Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans
Lutz, Joshua A, Sulima, Agnieszka, Gutman, Eugene S, Bow, Eric W, Luo, Dan, Kaska, Sophia, Prisinzano, Thomas E, Paronis, Carol A, Bergman, Jack, Imler, Gregory H, Kerr, Andrew T, Jacobson, Arthur E, Rice, Kenner C
Published in Molecules (Basel, Switzerland) (15.06.2023)
Published in Molecules (Basel, Switzerland) (15.06.2023)
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A Journey through Diastereomeric Space: The Design, Synthesis, In Vitro and In Vivo Pharmacological Activity, and Molecular Modeling of Novel Potent Diastereomeric MOR Agonists and Antagonists
Chambers, Dana R, Sulima, Agnieszka, Luo, Dan, Prisinzano, Thomas E, Goldberg, Alexander, Xie, Bing, Shi, Lei, Paronis, Carol A, Bergman, Jack, Nassehi, Nima, Selley, Dana E, Imler, Gregory H, Jacobson, Arthur E, Rice, Kenner C
Published in Molecules (Basel, Switzerland) (30.09.2022)
Published in Molecules (Basel, Switzerland) (30.09.2022)
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Altered sleep during spontaneous cannabinoid withdrawal in male mice
Missig, Galen, Mehta, Niyati, Robbins, James O, Good, Cameron H, Iliopoulos-Tsoutsouvas, Christos, Makriyannis, Alex, Nikas, Spyros P, Bergman, Jack, Carlezon, Jr, William A, Paronis, Carol A
Published in Behavioural pharmacology (01.04.2022)
Published in Behavioural pharmacology (01.04.2022)
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The Intriguing Effects of Substituents in the N -Phenethyl Moiety of Norhydromorphone: A Bifunctional Opioid from a Set of "Tail Wags Dog" Experiments
Wang, Meining, Irvin, Thomas C, Herdman, Christine A, Hanna, Ramsey D, Hassan, Sergio A, Lee, Yong-Sok, Kaska, Sophia, Crowley, Rachel Saylor, Prisinzano, Thomas E, Withey, Sarah L, Paronis, Carol A, Bergman, Jack, Inan, Saadet, Geller, Ellen B, Adler, Martin W, Kopajtic, Theresa A, Katz, Jonathan L, Chadderdon, Aaron M, Traynor, John R, Jacobson, Arthur E, Rice, Kenner C
Published in Molecules (Basel, Switzerland) (06.06.2020)
Published in Molecules (Basel, Switzerland) (06.06.2020)
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Probing the Carboxyester Side Chain in Controlled Deactivation (−)‑Δ8‑Tetrahydrocannabinols
Nikas, Spyros P, Sharma, Rishi, Paronis, Carol A, Kulkarni, Shashank, Thakur, Ganesh A, Hurst, Dow, Wood, JodiAnne T, Gifford, Roger S, Rajarshi, Girija, Liu, Yingpeng, Raghav, Jimit Girish, Guo, Jason Jianxin, Järbe, Torbjörn U.C, Reggio, Patricia H, Bergman, Jack, Makriyannis, Alexandros
Published in Journal of medicinal chemistry (22.01.2015)
Published in Journal of medicinal chemistry (22.01.2015)
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Δ(9)-Tetrahydrocannabinol acts as a partial agonist/antagonist in mice
Paronis, Carol A, Nikas, Spyros P, Shukla, Vidyanand G, Makriyannis, Alexandros
Published in Behavioural pharmacology (01.12.2012)
Published in Behavioural pharmacology (01.12.2012)
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Reinforcing effects of synthetic cathinones in rhesus monkeys: Dose-response and behavioral economic analyses
de Moura, Fernando B., Sherwood, Alexander, Prisinzano, Thomas E., Paronis, Carol A., Bergman, Jack, Kohut, Stephen J.
Published in Pharmacology, biochemistry and behavior (01.03.2021)
Published in Pharmacology, biochemistry and behavior (01.03.2021)
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Cannabinoid-induced lower lip retraction in rats
Chopda, Girish R., Nikas, Spyros P., Sharma, Rishi, Kulkarni, Shashank, Makriyannis, Alexandros, Paronis, Carol A.
Published in Psychopharmacology (01.04.2019)
Published in Psychopharmacology (01.04.2019)
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Improved cyclobutyl nabilone analogs as potent CB1 receptor agonists
Papanastasiou, Ioannis P., Georgiadis, Markos-Orestis, Iliopoulos-Tsoutsouvas, Christos, Paronis, Carol A., Brust, Christina A., Tran, Ngan K., Ji, Lipin, Ma, Xiaoyu, Wood, JodiAnne T., Zvonok, Nikolai, Tong, Fei, Bohn, Laura M., Nikas, Spyros P., Makriyannis, Alexandros
Published in European journal of medicinal chemistry (15.02.2022)
Published in European journal of medicinal chemistry (15.02.2022)
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Discriminative-Stimulus Effects of Synthetic Cathinones in Squirrel Monkeys
Wakeford, Alison G P, Sherwood, Alexander M, Prisinzano, Thomas E, Bergman, Jack, Kohut, Stephen J, Paronis, Carol A
Published in The international journal of neuropsychopharmacology (01.08.2021)
Published in The international journal of neuropsychopharmacology (01.08.2021)
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Tolerance to the Diuretic Effects of Cannabinoids and Cross-Tolerance to a κ-Opioid Agonist in THC-Treated Mice
Chopda, Girish R, Parge, Viraj, Thakur, Ganesh A, Gatley, S John, Makriyannis, Alexandros, Paronis, Carol A
Published in The Journal of pharmacology and experimental therapeutics (01.08.2016)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2016)
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