Enhancing the therapeutic window for Spectinamide anti-tuberculosis Agents: Synthesis, Evaluation, and activation of phosphate prodrug 3408
Liu, Jiuyu, Lukka, Pradeep B., Ektnitphong, Victoria A., Parmar, Keyur R., Wagh, Santosh, Lu, Yan, Lee, Robin B., Scherbakov, Dimitri, Wang, Han, Zimmerman, Matthew D, Meibohm, Bernd, Robertson, Gregory T., Dartois, Vêronique, Böttger, Erik C., Lenaerts, Anne J., Lee, Richard E.
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
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Journal Article
Efficacy of a brain-penetrant antiviral in lethal Venezuelan and eastern equine encephalitis mouse models
Cao, Xufeng, Yang, Dong, Parvathareddy, Jyothi, Chu, Yong-Kyu, Kim, Eun Jung, Fitz-Henley, Jhewelle N, Li, Xiaoyu, Lukka, Pradeep B, Parmar, Keyur R, Temrikar, Zaid H, Dhole, Priya, Adcock, Robert Scott, Gabbard, Jon, Bansal, Shruti, Lee, Jasper, Zalduondo, Lillian, Hayes, Ernestine, Stabenow, Jennifer, Meibohm, Bernd, Fitzpatrick, Elizabeth A, Bailey, Kevin, Campos, Rafael K, Julander, Justin G, Rossi, Shannan L, Chung, Donghoon, Jonsson, Colleen B, Golden, Jennifer E
Published in Science translational medicine (12.04.2023)
Published in Science translational medicine (12.04.2023)
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Journal Article
A systematic review of decentralized finance protocols
Shah, Kaushal, Lathiya, Dhruvil, Lukhi, Naimish, Parmar, Keyur, Sanghvi, Harshal
Published in International journal of intelligent networks (2023)
Published in International journal of intelligent networks (2023)
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Journal Article
Development of a Minimalistic Physiologically Based Pharmacokinetic (mPBPK) Model for the Preclinical Development of Spectinamide Antibiotics
Parmar, Keyur R, Lukka, Pradeep B, Wagh, Santosh, Temrikar, Zaid H, Liu, Jiuyu, Lee, Richard E, Braunstein, Miriam, Hickey, Anthony J, Robertson, Gregory T, Gonzalez-Juarrero, Mercedes, Edginton, Andrea, Meibohm, Bernd
Published in Pharmaceutics (01.06.2023)
Published in Pharmaceutics (01.06.2023)
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Journal Article
Novel, Brain-Permeable, Cross-Species Benzothiazole Inhibitors of Microsomal Prostaglandin E Synthase‑1 (mPGES-1) Dampen Neuroinflammation In Vitro and In Vivo
Sluter, Madison N., Bhuniya, Rajib, Yuan, Xinrui, Ramaraju, Andhavaram, Chen, Yu, Yu, Ying, Parmar, Keyur R., Temrikar, Zaid H., Srivastava, Ashish, Meibohm, Bernd, Jiang, Jianxiong, Yang, Chao-Yie
Published in ACS pharmacology & translational science (14.04.2023)
Published in ACS pharmacology & translational science (14.04.2023)
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Journal Article
A rare complication of iliac bone grafting
Parmar, Keyur, Bhatia, Chisel, Bhardwaj, Sushma, Singh, Simrandeep, Kaushik, Robin
Published in International Journal of Abdominal Wall and Hernia Surgery (01.07.2020)
Published in International Journal of Abdominal Wall and Hernia Surgery (01.07.2020)
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Journal Article
PGASH: Provable group-based authentication scheme for Internet of Healthcare Things
Trivedi, Chandan, Parmar, Keyur, Rao, Udai Pratap
Published in Peer-to-peer networking and applications (01.03.2024)
Published in Peer-to-peer networking and applications (01.03.2024)
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Journal Article
Phytochemically analysed extract of Ageratina adenophora (Sprengel) R.M.King & H. Rob. initiates caspase 3-dependant apoptosis in colorectal cancer cell: A synergistic approach with chemotherapeutic drugs
Chanu, Khaidem Devika, Thoithoisana, Soibam, Kar, Amit, Mukherjee, Pulok Kumar, Radhakrishnanand, P, Parmar, Keyur, Sharma, Nanaocha
Published in Journal of ethnopharmacology (25.03.2024)
Published in Journal of ethnopharmacology (25.03.2024)
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Journal Article
Concealed data aggregation in wireless sensor networks: A comprehensive survey
Parmar, Keyur, Jinwala, Devesh C.
Published in Computer networks (Amsterdam, Netherlands : 1999) (05.07.2016)
Published in Computer networks (Amsterdam, Netherlands : 1999) (05.07.2016)
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Journal Article
SB226, an inhibitor of tubulin polymerization, inhibits paclitaxel-resistant melanoma growth and spontaneous metastasis
Deng, Shanshan, Banerjee, Souvik, Chen, Hao, Pochampally, Satyanarayana, Wang, Yuxi, Yun, Mi-Kyung, White, Stephen W., Parmar, Keyur, Meibohm, Bernd, Hartman, Kelli L., Wu, Zhongzhi, Miller, Duane D., Li, Wei
Published in Cancer letters (28.02.2023)
Published in Cancer letters (28.02.2023)
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Journal Article
X‑ray Crystallography-Guided Design, Antitumor Efficacy, and QSAR Analysis of Metabolically Stable Cyclopenta-Pyrimidinyl Dihydroquinoxalinone as a Potent Tubulin Polymerization Inhibitor
Banerjee, Souvik, Mahmud, Foyez, Deng, Shanshan, Ma, Lingling, Yun, Mi-Kyung, Fakayode, Sayo O, Arnst, Kinsie E, Yang, Lei, Chen, Hao, Wu, Zhongzhi, Lukka, Pradeep B, Parmar, Keyur, Meibohm, Bernd, White, Stephen W, Wang, Yuxi, Li, Wei, Miller, Duane D
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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Journal Article
Enantioselective polar‐organic mode high‐performance liquid chromatographic separation of lifitegrast on immobilized polysaccharide stationary phase and its application to pH‐dependent chiral interconversion studies
Kandula, Jony Susanna, Rayala, Veera Venkata Satya Prasanna Kumari, Parmar, Keyur, Ponnapalli, Veerabhadra Swamy, Gantala, Mahendar, P., Radhakrishnanand
Published in Chirality (New York, N.Y.) (01.02.2024)
Published in Chirality (New York, N.Y.) (01.02.2024)
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Journal Article
Comparative study of perioperative morbidities of the conventional and ultrasound-guided suprapubic catheterization in the patients of urinary retention during emergency
Chandra, Mahesh, Parmar, Keyur, Wasnik, Seema
Published in International journal of research in medical sciences (25.09.2019)
Published in International journal of research in medical sciences (25.09.2019)
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Journal Article