Asymmetric 1,4-Reductions of Hindered β-Substituted Cycloalkenones Using Catalytic SEGPHOS−Ligated CuH
Lipshutz, Bruce H, Servesko, Jeff M, Petersen, Tue B, Papa, Patrick P, Lover, Andrew A
Published in Organic letters (15.04.2004)
Published in Organic letters (15.04.2004)
Get full text
Journal Article
Discovery and optimization of thieno[2,3-d]pyrimidines as B-Raf inhibitors
Packard, Garrick K., Papa, Patrick, Riggs, Jennifer R., Erdman, Paul, Tehrani, Lida, Robinson, Dale, Harris, Roy, Shevlin, Graziella, Perrin-Ninkovic, Sophie, Hilgraf, Robert, McCarrick, Margaret A., Tran, Tam, Fleming, Yuedi, Bai, April, Richardson, Samantha, Katz, Jason, Tang, Yang, Leisten, Jim, Moghaddam, Mehran, Cathers, Brian, Zhu, Dan, Sakata, Steven
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Get full text
Journal Article
A convenient, efficient method for conjugate reductions using catalytic quantities of Cu(I)
Lipshutz, Bruce H., Keith, John, Papa, Patrick, Vivian, Randall
Published in Tetrahedron letters (25.06.1998)
Published in Tetrahedron letters (25.06.1998)
Get full text
Journal Article
Design and Synthesis of Novel Cereblon Binders for Use in Targeted Protein Degradation
Norris, Stephen, Ba, Xiaochu, Rhodes, Jayce, Huang, Dehua, Khambatta, Gody, Buenviaje, Jennifer, Nayak, Surendra, Meiring, Joseph, Reiss, Samantha, Xu, Shuichan, Shi, Lihong, Whitefield, Brandon, Alexander, Matt, Horn, Evan J., Correa, Matthew, Tehrani, Lida, Hansen, Joshua D., Papa, Patrick, Mortensen, Deborah S.
Published in Journal of medicinal chemistry (14.12.2023)
Published in Journal of medicinal chemistry (14.12.2023)
Get full text
Journal Article
Correction to “Design and Synthesis of Novel Cereblon Binders for Use in Targeted Protein Degradation”
Norris, Stephen, Ba, Xiaochu, Rhodes, Jayce, Huang, Dehua, Khambatta, Gody, Buenviaje, Jennifer, Nayak, Surendra, Meiring, Joseph, Reiss, Samantha, Xu, Shuichan, Shi, Lihong, Whitefield, Brandon, Alexander, Matt, Horn, Evan J., Correa, Matthew, Tehrani, Lida, Hansen, Joshua D., Papa, Patrick, Mortensen, Deborah S., Brazeau, Jean-François
Published in Journal of medicinal chemistry (22.08.2024)
Published in Journal of medicinal chemistry (22.08.2024)
Get full text
Journal Article
Discovery of the Selective Protein Kinase C-theta Kinase Inhibitor, CC-90005
Papa, Patrick, Whitefield, Brandon, Mortensen, Deborah S., Cashion, Dan, Huang, Dehua, Torres, Eduardo, Parnes, Jason, Sapienza, John, Hansen, Joshua, Correa, Matthew, Delgado, Mercedes, Harris, Roy, Hegde, Sayee, Norris, Stephen, Bahmanyar, Sogole, Plantevin-Krenitsky, Veronique, Liu, Zheng, Leftheris, Katerina, Kulkarni, Ashutosh, Bennett, Brydon, Hur, Eun Mi, Ringheim, Garth, Khambatta, Godrej, Chan, Henry, Muir, Jeffrey, Blease, Kate, Burnett, Kelven, LeBrun, Laurie, Morrison, Lisa, Celeridad, Maria, Khattri, Roli, Cathers, Brian E.
