Expanding DP4: application to drug compounds and automation
Ermanis, Kristaps, Parkes, Kevin E B, Agback, Tatiana, Goodman, Jonathan M
Published in Organic & biomolecular chemistry (28.04.2016)
Published in Organic & biomolecular chemistry (28.04.2016)
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Journal Article
Discovery of USP7 small-molecule allosteric inhibitors
Engström, Olof, Belda, Oscar, Kullman-Magnusson, Mari, Rapp, Mikaela, Böhm, Kerstin, Paul, Ralf, Henderson, Ian, Derbyshire, Dean, Karlström, Sofia, Parkes, Kevin E.B., Zhao, Hongtao
Published in Bioorganic & medicinal chemistry letters (15.10.2020)
Published in Bioorganic & medicinal chemistry letters (15.10.2020)
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Journal Article
Use of a Pharmacophore Model To Discover a New Class of Influenza Endonuclease Inhibitors
Parkes, Kevin E. B, Ermert, Philipp, Fässler, Jürg, Ives, Jane, Martin, Joseph A, Merrett, John H, Obrecht, Daniel, Williams, Glyn, Klumpp, Klaus
Published in Journal of medicinal chemistry (27.03.2003)
Published in Journal of medicinal chemistry (27.03.2003)
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Journal Article
Two‐metal ion mechanism of RNA cleavage by HIV RNase H and mechanism‐based design of selective HIV RNase H inhibitors
Klumpp, Klaus, Hang, Julie Qi, Rajendran, Surendran, Yang, Yanli, Derosier, Andre, Wong Kai In, Philippe, Overton, Hilary, Parkes, Kevin E. B., Cammack, Nick, Martin, Joseph A.
Published in Nucleic acids research (01.12.2003)
Published in Nucleic acids research (01.12.2003)
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Journal Article
Assessing the Role of Polarization in Docking
Illingworth, Christopher J. R, Morris, Garrett M, Parkes, Kevin E. B, Snell, Christopher R, Reynolds, Christopher A
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (27.11.2008)
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (27.11.2008)
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Journal Article
Connectivity and binding-site recognition: Applications relevant to drug design
Illingworth, Christopher J.R, Scott, Paul D, Parkes, Kevin E.B, Snell, Christopher R, Campbell, Matthew P, Reynolds, Christopher A
Published in Journal of computational chemistry (30.11.2010)
Published in Journal of computational chemistry (30.11.2010)
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Journal Article
Closed loop folding units from structural alignments: Experimental foldons revisited
Chintapalli, Sree V, Yew, Boon K, Illingworth, Christopher J.R, Upton, Graham J.G, Reeves, Philip J, Parkes, Kevin E.B, Snell, Christopher R, Reynolds, Christopher A
Published in Journal of computational chemistry (30.11.2010)
Published in Journal of computational chemistry (30.11.2010)
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Journal Article
Toward a Consistent Treatment of Polarization in Model QM/MM Calculations
Illingworth, Christopher J. R, Parkes, Kevin E. B, Snell, Christopher R, Ferenczy, György G, Reynolds, Christopher A
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (27.11.2008)
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (27.11.2008)
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Journal Article
Criteria for confirming sequence periodicity identified by Fourier transform analysis: Application to GCR2, a candidate plant GPCR?
Illingworth, Christopher J.R., Parkes, Kevin E., Snell, Christopher R., Mullineaux, Philip M., Reynolds, Christopher A.
Published in Biophysical chemistry (01.03.2008)
Published in Biophysical chemistry (01.03.2008)
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Journal Article
Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application
Kesteleyn, Bart, Amssoms, Katie, Schepens, Wim, Hache, Geerwin, Verschueren, Wim, Van De Vreken, Wim, Rombauts, Klara, Meurs, Greet, Sterkens, Patrick, Stoops, Bart, Baert, Lieven, Austin, Nigel, Wegner, Jörg, Masungi, Chantal, Dierynck, Inge, Lundgren, Stina, Jönsson, Daniel, Parkes, Kevin, Kalayanov, Genadiy, Wallberg, Hans, Rosenquist, Åsa, Samuelsson, Bertil, Van Emelen, Kristof, Thuring, Jan Willem
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Journal Article
Activity of the isolated HIV RNase H domain and specific inhibition by N-hydroxyimides
Hang, Julie Qi, Rajendran, Surendran, Yang, Yanli, Li, Yu, Wong Kai In, Philippe, Overton, Hilary, Parkes, Kevin E.B., Cammack, Nick, Martin, Joseph A., Klumpp, Klaus
Published in Biochemical and biophysical research communications (30.04.2004)
Published in Biochemical and biophysical research communications (30.04.2004)
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Journal Article
Rational Design of Peptide-Based HIV Proteinase Inhibitors
Roberts, Noel A., Martin, Joseph A., Kinchington, Derek, Broadhurst, Anne V., Craig, J. Charles, Duncan, Ian B., Galpin, Sarah A., Handa, Balraj K., Kay, John, Kröhn, Antonin, Lambert, Robert W., Merrett, John H., Mills, John S., Kevin E. B. Parkes, Redshaw, Sally, Ritchie, Alison J., Taylor, Debra L., Thomas, Gareth J., Machin, Peter J.
Published in Science (American Association for the Advancement of Science) (20.04.1990)
Published in Science (American Association for the Advancement of Science) (20.04.1990)
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Journal Article
Nucleoside Analogues as Highly Potent and Selective Inhibitors of Herpes Simplex Virus Thymidine Kinase
Martin, Joseph A, Lambert, Robert W, Merrett, John H, Parkes, Kevin E.B, Thomas, Gareth J, Baker, Stewart J, Bushnell, David J, Cansfield, Julie E, Dunsdon, Stephen J, Freeman, Andrew C, Hopkins, Richard A, Johns, Ian R, Keech, Elizabeth, Simmonite, Heather, Walmsley, Andrea, Wong Kai-In, Philippe, Holland, Mark
Published in Bioorganic & medicinal chemistry letters (09.07.2001)
Published in Bioorganic & medicinal chemistry letters (09.07.2001)
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Journal Article
Radical-polar crossover reactions with a water-soluble tetrathiafulvalene derivative
Patro, Balaram, Merrett, Martin C, Makin, Scott D, Murphy, John A, Parkes, Kevin E.B
Published in Tetrahedron letters (15.01.2000)
Published in Tetrahedron letters (15.01.2000)
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Journal Article
Studies toward the Large-Scale Synthesis of the HIV Proteinase Inhibitor Ro 31-8959
Parkes, Kevin E. B, Bushnell, David J, Crackett, Peter H, Dunsdon, Stephen J, Freeman, Andrew C, Gunn, Michelle P, Hopkins, Richard A, Lambert, Robert W, Martin, Joseph A
Published in Journal of organic chemistry (01.07.1994)
Published in Journal of organic chemistry (01.07.1994)
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Journal Article
Confident application of a global human liver microsomal activity QSAR
Stålring, Jonna, Sohlenius-Sternbeck, Anna-Karin, Terelius, Ylva, Parkes, Kevin
Published in Future medicinal chemistry (01.07.2018)
Published in Future medicinal chemistry (01.07.2018)
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