Development of a Minimalistic Physiologically Based Pharmacokinetic (mPBPK) Model for the Preclinical Development of Spectinamide Antibiotics
Parmar, Keyur R, Lukka, Pradeep B, Wagh, Santosh, Temrikar, Zaid H, Liu, Jiuyu, Lee, Richard E, Braunstein, Miriam, Hickey, Anthony J, Robertson, Gregory T, Gonzalez-Juarrero, Mercedes, Edginton, Andrea, Meibohm, Bernd
Published in Pharmaceutics (01.06.2023)
Published in Pharmaceutics (01.06.2023)
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Enhancing the therapeutic window for Spectinamide anti-tuberculosis Agents: Synthesis, Evaluation, and activation of phosphate prodrug 3408
Liu, Jiuyu, Lukka, Pradeep B., Ektnitphong, Victoria A., Parmar, Keyur R., Wagh, Santosh, Lu, Yan, Lee, Robin B., Scherbakov, Dimitri, Wang, Han, Zimmerman, Matthew D, Meibohm, Bernd, Robertson, Gregory T., Dartois, Vêronique, Böttger, Erik C., Lenaerts, Anne J., Lee, Richard E.
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
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Efficacy of a brain-penetrant antiviral in lethal Venezuelan and eastern equine encephalitis mouse models
Cao, Xufeng, Yang, Dong, Parvathareddy, Jyothi, Chu, Yong-Kyu, Kim, Eun Jung, Fitz-Henley, Jhewelle N, Li, Xiaoyu, Lukka, Pradeep B, Parmar, Keyur R, Temrikar, Zaid H, Dhole, Priya, Adcock, Robert Scott, Gabbard, Jon, Bansal, Shruti, Lee, Jasper, Zalduondo, Lillian, Hayes, Ernestine, Stabenow, Jennifer, Meibohm, Bernd, Fitzpatrick, Elizabeth A, Bailey, Kevin, Campos, Rafael K, Julander, Justin G, Rossi, Shannan L, Chung, Donghoon, Jonsson, Colleen B, Golden, Jennifer E
Published in Science translational medicine (12.04.2023)
Published in Science translational medicine (12.04.2023)
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Novel, Brain-Permeable, Cross-Species Benzothiazole Inhibitors of Microsomal Prostaglandin E Synthase‑1 (mPGES-1) Dampen Neuroinflammation In Vitro and In Vivo
Sluter, Madison N., Bhuniya, Rajib, Yuan, Xinrui, Ramaraju, Andhavaram, Chen, Yu, Yu, Ying, Parmar, Keyur R., Temrikar, Zaid H., Srivastava, Ashish, Meibohm, Bernd, Jiang, Jianxiong, Yang, Chao-Yie
Published in ACS pharmacology & translational science (14.04.2023)
Published in ACS pharmacology & translational science (14.04.2023)
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