Published in Journal of medicinal chemistry (26.08.2021)
Published in Journal of medicinal chemistry (26.08.2021)
Get full text
Journal Article
Optimization of a Series of Triazole Containing Mammalian Target of Rapamycin (mTOR) Kinase Inhibitors and the Discovery of CC-115
Mortensen, Deborah S., Perrin-Ninkovic, Sophie M., Shevlin, Graziella, Elsner, Jan, Zhao, Jingjing, Whitefield, Brandon, Tehrani, Lida, Sapienza, John, Riggs, Jennifer R., Parnes, Jason S., Papa, Patrick, Packard, Garrick, Lee, Branden G.S., Harris, Roy, Correa, Matthew, Bahmanyar, Sogole, Richardson, Samantha J., Peng, Sophie X., Leisten, Jim, Khambatta, Godrej, Hickman, Matt, Gamez, James C., Bisonette, René R., Apuy, Julius, Cathers, Brian E., Canan, Stacie S., Moghaddam, Mehran F., Raymon, Heather K., Worland, Peter, Narla, Rama Krishna, Fultz, Kimberly E., Sankar, Sabita
Published in Journal of medicinal chemistry (23.07.2015)
Published in Journal of medicinal chemistry (23.07.2015)
Get full text
Journal Article
Triisopropylsilyloxycarbonyl (“Tsoc”): A New Protecting Group for 1° and 2° Amines
Lipshutz, Bruce H, Papa, Patrick, Keith, John M
Published in Journal of organic chemistry (28.05.1999)
Published in Journal of organic chemistry (28.05.1999)
Get full text
Journal Article
Discovery of Mammalian Target of Rapamycin (mTOR) Kinase Inhibitor CC-223
Mortensen, Deborah S, Perrin-Ninkovic, Sophie M, Shevlin, Graziella, Zhao, Jingjing, Packard, Garrick, Bahmanyar, Sogole, Correa, Matthew, Elsner, Jan, Harris, Roy, Lee, Branden G. S, Papa, Patrick, Parnes, Jason S, Riggs, Jennifer R, Sapienza, John, Tehrani, Lida, Whitefield, Brandon, Apuy, Julius, Bisonette, René R, Gamez, James C, Hickman, Matt, Khambatta, Godrej, Leisten, Jim, Peng, Sophie X, Richardson, Samantha J, Cathers, Brian E, Canan, Stacie S, Moghaddam, Mehran F, Raymon, Heather K, Worland, Peter, Narla, Rama Krishna, Fultz, Kimberly E, Sankar, Sabita
Published in Journal of medicinal chemistry (09.07.2015)
Published in Journal of medicinal chemistry (09.07.2015)
Get full text
Journal Article
Copper Hydride- Catalyzed Tandem 1,4-Reduction/Alkylation Reactions
Lipshutz, Bruce H., Chrisman, Will, Noson, Kevin, Papa, Patrick, Sclafani, Joseph A., Vivian, Randall W., Keith, John M.
Published in Tetrahedron (28.04.2000)
Published in Tetrahedron (28.04.2000)
Get full text
Journal Article
mTOR KINASE INHIBITOR FOR ONCOLOGICAL BEHAVIORS AND DISEASES RELATED TO mTOR/PI3K/AKT PATHWAY
JINGJING ZHAO, JAN ELSNER, JOHN SAPIENZA, DEBORAH MORTENSEN, SABITA SANKAR, RAMA K NARLA, LIDA TEHRANI, KIMBERLY FULTZ, SOPHIE PERRIN-NINKOVIC, JASON PARNES, GARRICK PACKARD, PATRICK PAPA, BRANDEN LEE, XU WEIMING, GRAZIELLA SHEVLIN, ROY L HARRIS, JENNIFER RIGGS, LOUI MADAKAMUTIL
Year of Publication 19.01.2017
Get full text
Year of Publication 19.01.2017
Patent
A Novel mTOR Kinase Inhibitor Causes Growth Inhibition, Cell Cycle Arrest, Apoptosis and Autophagic Cell Death in Mantle Cell Lymphoma Cell Lines: A Distinct Profile from Rapamycin
Xu, Weiming, Kang, Christine, Delgado, Mercedes, Perrin-Ninkovic, Sophie M, Papa, Patrick W, Riggs, Jennifer R, Sapienza, John, Albers, Ronald J, Lee, Branden G.S, Harris, Roy L, Mortensen, Deborah S, Worland, Peter, Sankar, Sabita
Published in Blood (16.11.2008)
Published in Blood (16.11.2008)
Get full text
Journal Article
METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS
ZHAO JINGJING, ANUSUYA CHOUDHURY, JAN ELSNER, DEBORAH MORTENSEN, MOHIT ATUL KOTHARE, BRANDEN GINGSEE LEE, SOPHIE PERRIN-NINKOVIC, SAPIENZA JOHN, GARRICK PACKARD, JUAN ANTONIO GAMBOA, WILLIAM WEI-HWA LEONG, MATTHEW MICHAEL KREILEIN, BEAUCHAMPS MARIE GEORGES, PATRICK ANTHONY JOKIEL, PHILIP PYE, PATRICK PAPA, GRAZIELLA SHEVLIN, ROY L HARRIS, JENNIFER RIGGS
Year of Publication 19.01.2017
Get full text
Year of Publication 19.01.2017
Patent
mTOR KINASE INHIBITOR FOR ONCOLOGICAL SYMPTOM AND DISEASE RELATED TO mTOR/PI3K/AKT PATHWAY
JINGJING ZHAO, JAN ELSNER, JOHN SAPIENZA, DEBORAH MORTENSEN, SABITA SANKAR, RAMA K NARLA, LIDA TEHRANI, KIMBERLY FULTZ, SOPHIE PERRIN-NINKOVIC, JASON PARNES, GARRICK PACKARD, PATRICK PAPA, BRANDEN LEE, XU WEIMING, GRAZIELLA SHEVLIN, ROY L HARRIS, JENNIFER RIGGS, LOUI MADAKAMUTIL
Year of Publication 14.05.2015
Get full text
Year of Publication 14.05.2015
Patent