Ligand-binding dynamics rewire cellular signaling via estrogen receptor-α
Srinivasan, Sathish, Nwachukwu, Jerome C, Parent, Alex A, Cavett, Valerie, Nowak, Jason, Hughes, Travis S, Kojetin, Douglas J, Katzenellenbogen, John A, Nettles, Kendall W
Published in Nature chemical biology (01.05.2013)
Published in Nature chemical biology (01.05.2013)
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Ligand-binding dynamics rewire cellular signaling via estrogen receptor-[alpha]
Srinivasan, Sathish, Nwachukwu, Jerome C, Parent, Alex A, Cavett, Valerie, Nowak, Jason, Hughes, Travis S, Kojetin, Douglas J, Katzenellenbogen, John A, Nettles, Kendall W
Published in Nature chemical biology (06.05.2013)
Published in Nature chemical biology (06.05.2013)
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Sting-Mediated Interferon Signaling Exerts Potent Antileukemic Effects in High-Risk Myeloid and Monocytic Malignancies
Wei, Yue, Li, Ziyi, Yang, Hui, Zheng, Hong, Appleman, Vicky, Hatten, Tiquella, Huang, Yu-Chung, Raizer, Jeffrey, Parent, Alex, Lineberry, Neil, Garcia-Manero, Guillermo, Montalban-Bravo, Guillermo
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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Abstract 6734: Preclinical impact of pretreatment with CRS mitigation agents on pharmacodynamic response to TAK-500, a systemically delivered CCR2-targeted STING agonist iADC
Rosentrater, Emily, Ganno, Michelle L., Hatten, Tiquella, Mack, Henry, Bollampalli, Arjun Reddy, Zhang, Dong Mei, Parent, Alex, Raizer, Jeffrey, Gregory, Richard C., Lineberry, Neil, Appleman, Vicky
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract 6732: Immunomodulatory and anti-tumor effect of a CCR2-targeted STING agonist iADC in human lung cancer
Porciuncula, Angelo, Appleman, Vicky A., Parent, Alex, Raizer, Jeff, Gregory, Richard C., Lineberry, Neil, Abu-Yousif, Adnan O., Schalper, Kurt A.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Resveratrol modulates the inflammatory response via an estrogen receptor-signal integration network
Nwachukwu, Jerome C, Srinivasan, Sathish, Bruno, Nelson E, Parent, Alexander A, Hughes, Travis S, Pollock, Julie A, Gjyshi, Olsi, Cavett, Valerie, Nowak, Jason, Garcia-Ordonez, Ruben D, Houtman, René, Griffin, Patrick R, Kojetin, Douglas J, Katzenellenbogen, John A, Conkright, Michael D, Nettles, Kendall W
Published in eLife (25.04.2014)
Published in eLife (25.04.2014)
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Coupling of receptor conformation and ligand orientation determine graded activity
Nettles, Kendall W, Bruning, John B, Parent, Alexander A, Gil, German, Zhao, Min, Nowak, Jason, Pace, Margaret C, Smith, Carolyn L, Afonine, Pavel V, Adams, Paul D, Katzenellenbogen, John A
Published in Nature chemical biology (01.11.2010)
Published in Nature chemical biology (01.11.2010)
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Abstract 1841: TAK-500 is a clinical stage immune-cell directed antibody drug conjugate (iADC) inducing STING activation in CCR2-expressing intratumor myeloid cells and favorable immunomodulation
Schalper, Kurt A., Matsuda, Atsushi, Ganno-Sherwood, Michelle, Maldonado-Lopez, Angel E., Rosentrater, Emily, Porciuncula, Angelo, Zhang, Dong Mei, Christensen, Camilla L., Merrigan, Samantha A., Hatten, Tiquella, Lee, Hong Myung, Lee, Min Young, Dong, Linlin, Huang, Jian, Iartchouk, Natasha, Wang, Jianing, Xu, He, Yoneyama, Tomoki, Piatkov, Konstantin I., Harbison, Carole E., Parent, Alex, Lineberry, Neil, Abu-Yousif, Adnan O., Appleman, Vicky
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Estimating the cost of generic quantum pre-image attacks on SHA-2 and SHA-3
Matthew, Amy, Olivia Di Matteo, Gheorghiu, Vlad, Mosca, Michele, Parent, Alex, Schanck, John
Published in arXiv.org (30.11.2016)
Published in arXiv.org (30.11.2016)
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