The Joint European Compound Library: boosting precompetitive research
Besnard, Jérémy, Jones, Philip S., Hopkins, Andrew L., Pannifer, Andrew D.
Published in Drug discovery today (01.02.2015)
Published in Drug discovery today (01.02.2015)
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Design and Structure of Stapled Peptides Binding to Estrogen Receptors
Phillips, Chris, Roberts, Lee R, Schade, Markus, Bazin, Richard, Bent, Andrew, Davies, Nichola L, Moore, Rob, Pannifer, Andrew D, Pickford, Andrew R, Prior, Stephen H, Read, Christopher M, Scott, Andrew, Brown, David G, Xu, Bin, Irving, Stephen L
Published in Journal of the American Chemical Society (29.06.2011)
Published in Journal of the American Chemical Society (29.06.2011)
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The European Lead Factory: Results from a decade of collaborative, public–private, drug discovery programs
van Vlijmen, Herman, Pannifer, Andrew D., Cochrane, Phil, Basting, Daniel, Li, Volkhart M, Engkvist, Ola, Ortholand, Jean-Yves, Wagener, Markus, Duffy, James, Finsinger, Dirk, Davis, Jeremy, van Helden, Steven P., de Vlieger, Jon S.B.
Published in Drug discovery today (01.03.2024)
Published in Drug discovery today (01.03.2024)
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The ELF Honest Data Broker: informatics enabling public–private collaboration in a precompetitive arena
Paillard, Guillaume, Cochrane, Philip, Jones, Philip S., van Hoorn, Willem P., Caracoti, Andrei, van Vlijmen, Herman, Pannifer, Andrew D.
Published in Drug discovery today (01.01.2016)
Published in Drug discovery today (01.01.2016)
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IMI European Lead Factory - democratizing access to high-throughput screening
Jones, Philip S, Boucharens, Sylviane, McElroy, Stuart P, Morrison, Angus, Honarnejad, Saman, van Boeckel, Stan, van den Hurk, Helma, Basting, Daniel, Hüser, Jörg, Jaroch, Stefan, Ottow, Eckhard, Benningshof, Jorg, Folmer, Rutger H A, Leemhuis, Frank, Kramer-Verhulst, Patricia M, Nies, Vera J M, Orrling, Kristina M, Rijnders, Ton, Pfander, Claudia, Engkvist, Ola, Pairaudeau, Garry, Simpson, Peter B, Ortholand, Jean-Yves, Roche, Didier, Dömling, Alexander, Kühnert, Sven M, Roevens, Peter W M, van Vlijmen, Herman, van Wanrooij, Eva J A, Verbruggen, Christophe, Nussbaumer, Peter, Ovaa, Huib, van der Stelt, Mario, Simonsen, Klaus Baek, Tagmose, Lena, Waldmann, Herbert, Duffy, James, Finsinger, Dirk, Jurzak, Mirek, Burgess-Brown, Nicola A, Lee, Wen H, Rutjes, Floris P J T, Haag, Hubert, Kallus, Christopher, Mors, Hartmut, Dorval, Thierry, Lesur, Brigitte, Ramon Olayo, Fernando, Hamza, Daniel, Jones, Geraint, Pearce, Christopher, Piechot, Alexander, Tzalis, Dimitrios, Clausen, Mads H, Davis, Jeremy, Derouane, Daphné, Vermeiren, Céline, Kaiser, Markus, Stockman, Robert A, Barrault, Denise V, Pannifer, Andrew D, Swedlow, Jason R, Nelson, Adam S, Orru, Romano V A, Ruijter, Eelco, van Helden, Steven P, Li, Volkhart M, Vries, Ton, de Vlieger, Jon S B
Published in Nature reviews. Drug discovery (01.04.2022)
Published in Nature reviews. Drug discovery (01.04.2022)
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Journal Article
Crystal structure of the anthrax lethal factor
Liddington, Robert C, Pannifer, Andrew D, Wong, Thiang Yian, Schwarzenbacher, Robert, Renatus, Martin, Petosa, Carlo, Bienkowska, Jadwiga, Lacy, D. Borden, Collier, R. John, Park, Sukjoon, Leppla, Stephen H, Hanna, Philip
Published in Nature (London) (08.11.2001)
Published in Nature (London) (08.11.2001)
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Journal Article
Identification of A Novel Class of Benzofuran Oxoacetic Acid-Derived Ligands that Selectively Activate Cellular EPAC1
Beck, Elizabeth M, Parnell, Euan, Cowley, Angela, Porter, Alison, Gillespie, Jonathan, Robinson, John, Robinson, Lindsay, Pannifer, Andrew D, Hamon, Veronique, Jones, Philip, Morrison, Angus, McElroy, Stuart, Timmerman, Martin, Rutjes, Helma, Mahajan, Pravin, Wiejak, Jolanta, Luchowska-Stańska, Urszula, Morgan, David, Barker, Graeme, Rehmann, Holger, Yarwood, Stephen J
Published in Cells (Basel, Switzerland) (12.11.2019)
Published in Cells (Basel, Switzerland) (12.11.2019)
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SAR and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors
Heron, Nicola M., Anderson, Malcolm, Blowers, David P., Breed, Jason, Eden, Jonathan M., Green, Stephen, Hill, George B., Johnson, Trevor, Jung, Frederic H., McMiken, Helen H.J., Mortlock, Andrew A., Pannifer, Andrew D., Pauptit, Richard A., Pink, Jennifer, Roberts, Nicola J., Rowsell, Siân
