Ligand-based G Protein Coupled Receptor pharmacophore modeling: Assessing the role of ligand function in model development
Castleman, P., Szwabowski, G., Bowman, D., Cole, J., Parrill, A.L., Baker, D.L.
Published in Journal of molecular graphics & modelling (01.03.2022)
Published in Journal of molecular graphics & modelling (01.03.2022)
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Short-Chain Phosphatidates Are Subtype-Selective Antagonists of Lysophosphatidic Acid Receptors
Fischer, D J, Nusser, N, Virag, T, Yokoyama, K, Wang Da, Baker, D L, Bautista, D, Parrill, A L, Tigyi, G
Published in Molecular pharmacology (01.10.2001)
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Published in Molecular pharmacology (01.10.2001)
Journal Article
Identification of Edg1 Receptor Residues That Recognize Sphingosine 1-Phosphate
Parrill, Abby L., Wang, De-an, Bautista, Debra L., Van Brocklyn, James R., Lorincz, Zsolt, Fischer, David J., Baker, Daniel L., Liliom, Karoly, Spiegel, Sarah, Tigyi, Gabor
Published in The Journal of biological chemistry (15.12.2000)
Published in The Journal of biological chemistry (15.12.2000)
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Molecular Models of N-Benzyladriamycin-14-valerate (AD 198) in Complex with the Phorbol Ester-Binding C1b Domain of Protein Kinase C-δ
Roaten, J. Brent, Kazanietz, Marcelo G, Sweatman, Trevor W, Lothstein, Leonard, Israel, Mervyn, Parrill, Abby L
Published in Journal of medicinal chemistry (29.03.2001)
Published in Journal of medicinal chemistry (29.03.2001)
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Journal Article
Structural Features of EDG1 Receptor-Ligand Complexes Revealed by Computational Modeling and Mutagenesis
PARRILL, ABBY L., BAKER, DANIEL L., WANG, DE-AN, FISCHER, DAVID J., BAUTISTA, DEBRA L., VAN BROCKLYN, JAMES, SPIEGEL, SARAH, TIGYI, GABOR
Published in Annals of the New York Academy of Sciences (01.04.2000)
Published in Annals of the New York Academy of Sciences (01.04.2000)
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Journal Article
CLEW: The Generation of Pharmacophore Hypotheses Through Machine Learning
Dolata, D. P., Parrill, A. L., Walters, W. P.
Published in SAR and QSAR in environmental research (01.01.1998)
Published in SAR and QSAR in environmental research (01.01.1998)
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Targeting the hydrophobic pocket of autotaxin with virtual screening of inhibitors identifies a common aromatic sulfonamide structural motif
Fells, James I., Lee, Sue Chin, Norman, Derek D., Tsukahara, Ryoko, Kirby, Jason R., Nelson, Sandra, Seibel, William, Papoian, Ruben, Patil, Renukadevi, Miller, Duane D., Parrill, Abby L., Pham, Truc‐Chi, Baker, Daniel L., Bittman, Robert, Tigyi, Gabor
Published in The FEBS journal (01.02.2014)
Published in The FEBS journal (01.02.2014)
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Journal Article
Dynamic modeling of EDG1 receptor structural changes induced by site-directed mutations
Bautista, D.L, Baker, D.L, Wang, D, Fischer, D.J, Van Brocklyn, J, Spiegel, S, Tigyi, G, Parrill, A.L
Published in Journal of molecular structure. Theochem (08.09.2000)
Published in Journal of molecular structure. Theochem (08.09.2000)
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Synthesis and pharmacological evaluation of second-generation phosphatidic acid derivatives as lysophosphatidic acid receptor ligands
Durgam, Gangadhar G., Tsukahara, Ryoko, Makarova, Natalia, Walker, Michelle D., Fujiwara, Yuko, Pigg, Kathryn R., Baker, Daniel L., Sardar, Vineet M., Parrill, Abby L., Tigyi, Gabor, Miller, Duane D.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Journal Article
Solid phase synthesis and secondary structural studies of (1 - 5) amide-linked sialooligomers
Szabo, L, Smith, BL, McReynolds, KD, Parrill, AL, Morris, ER, Gervay, J
Published in Journal of organic chemistry (20.02.1998)
Published in Journal of organic chemistry (20.02.1998)
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Journal Article
Fatty Alcohol Phosphates are Subtype-Selective Agonists and Antagonists of Lysophosphatidic Acid Receptors
Virag, Tamas, Elrod, Don B, Liliom, Karoly, Sardar, Vineet M, Parrill, Abby L, Yokoyama, Kazuaki, Durgam, Gangadhar, Deng, Wenlin, Miller, Duane D, Tigyi, Gabor
Published in Molecular pharmacology (01.05.2003)
Published in Molecular pharmacology (01.05.2003)
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