From Inhibition to Degradation: Targeting the Antiapoptotic Protein Myeloid Cell Leukemia 1 (MCL1)
Papatzimas, James W, Gorobets, Evgueni, Maity, Ranjan, Muniyat, Mir Ishruna, MacCallum, Justin L, Neri, Paola, Bahlis, Nizar J, Derksen, Darren J
Published in Journal of medicinal chemistry (13.06.2019)
Published in Journal of medicinal chemistry (13.06.2019)
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Journal Article
Pannexin-1 channel inhibition alleviates opioid withdrawal in rodents by modulating locus coeruleus to spinal cord circuitry
Kwok, Charlie H. T., Harding, Erika K., Burma, Nicole E., Markovic, Tamara, Massaly, Nicolas, van den Hoogen, Nynke J., Stokes-Heck, Sierra, Gambeta, Eder, Komarek, Kristina, Yoon, Hye Jean, Navis, Kathleen E., McAllister, Brendan B., Canet-Pons, Julia, Fan, Churmy, Dalgarno, Rebecca, Gorobets, Evgueni, Papatzimas, James W., Zhang, Zizhen, Kohro, Yuta, Anderson, Connor L., Thompson, Roger J., Derksen, Darren J., Morón, Jose A., Zamponi, Gerald W., Trang, Tuan
Published in Nature communications (24.07.2024)
Published in Nature communications (24.07.2024)
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Journal Article
DCAF16-Based Covalent Handle for the Rational Design of Monovalent Degraders
Lim, Melissa, Cong, Thang Do, Orr, Lauren M., Toriki, Ethan S., Kile, Andrew C., Papatzimas, James W., Lee, Elijah, Lin, Yihan, Nomura, Daniel K.
Published in ACS central science (24.07.2024)
Published in ACS central science (24.07.2024)
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Journal Article
Correction to “Rational Chemical Design of Molecular Glue Degraders”
Toriki, Ethan S., Papatzimas, James W., Nishikawa, Kaila, Dovala, Dustin, Frank, Andreas O., Hesse, Matthew J., Dankova, Daniela, Song, Jae-Geun, Bruce-Smythe, Megan, Struble, Heidi, Garcia, Francisco J., Brittain, Scott M., Kile, Andrew C., McGregor, Lynn M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in ACS central science (23.08.2023)
Published in ACS central science (23.08.2023)
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Journal Article
ADAM protease inhibition overcomes resistance of breast cancer stem-like cells to γδ T cell immunotherapy
Dutta, Indrani, Dieters-Castator, Dylan, Papatzimas, James W., Medina, Anais, Schueler, Julia, Derksen, Darren J., Lajoie, Gilles, Postovit, Lynne-Marie, Siegers, Gabrielle M.
Published in Cancer letters (01.01.2021)
Published in Cancer letters (01.01.2021)
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Journal Article
A vinylogous Norrish reaction as a strategy for light-mediated ring expansion
Gorobets, Evgueni, Papatzimas, James W, Dourado, Jorge, Yousefalizadeh, Goonay, Lee, JinGyu, Brownsey, Duncan K, Stamplecoskie, Kevin, Davis, Rebecca, Derksen, Darren J
Published in Chemical communications (Cambridge, England) (24.02.2022)
Published in Chemical communications (Cambridge, England) (24.02.2022)
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Journal Article
Rational Chemical Design of Molecular Glue Degraders
Toriki, Ethan S., Papatzimas, James W., Nishikawa, Kaila, Dovala, Dustin, Frank, Andreas O., Hesse, Matthew J., Dankova, Daniela, Song, Jae-Geun, Bruce-Smythe, Megan, Struble, Heidi, Garcia, Francisco J., Brittain, Scott M., Kile, Andrew C., McGregor, Lynn M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in ACS central science (24.05.2023)
Published in ACS central science (24.05.2023)
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Journal Article
Thiaporphyrin-mediated photocatalysis using red light
Lee, JinGyu, Papatzimas, James W., Bromby, Ashley D., Gorobets, Evgueni, Derksen, Darren J.
Published in RSC advances (01.01.2016)
Published in RSC advances (01.01.2016)
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Journal Article
Identification of ligand linkage vectors for the development of p300/CBP degraders
Brownsey, Duncan K, Rowley, Ben C, Gorobets, Evgueni, Mihara, Koichiro, Maity, Ranjan, Papatzimas, James W, Gelfand, Benjamin S, Hollenberg, Morley D, Bahlis, Nizar J, Derksen, Darren J
Published in MedChemComm (22.06.2022)
Published in MedChemComm (22.06.2022)
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Journal Article
A General Strategy for the Preparation of Thalidomide-Conjugate Linkers
Papatzimas, James W., Gorobets, Evgueni, Brownsey, Duncan K., Maity, Ranjan, Bahlis, Nizar J., Derksen, Darren J.
Published in Synlett (18.12.2017)
Published in Synlett (18.12.2017)
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