Catalytic properties and inhibition of proline-specific dipeptidyl peptidases II, IV and VII
Leiting, Barbara, Pryor, KellyAnn D, Wu, Joseph K, Marsilio, Frank, Patel, Reshma A, Craik, Charles S, Ellman, Jonathan A, Cummings, Richard T, Thornberry, Nancy A
Published in Biochemical journal (15.04.2003)
Published in Biochemical journal (15.04.2003)
Get full text
Journal Article
Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors
Xu, Jinyou, Wei, Lan, Mathvink, Robert, He, Jiafang, Park, You-Jung, He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Get full text
Journal Article
Discovery of potent, selective, and orally bioavailable oxadiazole-based dipeptidyl peptidase IV inhibitors
Xu, Jinyou, Wei, Lan, Mathvink, Robert J., Edmondson, Scott D., Eiermann, George J., He, Huaibing, Leone, Joseph F., Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Patel, Sangita B., Petrov, Aleksandr, Scapin, Giovanna, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
Get full text
Journal Article
Dipeptidyl peptidase IV inhibition for the treatment of type 2 diabetes : Potential importance of selectivity over dipeptidyl peptidases 8 and 9
LANKAS, George R, LEITING, Barbara, IPPOLITO, Dawn E, KIM, Dooseop, LYONS, Kathryn A, OK, Hyun O, PATEL, Reshma A, PETROV, Aleksandr N, PRYOR, Kelly Ann, XIAOXIA QIAN, REIGLE, Leah, WOODS, Andrea, ROY, Ranabir Sinha, WU, Joseph K, ZALLER, Dennis, XIAOPING ZHANG, LAN ZHU, WEBER, Ann E, THORNBERRY, Nancy A, EIERMANN, George J, BECONI, Maria G, BIFTU, Tesfaye, CHAN, Chi-Chung, EDMONDSON, Scott, FEENEY, William P, HUAIBING HE
Published in Diabetes (New York, N.Y.) (01.10.2005)
Published in Diabetes (New York, N.Y.) (01.10.2005)
Get full text
Journal Article
Diastereoselective synthesis and configuration-dependent activity of (3-substituted-cycloalkyl)glycine pyrrolidides and thiazolidides as dipeptidyl peptidase IV inhibitors
ASHTON, Wallace T, HONG DONG, SISCO, Rosemary M, DOSS, George A, LEITING, Barbara, PATEL, Reshma A, WU, Joseph K, MARSILIO, Frank, THOMBERRY, Nancy A, WEBER, Ann E
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Get full text
Journal Article
Fluoroolefins as amide bond mimics in dipeptidyl peptidase IV inhibitors
Edmondson, Scott D., Wei, Lan, Xu, Jinyou, Shang, Jackie, Xu, Shiyao, Pang, Jianmei, Chaudhary, Ashok, Dean, Dennis C., He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Patel, Reshma A., Patel, Sangita B., Scapin, Giovanna, Wu, Joseph K., Beconi, Maria G., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
Get full text
Journal Article
(2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4-[1,2,4]triazolo[1,5-a]- pyridin-6-ylphenyl)butanamide: A Selective α-Amino Amide Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes
Edmondson, Scott D, Mastracchio, Anthony, Mathvink, Robert J, He, Jiafang, Harper, Bart, Park, You-Jung, Beconi, Maria, Di Salvo, Jerry, Eiermann, George J, He, Huaibing, Leiting, Barbara, Leone, Joseph F, Levorse, Dorothy A, Lyons, Kathryn, Patel, Reshma A, Patel, Sangita B, Petrov, Aleksandr, Scapin, Giovanna, Shang, Jackie, Roy, Ranabir Sinha, Smith, Aaron, Wu, Joseph K, Xu, Shiyao, Zhu, Bing, Thornberry, Nancy A, Weber, Ann E
Published in Journal of medicinal chemistry (15.06.2006)
Published in Journal of medicinal chemistry (15.06.2006)
Get full text
Journal Article
(2R)-4-Oxo-4-[3-(Trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin- 7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine: A Potent, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes
Kim, Dooseop, Wang, Liping, Beconi, Maria, Eiermann, George J, Fisher, Michael H, He, Huaibing, Hickey, Gerard J, Kowalchick, Jennifer E, Leiting, Barbara, Lyons, Kathryn, Marsilio, Frank, McCann, Margaret E, Patel, Reshma A, Petrov, Aleksandr, Scapin, Giovanna, Patel, Sangita B, Roy, Ranabir Sinha, Wu, Joseph K, Wyvratt, Matthew J, Zhang, Bei B, Zhu, Lan, Thornberry, Nancy A, Weber, Ann E
Published in Journal of medicinal chemistry (13.01.2005)
Published in Journal of medicinal chemistry (13.01.2005)
Get full text
Journal Article
Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: Close analogs of JANUVIA™ (sitagliptin phosphate)
