Natural products and other inhibitors of F1FO ATP synthase
Patel, Bhargav A., D’Amico, Terin L., Blagg, Brian S.J.
Published in European journal of medicinal chemistry (01.12.2020)
Published in European journal of medicinal chemistry (01.12.2020)
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Journal Article
Bafetinib (INNO-406) reverses multidrug resistance by inhibiting the efflux function of ABCB1 and ABCG2 transporters
Zhang, Yun-Kai, Zhang, Guan-Nan, Wang, Yi-Jun, Patel, Bhargav A, Talele, Tanaji T, Yang, Dong-Hua, Chen, Zhe-Sheng
Published in Scientific reports (09.05.2016)
Published in Scientific reports (09.05.2016)
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Journal Article
Recent development in the discovery of PARP inhibitors as anticancer agents: a patent update (2016-2020)
Velagapudi, Uday Kiran, Patel, Bhargav A, Shao, Xuwei, Pathak, Sanjai Kumar, Ferraris, Dana V, Talele, Tanaji T
Published in Expert opinion on therapeutic patents (03.07.2021)
Published in Expert opinion on therapeutic patents (03.07.2021)
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Journal Article
Design and Synthesis of Human ABCB1 (P-Glycoprotein) Inhibitors by Peptide Coupling of Diverse Chemical Scaffolds on Carboxyl and Amino Termini of (S)‑Valine-Derived Thiazole Amino Acid
Singh, Satyakam, Prasad, Nagarajan Rajendra, Chufan, Eduardo E, Patel, Bhargav A, Wang, Yi-Jun, Chen, Zhe-Sheng, Ambudkar, Suresh V, Talele, Tanaji T
Published in Journal of medicinal chemistry (22.05.2014)
Published in Journal of medicinal chemistry (22.05.2014)
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Journal Article
In Vitro Antibacterial Activity of Rhodanine Derivatives against Pathogenic Clinical Isolates
AbdelKhalek, Ahmed, Ashby, Jr, Charles R, Patel, Bhargav A, Talele, Tanaji T, Seleem, Mohamed N
Published in PloS one (06.10.2016)
Published in PloS one (06.10.2016)
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Journal Article
Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1
Wang, Yi-Jun, Patel, Bhargav A, Anreddy, Nagaraju, Zhang, Yun-Kai, Zhang, Guan-Nan, Alqahtani, Saeed, Singh, Satyakam, Shukla, Suneet, Kaddoumi, Amal, Ambudkar, Suresh V, Talele, Tanaji T, Chen, Zhe-Sheng
Published in Scientific reports (09.02.2017)
Published in Scientific reports (09.02.2017)
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Journal Article
Novel 4-Thiazolidinones as Non-Nucleoside Inhibitors of Hepatitis C Virus NS5B RNA-Dependent RNA Polymerase
Çakır, Gizem, Küçükgüzel, İlkay, Guhamazumder, Rupa, Tatar, Esra, Manvar, Dinesh, Basu, Amartya, Patel, Bhargav A., Zia, Javairia, Talele, Tanaji T., Kaushik-Basu, Neerja
Published in Archiv der Pharmazie (Weinheim) (01.01.2015)
Published in Archiv der Pharmazie (Weinheim) (01.01.2015)
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Journal Article
Design, Synthesis, and Biological Evaluation of (S)-Valine Thiazole-Derived Cyclic and Noncyclic Peptidomimetic Oligomers as Modulators of Human P-Glycoprotein (ABCB1)
Singh, Satyakam, Prasad, Nagarajan Rajendra, Kapoor, Khyati, Chufan, Eduardo E., Patel, Bhargav A., Ambudkar, Suresh V., Talele, Tanaji T.
Published in Chembiochem : a European journal of chemical biology (03.01.2014)
Published in Chembiochem : a European journal of chemical biology (03.01.2014)
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Journal Article
CryoEM Structure with ATP Synthase Enables Late‐Stage Diversification of Cruentaren A
Dou, Xiaozheng, Guo, Hui, D'Amico, Terin, Abdallah, Leah, Subramanian, Chitra, Patel, Bhargav A., Cohen, Mark, Rubinstein, John L., Blagg, Brian S. J.
Published in Chemistry : a European journal (22.05.2023)
Published in Chemistry : a European journal (22.05.2023)
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Journal Article
Synthesis and Evaluation of Simplified Cruentaren A Analogues
Dou, Xiaozheng, Patel, Bhargav A., D’Amico, Terin, Subramanian, Chitra, Cousineau, Eric, Yi, Yi, Cohen, Mark, Blagg, Brian S. J.
