian, Yajing, Huh, Chan Woo, Yu, Jin-Quan
Published in ACS catalysis (06.08.2021)
Published in ACS catalysis (06.08.2021)
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Journal Article
Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer
Sharma, Shikhar, Chung, Chi-Yeh, Uryu, Sean, Petrovic, Jelena, Cao, Joan, Rickard, Amanda, Nady, Nataliya, Greasley, Samantha, Johnson, Eric, Brodsky, Oleg, Khan, Showkhin, Wang, Hui, Wang, Zhenxiong, Zhang, Yong, Tsaparikos, Konstantinos, Chen, Lei, Mazurek, Anthony, Lapek, John, Kung, Pei-Pei, Sutton, Scott, Richardson, Paul F., Greenwald, Eric C., Yamazaki, Shinji, Jones, Rhys, Maegley, Karen A., Bingham, Patrick, Lam, Hieu, Stupple, Alexandra E., Kamal, Aileen, Chueh, Anderly, Cuzzupe, Anthony, Morrow, Benjamin J., Ren, Bin, Carrasco-Pozo, Catalina, Tan, Chin Wee, Bhuva, Dharmesh D., Allan, Elizabeth, Surgenor, Elliot, Vaillant, François, Pehlivanoglu, Havva, Falk, Hendrik, Whittle, James R., Newman, Janet, Cursons, Joseph, Doherty, Judy P., White, Karen L., MacPherson, Laura, Devlin, Mark, Dennis, Matthew L., Hattarki, Meghan K., De Silva, Melanie, Camerino, Michelle A., Butler, Miriam S., Dolezal, Olan, Pilling, Patricia, Foitzik, Richard, Stupple, Paul A., Lagiakos, H. Rachel, Walker, Scott R., Hediyeh-Zadeh, Soroor, Nuttall, Stewart, Spall, Sukhdeep K., Charman, Susan A., Connor, Theresa, Peat, Thomas S., Avery, Vicky M., Bozikis, Ylva E., Yang, Yuqing, Zhang, Ming, Monahan, Brendon J., Voss, Anne K., Thomas, Tim, Street, Ian P., Dawson, Sarah-Jane, Dawson, Mark A., Lindeman, Geoffrey J., Davis, Melissa J., Visvader, Jane E., Paul, Thomas A.
Published in Cell chemical biology (19.10.2023)
Published in Cell chemical biology (19.10.2023)
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Journal Article
Some Items of Interest to Process R&D Chemists and Engineers
Richardson, Paul F, Steven, Alan, Kargbo, Robert B, Mateos, Carlos, Zlota, Andrei A, Nawrat, Christopher C, Phelan, James P, Knight, John
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
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Journal Article
Some Items of Interest to Process R&D Chemists and Engineers
Richardson, Paul F, Steven, Alan, Kargbo, Robert B, Mateos, Carlos, Zlota, Andrei A, Nawrat, Christopher C, Ramirez, Antonio, Knight, John
Published in Organic process research & development (21.01.2022)
Published in Organic process research & development (21.01.2022)
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Journal Article
Some Items of Interest to Process R&D Chemists and Engineers
Richardson, Paul F, Steven, Alan, Kargbo, Robert B, Mateos, Carlos, Zlota, Andrei A, Nawrat, Christopher C, Phelan, James P, Knight, John
Published in Organic process research & development (19.11.2021)
Published in Organic process research & development (19.11.2021)
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Journal Article
Some Items of Interest to Process R&D Chemists and Engineers
Richardson, Paul F, Steven, Alan, Kargbo, Robert B, Mateos, Carlos, Zlota, Andrei A, Nawrat, Christopher C, Matcha, Kiran, Ramirez, Antonio, Knight, John
Published in Organic process research & development (17.09.2021)
Published in Organic process research & development (17.09.2021)
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Journal Article
Some Items of Interest to Process R&D Chemists and Engineers
Richardson, Paul F, Steven, Alan, Kargbo, Robert B, Mateos, Carlos, Zlota, Andrei A, Kelly, Christopher B, Zhao, Wenyi, Nawrat, Christopher C, Matcha, Kiran, Knight, John
Published in Organic process research & development (16.07.2021)
Published in Organic process research & development (16.07.2021)
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Correction to “Practical Singly and Doubly Electrophilic Aminating Agents: A New, More Sustainable Platform for Carbon–Nitrogen Bond Formation”
Kattamuri, Padmanabha V, Yin, Jun, Siriwongsup, Surached, Kwon, Doo-Hyun, Ess, Daniel H, Li, Qun, Li, Guigen, Yousufuddin, Muhammed, Richardson, Paul F, Sutton, Scott C, Kürti, László
Published in Journal of the American Chemical Society (20.02.2019)
Published in Journal of the American Chemical Society (20.02.2019)
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Cu-Catalyzed Hydroboration of Benzylidenecyclopropanes: Reaction Optimization, (Hetero)Aryl Scope, and Origins of Pathway Selectivity
Medina, Jose M, Kang, Taeho, Erbay, Tuğçe G, Shao, Huiling, Gallego, Gary M, Yang, Shouliang, Tran-Dubé, Michelle, Richardson, Paul F, Derosa, Joseph, Helsel, Ryan T, Patman, Ryan L, Wang, Fen, Ashcroft, Christopher P, Braganza, John F, McAlpine, Indrawan, Liu, Peng, Engle, Keary M
Published in ACS catalysis (06.12.2019)
Published in ACS catalysis (06.12.2019)
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Green Chemistry Articles of Interest to the Pharmaceutical Industry
Bryan, Marian C, Dalton, Charlotte, Díaz-Rodríguez, Alba, Doerfler, Jaika, Engl, Oliver D, Ferguson, Paul, Molina, Alejandro Gimenez, Han, Zhengxu S, Hosford, Joseph, Howell, Gareth P, Hutchby, Marc, Li, Wei, Munday, Rachel H, Navarro, Antonio, Parmentier, Michael, Pawlas, Jan, Richardson, Paul F, Smith, William J, Steven, Alan, Takale, Balaram S, Terrett, Jack A, Treitler, Daniel S, Zeng, Mingshuo
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
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Journal Article
Design, Synthesis, and Evaluation of NO-Donor Containing Carbonic Anhydrase Inhibitors To Lower Intraocular Pressure
Huang, Qinhua, Rui, Eugene Y, Cobbs, Morena, Dinh, Dac M, Gukasyan, Hovhannes J, Lafontaine, Jennifer A, Mehta, Saurabh, Patterson, Brian D, Rewolinski, David A, Richardson, Paul F, Edwards, Martin P
Published in Journal of medicinal chemistry (26.03.2015)
Published in Journal of medicinal chemistry (26.03.2015)
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