Kim, Dooseop, Kowalchick, Jennifer E., Edmondson, Scott D., Mastracchio, Anthony, Xu, Jinyou, Eiermann, George J., Leiting, Barbara, Wu, Joseph K., Pryor, KellyAnn D., Patel, Reshma A., He, Huaibing, Lyons, Kathryn A., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Get full text
Journal Article
Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors
Edmondson, Scott D., Mastracchio, Anthony, Cox, Jason M., Eiermann, George J., He, Huaibing, Lyons, Kathryn A., Patel, Reshma A., Patel, Sangita B., Petrov, Aleksandr, Scapin, Giovanna, Wu, Joseph K., Xu, Shiyao, Zhu, Bing, Thornberry, Nancy A., Roy, Ranabir Sinha, Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Get full text
Journal Article
Design, synthesis, and biological evaluation of triazolopiperazine-based β-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors
Kowalchick, Jennifer E., Leiting, Barbara, Pryor, KellyAnn D., Marsilio, Frank, Wu, Joseph K., He, Huaibing, Lyons, Kathryn A., Eiermann, George J., Petrov, Aleksandr, Scapin, Giovanna, Patel, Reshma A., Thornberry, Nancy A., Weber, Ann E., Kim, Dooseop
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Get full text
Journal Article
Substituted piperazines as novel dipeptidyl peptidase IV inhibitors
Brockunier, Linda L., He, Jiafang, Colwell, Lawrence F., Habulihaz, Bahanu, He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Teffera, Yohannes, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Get full text
Journal Article
Dipeptidyl peptidase IV inhibitors derived from β-aminoacylpiperidines bearing a fused thiazole, oxazole, isoxazole, or pyrazole
Ashton, Wallace T., Sisco, Rosemary M., Dong, Hong, Lyons, Kathryn A., He, Huaibing, Doss, George A., Leiting, Barbara, Patel, Reshma A., Wu, Joseph K., Marsilio, Frank, Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Get full text
Journal Article
Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors
Cox, Jason M., Harper, Bart, Mastracchio, Anthony, Leiting, Barbara, Sinha Roy, Ranabir, Patel, Reshma A., Wu, Joseph K., Lyons, Kathryn A., He, Huaibing, Xu, Shiyao, Zhu, Bing, Thornberry, Nancy A., Weber, Ann E., Edmondson, Scott D.
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Get full text
Journal Article
Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetes
Chen, Ping, Caldwell, Charles G., Mathvink, Robert J., Leiting, Barbara, Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., He, Huaibing, Lyons, Kathryn A., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Get full text
Journal Article
Fluoropyrrolidine amides as dipeptidyl peptidase IV inhibitors
CALDWELL, Charles G, PING CHEN, HUAIBING HE, LYONS, Kathryn A, THORNBERRY, Nancy A, WEBER, Ann E, JIAFANG HE, PARMEE, Emma R, LEITING, Barbara, MARSILIO, Frank, PATEL, Reshma A, WU, Joseph K, EIERMANN, George J, PETROV, Aleksandr
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Get full text
Journal Article
4-Aminophenylalanine and 4-aminocyclohexylalanine derivatives as potent, selective, and orally bioavailable inhibitors of dipeptidyl peptidase IV
Duffy, Joseph L., Kirk, Brian A., Wang, Liping, Eiermann, George J., He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Patel, Reshma A., Patel, Sangita B., Petrov, Alexsandr, Scapin, Giovanna, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Get full text
Journal Article
Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors
Edmondson, Scott D., Mastracchio, Anthony, Duffy, Joseph L., Eiermann, George J., He, Huaibing, Ita, Ida, Leiting, Barbara, Leone, Joseph F., Lyons, Kathryn A., Makarewicz, Amanda M., Patel, Reshma A., Petrov, Aleksandr, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
Get full text
Journal Article
Potent and selective proline derived dipeptidyl peptidase IV inhibitors
Edmondson, Scott D., Mastracchio, Anthony, Beconi, Maria, Colwell, Lawrence F., Habulihaz, Bahanu, He, Huaibing, Kumar, Sanjeev, Leiting, Barbara, Lyons, Kathryn A., Mao, Ann, Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., Zhu, Lan, Thornberry, Nancy A., Weber, Ann E., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Get full text
Journal Article
Discovery of potent and selective β-homophenylalanine based dipeptidyl peptidase IV inhibitors
Xu, Jinyou, Ok, Hyun O., Gonzalez, Edward J., Colwell, Lawrence F., Habulihaz, Bahanu, He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Get full text
Journal Article