Constitutively Elevated Blood Serotonin Is Associated with Bone Loss and Type 2 Diabetes in Rats
Erjavec, Igor, Bordukalo-Niksic, Tatjana, Brkljacic, Jelena, Grcevic, Danka, Mokrovic, Gordana, Kesic, Maja, Rogic, Dunja, Zavadoski, William, Paralkar, Vishwas M, Grgurevic, Lovorka, Trkulja, Vladimir, Cicin-Sain, Lipa, Vukicevic, Slobodan
Published in PloS one (23.02.2016)
Published in PloS one (23.02.2016)
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The application of target information and preclinical pharmacokinetic/pharmacodynamic modeling in predicting clinical doses of a Dickkopf-1 antibody for osteoporosis
Betts, Alison M, Clark, Tracey H, Yang, Jianxin, Treadway, Judith L, Li, Mei, Giovanelli, Michael A, Abdiche, Yasmina, Stone, Donna M, Paralkar, Vishwas M
Published in The Journal of pharmacology and experimental therapeutics (01.04.2010)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2010)
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Proline-rich tyrosine kinase 2 regulates osteoprogenitor cells and bone formation, and offers an anabolic treatment approach for osteoporosis
Buckbinder, Leonard, Crawford, David T, Qi, Hong, Ke, Hua Zhu, Olson, Lisa M, Long, Kelly R, Bonnette, Peter C, Baumann, Amy P, Hambor, John E, Grasser, William A. III, Pan, Lydia C, Owen, Thomas A, Luzzio, Michael J, Hulford, Catherine A, Gebhard, David F, Paralkar, Vishwas M, Simmons, Hollis A, Kath, John C, Roberts, W. Gregory, Smock, Steven L, Guzman-Perez, Angel, Brown, Thomas A, Li, Mei
Published in Proceedings of the National Academy of Sciences - PNAS (19.06.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (19.06.2007)
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Tumor-selective, antigen-independent delivery of a pH sensitive peptide-topoisomerase inhibitor conjugate suppresses tumor growth without systemic toxicity
Gayle, Sophia, Aiello, Robert, Leelatian, Nalin, Beckta, Jason M, Bechtold, Jane, Bourassa, Patricia, Csengery, Johanna, Maguire, Robert J, Marshall, Dan, Sundaram, Ranjini K, Van Doorn, Jinny, Jones, Kelli, Moore, Hunter, Lopresti-Morrow, Lori, Paradis, Timothy, Tylaska, Laurie, Zhang, Qing, Visca, Hannah, Reshetnyak, Yana K, Andreev, Oleg A, Engelman, Donald M, Glazer, Peter M, Bindra, Ranjit S, Paralkar, Vishwas M
Published in NAR cancer (01.06.2021)
Published in NAR cancer (01.06.2021)
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Anoxia induces macrophage inhibitory cytokine-1 (MIC-1) in glioblastoma cells independently of p53 and HIF-1
ALBERTONI, Michele, SHAW, Phillip H, VAN MEIR, Erwin G, HEGI, Monika E, NOZAKI, Michimasa, GODARD, Sophie, TENAN, Mirna, HAMOU, Marie-France, FAIRLIE, Douglas W, BREIT, Samuel N, PARALKAR, Vishwas M, DE TRIBOLET, Nicolas
Published in Oncogene (20.06.2002)
Published in Oncogene (20.06.2002)
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A Novel, Non‐Prostanoid EP2 Receptor‐Selective Prostaglandin E2 Agonist Stimulates Local Bone Formation and Enhances Fracture Healing
LI, Mei, KE, Hua Zhu, QI, Hong, Healy, David R, LI, Yan, Crawford, D Todd, Paralkar, Vishwas M, Owen, Thomas A, Cameron, Kimberly O, Lefker, Bruce A, Brown, Thomas A, Thompson, David D
