Synthesis of a selective HDAC6 inhibitor active in neuroblasts
Zwick, Vincent, Simões-Pires, Claudia A., Nurisso, Alessandra, Petit, Charlotte, Dos Santos Passos, Carolina, Randazzo, Giuseppe Marco, Martinet, Nadine, Bertrand, Philippe, Cuendet, Muriel
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
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Indole alkaloids and semisynthetic indole derivatives as multifunctional scaffolds aiming the inhibition of enzymes related to neurodegenerative diseases--a focus on Psychotria L. Genus
Klein, Jr, Luiz Carlos, Passos, Carolina Santos Dos, Moraes, Aline Pereira, Wakui, Vinicius Galvao, Konrath, Eduardo Luis, Nurisso, Alessandra, Carrupt, Pierre-Alain, de Oliveira, Cecilia Maria Alves, Kato, Lucilia, Henriques, Amelia Teresinha
Published in Current topics in medicinal chemistry (01.04.2014)
Published in Current topics in medicinal chemistry (01.04.2014)
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Monoamine oxidase inhibition by monoterpene indole alkaloids and fractions obtained from Psychotria suterella and Psychotria laciniata
dos Santos Passos, Carolina, Soldi, Tatiane Cristina, Torres Abib, Renata, Anders Apel, Miriam, Simões-Pires, Cláudia, Marcourt, Laurence, Gottfried, Carmem, Henriques, Amélia Teresinha
Published in Journal of enzyme inhibition and medicinal chemistry (01.06.2013)
Published in Journal of enzyme inhibition and medicinal chemistry (01.06.2013)
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Journal Article
Characterization of Lignanamides from Hemp (Cannabis sativa L.) Seed and Their Antioxidant and Acetylcholinesterase Inhibitory Activities
Yan, Xiaoli, Tang, Jiajing, dos Santos Passos, Carolina, Nurisso, Alessandra, Simões-Pires, Claudia Avello, Ji, Mei, Lou, Hongxiang, Fan, Peihong
Published in Journal of agricultural and food chemistry (16.12.2015)
Published in Journal of agricultural and food chemistry (16.12.2015)
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Journal Article
Gephyrin promotes autonomous assembly and synaptic localization of GABAergic postsynaptic components without presynaptic GABA release
Carricaburu, Etta, Benner, Orion, Burlingham, Scott R, Passos, Carolina Dos Santos, Hobaugh, Natalia, Karr, Charles H, Chanda, Soham
Published in Proceedings of the National Academy of Sciences - PNAS (25.06.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (25.06.2024)
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Crucial roles of the BRCA1-BARD1 E3 ubiquitin ligase activity in homology-directed DNA repair
Wang, Meiling, Li, Wenjing, Tomimatsu, Nozomi, Yu, Corey H., Ji, Jae-Hoon, Alejo, Salvador, Witus, Samuel R., Alimbetov, Dauren, Fitzgerald, O’Taveon, Wu, Bo, Wang, Qijing, Huang, Yuxin, Gan, Yaqi, Dong, Felix, Kwon, Youngho, Sareddy, Gangadhara R., Curiel, Tyler J., Habib, Amyn A., Hromas, Robert, dos Santos Passos, Carolina, Yao, Tingting, Ivanov, Dmitri N., Brzovic, Peter S., Burma, Sandeep, Klevit, Rachel E., Zhao, Weixing
Published in Molecular cell (19.10.2023)
Published in Molecular cell (19.10.2023)
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Induction of synapse formation by de novo neurotransmitter synthesis
Burlingham, Scott R, Wong, Nicole F, Peterkin, Lindsay, Lubow, Lily, Dos Santos Passos, Carolina, Benner, Orion, Ghebrial, Michael, Cast, Thomas P, Xu-Friedman, Matthew A, Südhof, Thomas C, Chanda, Soham
Published in Nature communications (01.06.2022)
Published in Nature communications (01.06.2022)
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A Rational Approach for the Identification of Non-Hydroxamate HDAC6-Selective Inhibitors
Goracci, Laura, Deschamps, Nathalie, Randazzo, Giuseppe Marco, Petit, Charlotte, Dos Santos Passos, Carolina, Carrupt, Pierre-Alain, Simões-Pires, Claudia, Nurisso, Alessandra
Published in Scientific reports (12.07.2016)
Published in Scientific reports (12.07.2016)
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Combining in vitro and in silico approaches to evaluate the multifunctional profile of rosmarinic acid from Blechnum brasiliense on targets related to neurodegeneration
Andrade, Juliana Maria de Mello, dos Santos Passos, Carolina, Kieling Rubio, Maria Angélica, Mendonça, Jacqueline Nakau, Lopes, Norberto Peporine, Henriques, Amélia Teresinha
Published in Chemico-biological interactions (25.07.2016)
Published in Chemico-biological interactions (25.07.2016)
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Kopsanone and N-oxide isolated from Aspidosperma macrocarpon Mart. (Apocynaceae) leaves and their MAO-A inhibitory activity
Peixoto, Matheus Ardenghi, Kato, Lucilia, Alves de Oliveira, Cecília Maria, Gontijo, Boniek, da Silva, Cleuza Conceição, Pomini, Armando Mateus, Klein-Júnior, Luiz C., Passos, Carolina dos Santos, Henriques, Amélia T., Bannwart, Geanderson, Santin, Silvana Maria de Oliveira
Published in Natural product research (02.12.2021)
Published in Natural product research (02.12.2021)
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Investigation of the in vitro and ex vivo acetylcholinesterase and antioxidant activities of traditionally used Lycopodium species from South America on alkaloid extracts
Konrath, Eduardo Luis, Neves, Bruna Medeiros, Lunardi, Paula Santana, Passos, Carolina dos Santos, Simões-Pires, André, Ortega, María Gabriela, Gonçalves, Carlos Alberto, Cabrera, José L., Moreira, José Cláudio Fonseca, Henriques, Amélia T.
