The role of lysine palmitoylation/myristoylation in the function of the TEAD transcription factors
Mesrouze, Yannick, Aguilar, Gustavo, Meyerhofer, Marco, Bokhovchuk, Fedir, Zimmermann, Catherine, Fontana, Patrizia, Vissières, Alexandra, Voshol, Hans, Erdmann, Dirk, Affolter, Markus, Chène, Patrick
Published in Scientific reports (23.03.2022)
Published in Scientific reports (23.03.2022)
Get full text
Journal Article
Dissection of the interaction between the intrinsically disordered YAP protein and the transcription factor TEAD
Mesrouze, Yannick, Bokhovchuk, Fedir, Meyerhofer, Marco, Fontana, Patrizia, Zimmermann, Catherine, Martin, Typhaine, Delaunay, Clara, Erdmann, Dirk, Schmelzle, Tobias, Chène, Patrick
Published in eLife (21.04.2017)
Published in eLife (21.04.2017)
Get full text
Journal Article
N‐terminal β‐strand in YAP is critical for stronger binding to scalloped relative to TEAD transcription factor
Fedir, Bokhovchuk, Yannick, Mesrouze, Marco, Meyerhofer, Patrizia, Fontana, Catherine, Zimmermann, Frédéric, Villard, Dirk, Erdmann, Joerg, Kallen, Clemens, Scheufler, Camilo, Velez‐Vega, Patrick, Chène
Published in Protein science (01.01.2023)
Published in Protein science (01.01.2023)
Get full text
Journal Article
Biochemical and Structural Characterization of a Peptidic Inhibitor of the YAP:TEAD Interaction That Binds to the α‑Helix Pocket on TEAD
Mesrouze, Yannick, Gubler, Hanspeter, Villard, Frédéric, Boesch, Ralf, Ottl, Johannes, Kallen, Joerg, Reid, Patrick C., Scheufler, Clemens, Marzinzik, Andreas L., Chène, Patrick
Published in ACS chemical biology (17.03.2023)
Published in ACS chemical biology (17.03.2023)
Get full text
Journal Article
Abstract 1239: NVP-HDM201: Biochemical and biophysical profile of a novel highly potent and selective PPI inhibitor of p53-Mdm2
Stachyra-Valat, Thérèse, Baysang, Frédéric, D’Alessandro, Anne-Cécile, Dirk, Erdmann, Furet, Pascal, Guagnano, Vito, Kallen, Joerg, Leder, Lukas, Mah, Robert, Masuya, Keiichi, Stutz, Stefan, Vaupel, Andrea, Hofmann, Francesco, Chène, Patrick, Jeay, Sébastien, Holzer, Philipp
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Get full text
Journal Article
Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors
Holzer, Philipp, Masuya, Keiichi, Furet, Pascal, Kallen, Joerg, Valat-Stachyra, Therese, Ferretti, Stéphane, Berghausen, Joerg, Bouisset-Leonard, Michèle, Buschmann, Nicole, Pissot-Soldermann, Carole, Rynn, Caroline, Ruetz, Stephan, Stutz, Stefan, Chène, Patrick, Jeay, Sébastien, Gessier, Francois
Published in Journal of medicinal chemistry (27.08.2015)
Published in Journal of medicinal chemistry (27.08.2015)
Get full text
Journal Article
An Early Association between the α‑Helix of the TEAD Binding Domain of YAP and TEAD Drives the Formation of the YAP:TEAD Complex
Bokhovchuk, Fedir, Mesrouze, Yannick, Meyerhofer, Marco, Zimmermann, Catherine, Fontana, Patrizia, Erdmann, Dirk, Jemth, Per, Chène, Patrick
Published in Biochemistry (Easton) (19.05.2020)
Published in Biochemistry (Easton) (19.05.2020)
Get full text
Journal Article
Identification and characterization of NVP-BEZ235, a new orally available dual phosphatidylinositol 3-kinase/mammalian target of rapamycin inhibitor with potent in vivo antitumor activity
Maira, Sauveur-Michel, Stauffer, Frédéric, Brueggen, Josef, Furet, Pascal, Schnell, Christian, Fritsch, Christine, Brachmann, Saskia, Chène, Patrick, De Pover, Alain, Schoemaker, Kevin, Fabbro, Doriano, Gabriel, Daniela, Simonen, Marjo, Murphy, Leon, Finan, Peter, Sellers, William, García-Echeverría, Carlos
Published in Molecular cancer therapeutics (01.07.2008)
Published in Molecular cancer therapeutics (01.07.2008)
Get full text
Journal Article
Design and Biochemical Characterization of Peptidic Inhibitors of the Myb/p300 Interaction
Jones, Matthew, Grosche, Philipp, Floersheimer, Andreas, André, Jérome, Gattlen, Raphael, Oser, Dieter, Tinchant, Juliette, Wille, Roman, Chie-Leon, Barbara, Gerspacher, Marc, Ertl, Peter, Ostermann, Nils, Altmann, Eva, Manchado, Eusebio, Vorherr, Thomas, Chène, Patrick
Published in Biochemistry (Easton) (04.04.2023)
Published in Biochemistry (Easton) (04.04.2023)
Get full text
Journal Article
Identification and characterization of NVP-BKM120, an orally available pan-class I PI3-kinase inhibitor
Maira, Sauveur-Michel, Pecchi, Sabina, Huang, Alan, Burger, Matthew, Knapp, Mark, Sterker, Dario, Schnell, Christian, Guthy, Daniel, Nagel, Tobi, Wiesmann, Marion, Brachmann, Saskia, Fritsch, Christine, Dorsch, Marion, Chène, Patrick, Shoemaker, Kevin, De Pover, Alain, Menezes, Daniel, Martiny-Baron, Georg, Fabbro, Doriano, Wilson, Christopher J, Schlegel, Robert, Hofmann, Francesco, García-Echeverría, Carlos, Sellers, William R, Voliva, Charles F
Published in Molecular cancer therapeutics (01.02.2012)
Published in Molecular cancer therapeutics (01.02.2012)
Get full text
Journal Article
Structure-based design of potent linear peptide inhibitors of the YAP-TEAD protein-protein interaction derived from the YAP omega-loop sequence
Furet, Pascal, Salem, Bahaa, Mesrouze, Yannick, Schmelzle, Tobias, Lewis, Ian, Kallen, Joerg, Chène, Patrick
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Get full text
Journal Article
Biochemical properties of VGLL4 from Homo sapiens and Tgi from Drosophila melanogaster and possible biological implications
Mesrouze, Yannick, Meyerhofer, Marco, Zimmermann, Catherine, Fontana, Patrizia, Erdmann, Dirk, Chène, Patrick
Published in Protein science (01.09.2021)
Published in Protein science (01.09.2021)
Get full text
Journal Article