Published in Journal of bone and mineral research (01.11.2003)
Published in Journal of bone and mineral research (01.11.2003)
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Antigen-independent tumor targeting by CBX-12 (alphalex ™ -exatecan) induces long-term antitumor immunity
Gayle, Sophia, Paradis, Timothy, Jones, Kelli, Vasquez, Juan, Paralkar, Vishwas M
Published in Immunotherapy (01.12.2022)
Published in Immunotherapy (01.12.2022)
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A Nonprostanoid EP4 Receptor Selective Prostaglandin E2 Agonist Restores Bone Mass and Strength in Aged, Ovariectomized Rats
Ke, Hua Zhu, Crawford, D Todd, Qi, Hong, Simmons, Hollis A, Owen, Thomas A, Paralkar, Vishwas M, Li, Mei, Lu, Bihong, Grasser, William A, Cameron, Kimberly O, Lefker, Bruce A, DaSilva‐Jardine, Paul, Scott, Dennis O, Zhang, Qing, Tian, Xiao Yan, Jee, Webster SS, Brown, Thomas A, Thompson, David D
Published in Journal of bone and mineral research (01.04.2006)
Published in Journal of bone and mineral research (01.04.2006)
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A novel role of bone morphogenetic protein 6 (BMP6) in glucose homeostasis
Pauk, Martina, Bordukalo-Niksic, Tatjana, Brkljacic, Jelena, Paralkar, Vishwas M., Brault, Amy L., Dumic-Cule, Ivo, Borovecki, Fran, Grgurevic, Lovorka, Vukicevic, Slobodan
Published in Acta diabetologica (01.03.2019)
Published in Acta diabetologica (01.03.2019)
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Circulating Bone Morphogenetic Protein 1-3 Isoform Increases Renal Fibrosis
GRGUREVIC, Lovorka, MACEK, Boris, STERN-PADOVAN, Ranka, PARALKAR, Vishwas M, VUKICEVIC, Slobodan, HEALY, David R, BRAULT, Amy L, ERJAVEC, Igor, CIPCIC, Antonio, GRGUREVIC, Ivica, ROGIC, Dunja, GALESIC, Kresimir, BRKLJACIC, Jelena
Published in Journal of the American Society of Nephrology (01.04.2011)
Published in Journal of the American Society of Nephrology (01.04.2011)
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Deletion of the P2X7 Nucleotide Receptor Reveals Its Regulatory Roles in Bone Formation and Resorption
Ke, Hua Zhu, Qi, Hong, Weidema, A. Frederik, Zhang, Qing, Panupinthu, Nattapon, Crawford, D. Todd, Grasser, William A, Paralkar, Vishwas M, Li, Mei, Audoly, Laurent P, Gabel, Christopher A, Jee, Webster S. S, Dixon, S. Jeffrey, Sims, Stephen M, Thompson, David D
Published in Molecular endocrinology (Baltimore, Md.) (01.07.2003)
Published in Molecular endocrinology (Baltimore, Md.) (01.07.2003)
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The discovery of novel calcium sensing receptor negative allosteric modulators
Balan, Gayatri, Bauman, Jonathan, Bhattacharya, Samit, Castrodad, Mayda, Healy, David R., Herr, Michael, Humphries, Paul, Jennings, Sandra, Kalgutkar, Amit S., Kapinos, Brendon, Khot, Vishal, Lazarra, Kimberly, Li, Mei, Li, Yan, Neagu, Constantin, Oliver, Robert, Piotrowski, David W., Price, David, Qi, Hong, Simmons, Holly A., Southers, James, Wei, Liuqing, Zhang, Yan, Paralkar, Vishwas M.