Published in Journal of ethnopharmacology (06.01.2012)
Published in Journal of ethnopharmacology (06.01.2012)
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Journal Article
Alkaloids from Psychotria Target Sirtuins: In Silico and In Vitro Interaction Studies
Sacconnay, Lionel, Ryckewaert, Lucie, dos Santos Passos, Carolina, Guerra, Maria Cristina, Kato, Lucilia, Alves de Oliveira, Cecilia Maria, Henriques, Amélia, Carrupt, Pierre-Alain, Simões-Pires, Claudia, Nurisso, Alessandra
Published in Planta medica (01.04.2015)
Published in Planta medica (01.04.2015)
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Monoamine Oxidase Inhibitory Activity of Biflavonoids from Branches of Garcinia gardneriana (Clusiaceae)
Recalde-Gil, Maria Angélica, Klein-Júnior, Luiz Carlos, dos Santos Passos, Carolina, Salton, Juliana, de Loreto Bordignon, Sérgio Augusto, Monace, Franco Delle, Filho, Valdir Cechinel, Henriques, Amélia Teresinha
Published in Natural product communications (01.04.2017)
Published in Natural product communications (01.04.2017)
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Journal Article
The catechol-O-methyltransferase inhibitory potential of Z-vallesiachotamine by in silico and in vitro approaches
dos Santos Passos, Carolina, Klein-Júnior, Luiz Carlos, de Mello Andrade, Juliana Maria, Matté, Cristiane, Henriques, Amélia Teresinha
Published in Revista brasileira de farmacognosia (01.07.2015)
Published in Revista brasileira de farmacognosia (01.07.2015)
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Journal Article
Multifunctional Monoamine Oxidases and Cholinesterases Inhibitory Effects, as well as UPLC-DAD-MS Chemical Profile of Alkaloid Fractions Obtained from Species of the Palicoureeae Tribe
Klein-Júnior, Luiz Carlos, Passos, Carolina dos Santos, Salton, Juliana, Bitencourt de, Fernanda Gobbi, Funez, Luís, de Andrade, Jean Paulo, Villalobos, Jonathan Parra, de Loreto Bordignon, Sérgio Augusto, Gasper, André Luís, Heyden, Yvan Vander, Henriques, Amélia Teresinha
Published in Natural product communications (01.09.2016)
Published in Natural product communications (01.09.2016)
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Alkaloids as a source of potential anticholinesterase inhibitors for the treatment of Alzheimer's disease
Konrath, Eduardo Luis, Passos, Carolina dos Santos, Klein, Jr, Luiz Carlos, Henriques, Amélia T
Published in Journal of pharmacy and pharmacology (01.12.2013)
Published in Journal of pharmacy and pharmacology (01.12.2013)
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5-Benzylidene-hydantoin is a new scaffold for SIRT inhibition: From virtual screening to activity assays
Sacconnay, Lionel, Ryckewaert, Lucie, Randazzo, Giuseppe Marco, Petit, Charlotte, Passos, Carolina Dos Santos, Jachno, Jelena, Michailovienė, Vilma, Zubrienė, Asta, Matulis, Daumantas, Carrupt, Pierre-Alain, Simões-Pires, Claudia Avello, Nurisso, Alessandra
Published in European journal of pharmaceutical sciences (31.03.2016)
Published in European journal of pharmaceutical sciences (31.03.2016)
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