Potent antimyeloma activity of the novel bromodomain inhibitors I-BET151 and I-BET762
Chaidos, Aristeidis, Caputo, Valentina, Gouvedenou, Katerina, Liu, Binbin, Marigo, Ilaria, Chaudhry, Mohammed Suhail, Rotolo, Antonia, Tough, David F., Smithers, Nicholas N., Bassil, Anna K., Chapman, Trevor D., Harker, Nicola R., Barbash, Olena, Tummino, Peter, Al-Mahdi, Niam, Haynes, Andrea C., Cutler, Leanne, Le, BaoChau, Rahemtulla, Amin, Roberts, Irene, Kleijnen, Maurits, Witherington, Jason J., Parr, Nigel J., Prinjha, Rab K., Karadimitris, Anastasios
Published in Blood (30.01.2014)
Published in Blood (30.01.2014)
Get full text
Journal Article
Selective inhibition of CD4⁺ T-cell cytokine production and autoimmunity by BET protein and c-Myc inhibitors
Bandukwala, Hozefa S, Gagnon, John, Togher, Susan, Greenbaum, Jason A, Lamperti, Edward D, Parr, Nigel J, Molesworth, Amy M. H, Smithers, Nicholas, Lee, Kevin, Witherington, Jason, Tough, David F, Prinjha, Rab K, Peters, Bjoern, Rao, Anjana
Published in Proceedings of the National Academy of Sciences - PNAS (04.09.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (04.09.2012)
Get full text
Journal Article
Assessing color cues of development, breeding status and reproductive condition in captive golden lion tamarins (Leontopithecus rosalia)
Moreira, Lais A A, Merrigan-Johnson, Carrie, Fetherstonhaugh, Laura, Parr, Nigel A, Higham, James P, Melin, Amanda D
Published in American journal of primatology (01.10.2023)
Published in American journal of primatology (01.10.2023)
Get full text
Journal Article
Discovery of Epigenetic Regulator I‑BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains
Mirguet, Olivier, Gosmini, Romain, Toum, Jérôme, Clément, Catherine A, Barnathan, Mélanie, Brusq, Jean-Marie, Mordaunt, Jacqueline E, Grimes, Richard M, Crowe, Miriam, Pineau, Olivier, Ajakane, Myriam, Daugan, Alain, Jeffrey, Phillip, Cutler, Leanne, Haynes, Andrea C, Smithers, Nicholas N, Chung, Chun-wa, Bamborough, Paul, Uings, Iain J, Lewis, Antonia, Witherington, Jason, Parr, Nigel, Prinjha, Rab K, Nicodème, Edwige
Published in Journal of medicinal chemistry (10.10.2013)
Published in Journal of medicinal chemistry (10.10.2013)
Get full text
Journal Article
Optimization of Novel Indazoles as Highly Potent and Selective Inhibitors of Phosphoinositide 3‑Kinase δ for the Treatment of Respiratory Disease
Down, Kenneth, Amour, Augustin, Baldwin, Ian R, Cooper, Anthony W. J, Deakin, Angela M, Felton, Leigh M, Guntrip, Stephen B, Hardy, Charlotte, Harrison, Zoë A, Jones, Katherine L, Jones, Paul, Keeling, Suzanne E, Le, Joelle, Livia, Stefano, Lucas, Fiona, Lunniss, Christopher J, Parr, Nigel J, Robinson, Ed, Rowland, Paul, Smith, Sarah, Thomas, Daniel A, Vitulli, Giovanni, Washio, Yoshiaki, Hamblin, J. Nicole
Published in Journal of medicinal chemistry (24.09.2015)
Published in Journal of medicinal chemistry (24.09.2015)
Get full text
Journal Article
Long‐term changes in bone mineral density and predicted fracture risk in patients receiving androgen‐deprivation therapy for prostate cancer, with stratification of treatment based on presenting values
Wadhwa, Vivek K., Weston, Robin, Mistry, Rahul, Parr, Nigel J.
Published in BJU international (01.09.2009)
Published in BJU international (01.09.2009)
Get full text
Journal Article
BET inhibition silences expression of MYCN and BCL2 and induces cytotoxicity in neuroblastoma tumor models
Wyce, Anastasia, Ganji, Gopinath, Smitheman, Kimberly N, Chung, Chun-Wa, Korenchuk, Susan, Bai, Yuchen, Barbash, Olena, Le, BaoChau, Craggs, Peter D, McCabe, Michael T, Kennedy-Wilson, Karen M, Sanchez, Lydia V, Gosmini, Romain L, Parr, Nigel, McHugh, Charles F, Dhanak, Dashyant, Prinjha, Rab K, Auger, Kurt R, Tummino, Peter J
Published in PloS one (23.08.2013)
Published in PloS one (23.08.2013)
Get full text
Journal Article
Discovery of a Novel Bromodomain and Extra Terminal Domain (BET) Protein Inhibitor, I-BET282E, Suitable for Clinical Progression
Jones, Katherine L., Beaumont, Dominic M., Bernard, Sharon G., Bit, Rino A., Campbell, Simon P., Chung, Chun-wa, Cutler, Leanne, Demont, Emmanuel H., Dennis, Kate, Gordon, Laurie, Gray, James R., Haase, Michael, Lewis, Antonia J., McCleary, Scott, Mitchell, Darren J., Moore, Susanne M., Parr, Nigel, Robb, Olivia J., Smithers, Nicholas, Soden, Peter E., Suckling, Colin J., Taylor, Simon, Walker, Ann L., Watson, Robert J., Prinjha, Rab K.