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
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Discovery of CP-533536 : An EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation
CAMERON, Kimberly O, LEFKER, Bruce A, LI YU, THOMPSON, David D, KE, Hua Z, MEI LI, ZAWISTOSKI, Michael P, TJOA, Christina M, WRIGHT, Ann S, DENINNO, Shari L, PARALKAR, Vishwas M, OWEN, Thomas A
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Short-acting 5-(trifluoromethyl)pyrido[4,3- d]pyrimidin-4(3 H)-one derivatives as orally-active calcium-sensing receptor antagonists
Didiuk, Mary T., Griffith, David A., Benbow, John W., Liu, Kevin K.C., Walker, Daniel P., Christopher Bi, F., Morris, Joel, Guzman-Perez, Angel, Gao, Hua, Bechle, Bruce M., Kelley, Ryan M., Yang, Xiaojing, Dirico, Kenneth, Ahmed, Syed, Hungerford, William, DiBrinno, Joseph, Zawistoski, Michael P., Bagley, Scott W., Li, Jianke, Zeng, Yuan, Santucci, Stephanie, Oliver, Robert, Corbett, Matthew, Olson, Thanh, Chen, Chiliu, Li, Mei, Paralkar, Vishwas M., Riccardi, Keith A., Healy, David R., Kalgutkar, Amit S., Maurer, Tristan S., Nguyen, Hang T., Frederick, Kosea S.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Effects of CP-336,156, a New, Nonsteroidal Estrogen Agonist/Antagonist, on Bone, Serum Cholesterol, Uterus, and Body Composition in Rat Models
Ke, Hua Zhu, Paralkar, Vishwas M, Grasser, William A, Crawford, D. Todd, Qi, Hong, Simmons, Hollis A, Pirie, Christine M, Chidsey-Frink, Kristin L, Owen, Thomas A, Smock, Steven L, Chen, Hong Ka, Jee, Webster S. S, Cameron, Kimberly O, Rosati, Robert L, Brown, Thomas A, Dasilva-Jardine, Paul, Thompson, David D
Published in Endocrinology (Philadelphia) (01.04.1998)
Published in Endocrinology (Philadelphia) (01.04.1998)
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Metabolism-Guided Design of Short-Acting Calcium-Sensing Receptor Antagonists
Southers, James A, Bauman, Jonathan N, Price, David A, Humphries, Paul S, Balan, Gayatri, Sagal, John F, Maurer, Tristan S, Zhang, Yan, Oliver, Robert, Herr, Michael, Healy, David R, Li, Mei, Kapinos, Brendon, Fate, Gwendolyn D, Riccardi, Keith A, Paralkar, Vishwas M, Brown, Thomas A, Kalgutkar, Amit S
Published in ACS medicinal chemistry letters (12.08.2010)
Published in ACS medicinal chemistry letters (12.08.2010)
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Discovery of highly selective EP4 receptor agonists that stimulate new bone formation and restore bone mass in ovariectomized rats
Cameron, Kimberly O., Lefker, Bruce A., Chu-Moyer, Margaret Y., Crawford, David T., Jardine, Paul DaSilva, DeNinno, Shari L., Gilbert, Sandra, Grasser, William A., Ke, HuaZhu, Lu, Bihong, Owen, Thomas A., Paralkar, Vishwas M., Qi, Hong, Scott, Dennis O., Thompson, David D., Tjoa, Christina M., Zawistoski, Michael P.
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Recombinant Human Bone Morphogenetic Protein 2B Stimulates PC12 Cell Differentiation: Potentiation and Binding to Type IV Collagen
Paralkar, Vishwas M., Weeks, Benjamin S., Yu M. Yu, Kleinman, Hynda K., Reddi, A. Hari
Published in The Journal of cell biology (01.12.1992)
Published in The Journal of cell biology (01.12.1992)
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DNA sequence motifs are associated with aberrant homologous recombination in the mouse macrophage migration inhibitory factor (Mif) locus
Kobayashi, Shigetoshi, Yoshida, Kunihiro, Ohshima, Toshio, Esumi, Noriko, Paralkar, Vishwas M, Wistow, Graeme J, Kulkarni, Ashok B
Published in Gene (17.07.1998)
Published in Gene (17.07.1998)
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Cloning and Characterization of a Novel Member of the Transforming Growth Factor-β/Bone Morphogenetic Protein Family
Paralkar, Vishwas M., Vail, Amy L., Grasser, William A., Brown, Thomas A., Xu, Hong, Vukicevic, Slobodan, Ke, Hua Zhu, Qi, Hong, Owen, Thomas A., Thompson, David D.
Published in The Journal of biological chemistry (29.05.1998)
Published in The Journal of biological chemistry (29.05.1998)
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