Published in Journal of organic chemistry (05.08.2022)
Published in Journal of organic chemistry (05.08.2022)
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Journal Article
Design and Synthesis of Poly(ADP-ribose) Polymerase Inhibitors: Impact of Adenosine Pocket-Binding Motif Appendage to the 3‑Oxo-2,3-dihydrobenzofuran-7-carboxamide on Potency and Selectivity
Velagapudi, Uday Kiran, Langelier, Marie-France, Delgado-Martin, Cristina, Diolaiti, Morgan E, Bakker, Sietske, Ashworth, Alan, Patel, Bhargav A, Shao, Xuwei, Pascal, John M, Talele, Tanaji T
Published in Journal of medicinal chemistry (13.06.2019)
Published in Journal of medicinal chemistry (13.06.2019)
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Journal Article
Comprehensive Synthesis of Amino Acid-Derived Thiazole Peptidomimetic Analogues to Understand the Enigmatic Drug/Substrate-Binding Site of P‑Glycoprotein
Patel, Bhargav A, Abel, Biebele, Barbuti, Anna Maria, Velagapudi, Uday Kiran, Chen, Zhe-Sheng, Ambudkar, Suresh V, Talele, Tanaji T
Published in Journal of medicinal chemistry (08.02.2018)
Published in Journal of medicinal chemistry (08.02.2018)
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Journal Article
Manassantin A inhibits tumour growth under hypoxia through the activation of chaperone-mediated autophagy by modulating Hsp90 activity
Byun, Jun-Kyu, Lee, Sun Hee, Moon, Eui Jung, Park, Myo-Hyeon, Jang, Hyeonha, Weitzel, Douglas H, Kim, Hyun-Hwi, Basnet, Nikita, Kwon, Do-Yeon, Lee, Chen-Ting, Stephenson, Tesia N, Jeong, Ji-Hak, Patel, Bhargav A, Park, Sung Jean, Chi, Jen-Tsan, Dewhirst, Mark W, Hong, Jiyong, Lee, You Mie
Published in British journal of cancer (01.04.2023)
Published in British journal of cancer (01.04.2023)
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Journal Article
The BTK Inhibitor Ibrutinib (PCI-32765) Overcomes Paclitaxel Resistance in ABCB1- and ABCC10-Overexpressing Cells and Tumors
Zhang, Hui, Patel, Atish, Wang, Yi-Jun, Zhang, Yun-Kai, Kathawala, Rishil J, Qiu, Long-Hui, Patel, Bhargav A, Huang, Li-Hua, Shukla, Suneet, Yang, Dong-Hua, Ambudkar, Suresh V, Fu, Li-Wu, Chen, Zhe-Sheng
Published in Molecular cancer therapeutics (01.06.2017)
Published in Molecular cancer therapeutics (01.06.2017)
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Journal Article
The synthesis and SAR study of phenylalanine-derived (Z)-5-arylmethylidene rhodanines as anti-methicillin-resistant Staphylococcus aureus (MRSA) compounds
Patel, Bhargav A., Ashby, Charles R., Hardej, Diane, Talele, Tanaji T.
Published in Bioorganic & medicinal chemistry letters (15.10.2013)
Published in Bioorganic & medicinal chemistry letters (15.10.2013)
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Journal Article
Semi-synthetic ocotillol analogues as selective ABCB1-mediated drug resistance reversal agents
Zhang, Yun-Kai, Zhang, Hengyuan, Zhang, Guan-Nan, Wang, Yi-Jun, Kathawala, Rishil J, Si, Rui, Patel, Bhargav A, Xu, Jinyi, Chen, Zhe-Sheng
Published in Oncotarget (15.09.2015)
Published in Oncotarget (15.09.2015)
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Journal Article
Dual inhibition of Staphylococcus aureus DNA gyrase and topoisomerase IV activity by phenylalanine-derived (Z)-5-arylmethylidene rhodanines
Werner, Malela M., Patel, Bhargav A., Talele, Tanaji T., Ashby, Charles R., Li, Zhiyu, Zauhar, Randy J.
Published in Bioorganic & medicinal chemistry (15.09.2015)
Published in Bioorganic & medicinal chemistry (15.09.2015)
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Journal Article
Design and synthesis of l- and d-phenylalanine derived rhodanines with novel C5-arylidenes as inhibitors of HCV NS5B polymerase
Patel, Bhargav A., Krishnan, Ramalingam, Khadtare, Nikhil, Gurukumar, K.R., Basu, Amartya, Arora, Payal, Bhatt, Aaditya, Patel, Maulik R., Dana, Dibyendu, Kumar, Sanjai, Kaushik-Basu, Neerja, Talele, Tanaji T.
Published in Bioorganic & medicinal chemistry (01.06.2013)
Published in Bioorganic & medicinal chemistry (01.06.2013)
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Journal Article
Natural products and other inhibitors of F 1 F O ATP synthase
Patel, Bhargav A, D'Amico, Terin L, Blagg, Brian S J
Published in European journal of medicinal chemistry (01.12.2020)
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Published in European journal of medicinal chemistry (01.12.2020)
Journal Article