Published in Journal of medicinal chemistry (26.08.2021)
Published in Journal of medicinal chemistry (26.08.2021)
Get full text
Journal Article
Phase 1 and preclinical profiling of ESM‐HDAC391, a myeloid‐targeted histone deacetylase inhibitor, shows enhanced pharmacology and monocytopaenia
Furze, Rebecca C., Molnar, Judit, Parr, Nigel J., Ahmad, Faiz, Henry, Yvette, Howe, David, Singh, Rajendra, Toal, Martin, Bassil, Anna K., Bernard, Sharon G., Davis, Robert P., Gibson, Adele, Maller, N. Claire, Sharp, Catriona, Tough, David F., Prinjha, Rab K., Lewis, Huw D.
Published in British journal of clinical pharmacology (01.12.2022)
Published in British journal of clinical pharmacology (01.12.2022)
Get full text
Journal Article
Drivers of home range characteristics across spatiotemporal scales in a Neotropical primate, Cebus capucinus
Campos, Fernando A., Bergstrom, Mackenzie L., Childers, Andrew, Hogan, Jeremy D., Jack, Katharine M., Melin, Amanda D., Mosdossy, Krisztina N., Myers, Monica S., Parr, Nigel A., Sargeant, Elizabeth, Schoof, Valérie A.M., Fedigan, Linda M.
Published in Animal behaviour (01.05.2014)
Published in Animal behaviour (01.05.2014)
Get full text
Journal Article
The treatment of penile carcinoma in situ (CIS) within a UK supra‐regional network
Lucky, Marc, Murthy, Kusuma V.R., Rogers, Beverley, Jones, Stephen, Lau, Maurice W., Sangar, Vijay K., Parr, Nigel J.
Published in BJU international (01.04.2015)
Published in BJU international (01.04.2015)
Get full text
Journal Article
Guidance for the assessment and management of prostate cancer treatment-induced bone loss. A consensus position statement from an expert group
Brown, Janet E., Handforth, Catherine, Compston, Juliet E., Cross, William, Parr, Nigel, Selby, Peter, Wood, Steven, Drudge-Coates, Lawrence, Walsh, Jennifer S., Mitchell, Caroline, Collinson, Fiona J., Coleman, Robert E., James, Nicholas, Francis, Roger, Reid, David M., McCloskey, Eugene
Published in Journal of bone oncology (01.12.2020)
Published in Journal of bone oncology (01.12.2020)
Get full text
Journal Article
The structure based design of dual HDAC/BET inhibitors as novel epigenetic probes
Atkinson, Stephen J., Soden, Peter E., Angell, Davina C., Bantscheff, Marcus, Chung, Chun-wa, Giblin, Kathryn A., Smithers, Nicholas, Furze, Rebecca C., Gordon, Laurie, Drewes, Gerard, Rioja, Inmaculada, Witherington, Jason, Parr, Nigel J., Prinjha, Rab K.
Published in MedChemComm (2014)
Published in MedChemComm (2014)
Get full text
Journal Article
Predictors of Parasitism in Wild White-Faced Capuchins (Cebus capucinus)
Parr, Nigel A., Fedigan, Linda M., Kutz, Susan J.
Published in International journal of primatology (01.12.2013)
Published in International journal of primatology (01.12.2013)
Get full text
Journal Article
Should centralized histopathological review in penile cancer be the global standard?
Tang, Vincent, Clarke, Laurence, Gall, Zara, Shanks, Jonathan H., Nonaka, Daisuke, Parr, Nigel J., Elliott, P. Anthony, Clarke, Noel W., Ramani, Vijay, Lau, Maurice W., Sangar, Vijay K.
Published in BJU international (01.09.2014)
Published in BJU international (01.09.2014)
Get full text
Journal Article
Chemical Composition of Gases Surgeons Are Exposed to During Endoscopic Urological Resections
Weston, Robin, Stephenson, Richard N, Kutarski, Paul W, Parr, Nigel J
Published in Urology (Ridgewood, N.J.) (01.11.2009)
Published in Urology (Ridgewood, N.J.) (01.11.2009)
Get full text
Journal Article