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Structure-based design of protein tyrosine phosphatase-1B inhibitors
Black, Emma, Breed, Jason, Breeze, Alexander L., Embrey, Kevin, Garcia, Robert, Gero, Thomas W., Godfrey, Linda, Kenny, Peter W., Morley, Andrew D., Minshull, Claire A., Pannifer, Andrew D., Read, Jon, Rees, Amanda, Russell, Daniel J., Toader, Dorin, Tucker, Julie
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
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Journal Article
Novel thienopyrrole glycogen phosphorylase inhibitors: Synthesis, in vitro SAR and crystallographic studies
Whittamore, Paul R.O., Addie, Matthew S., Bennett, Stuart N.L., Birch, Alan M., Butters, Michael, Godfrey, Linda, Kenny, Peter W., Morley, Andrew D., Murray, Paul M., Oikonomakos, Nikos G., Otterbein, Ludovic R., Pannifer, Andrew D., Parker, Jeremy S., Readman, Kristy, Siedlecki, Pawel S., Schofield, Paul, Stocker, Andy, Taylor, Melvyn J., Townsend, Linda A., Whalley, David P., Whitehouse, Jennifer
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
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Imitation of beta-lactam binding enables broad-spectrum metallo-beta-lactamase inhibitors
Brem, Jurgen, Panduwawala, Tharindi, Hansen, Jon Ulf, Hewitt, Joanne, Liepins, Edgars, Donets, Pawel, Espina, Laura, Farley, Alistair J. M., Shubin, Kirill, Campillos, Gonzalo Gomez, Kiuru, Paula, Shishodia, Shifali, Krahn, Daniel, Lesniak, Robert K., Schmidt (Adrian), Juliane, Calvopina, Karina, Turrientes, Maria-Carmen, Kavanagh, Madeline E., Lubriks, Dmitrijs, Hinchliffe, Philip, Langley, Gareth W., Aboklaish, Ali F., Eneroth, Anders, Backlund, Maria, Baran, Andrei G., Nielsen, Elisabet, Speake, Michael, Kuka, Janis, Robinson, John, Grinberga, Solveiga, Robinson, Lindsay, McDonough, Michael A., Rydzik, Anna M., Leissing, Thomas M., Jimenez-Castellanos, Juan Carlos, Avison, Matthew B., Pinto, Solange Da Silva, Pannifer, Andrew D., Martjuga, Marina, Widlake, Emma, Priede, Martins, Navratilova, Iva Hopkins, Gniadkowski, Marek, Belfrage, Anna Karin, Brandt, Peter, Yli-Kauhaluoma, Jari, Bacque, Eric, Page, Malcolm G. P., Bjorkling, Fredrik, Tyrrell, Jonathan M., Spencer, James, Lang, Pauline A., Baranczewski, Pawel, Canton, Rafael, McElroy, Stuart P., Jones, Philip S., Baquero, Fernando, Suna, Edgars, Morrison, Angus, Walsh, Timothy R., Schofield, Christopher J.
Published in Nature chemistry (01.01.2022)
Published in Nature chemistry (01.01.2022)
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Structural Insights into a Unique Inhibitor Binding Pocket in Kinesin Spindle Protein
Ulaganathan, Venkatasubramanian, Talapatra, Sandeep K, Rath, Oliver, Pannifer, Andrew, Hackney, David D, Kozielski, Frank
Published in Journal of the American Chemical Society (13.02.2013)
Published in Journal of the American Chemical Society (13.02.2013)
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Structure-based design, synthesis and biological evaluation of a novel series of isoquinolone and pyrazolo[4,3-c]pyridine inhibitors of fascin 1 as potential anti-metastatic agents
Francis, Stuart, Croft, Daniel, Schüttelkopf, Alexander W., Parry, Charles, Pugliese, Angelo, Cameron, Ken, Claydon, Sophie, Drysdale, Martin, Gardner, Claire, Gohlke, Andrea, Goodwin, Gillian, Gray, Christopher H., Konczal, Jennifer, McDonald, Laura, Mezna, Mokdad, Pannifer, Andrew, Paul, Nikki R., Machesky, Laura, McKinnon, Heather, Bower, Justin
Published in Bioorganic & medicinal chemistry letters (15.04.2019)
Published in Bioorganic & medicinal chemistry letters (15.04.2019)
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Journal Article
The importance of triaging in determining the quality of output from high-throughput screening
Jones, Philip, McElroy, Stuart, Morrison, Angus, Pannifer, Andrew
Published in Future medicinal chemistry (01.01.2015)
Published in Future medicinal chemistry (01.01.2015)
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Abstract LB-B17: Characterization of small molecule inhibitors of the Nrf2-Keap1 interaction using MicroScale Thermophoresis
Rainard, Julie M., Morrison, Angus J., Pannifer, Andrew D., Jones, Philip S., Mead, Richard J., McElroy, Stuart P.
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Synthesis and Structure‐Activity Relationships of N‐(4‐Benzamidino)‐Oxazolidinones: Potent and Selective Inhibitors of Kallikrein‐Related Peptidase 6
De Vita, Elena, Smits, Niels, Hurk, Helma, Beck, Elizabeth M., Hewitt, Joanne, Baillie, Gemma, Russell, Emily, Pannifer, Andrew, Hamon, Véronique, Morrison, Angus, McElroy, Stuart P., Jones, Philip, Ignatenko, Natalia A., Gunkel, Nikolas, Miller, Aubry K.
Published in ChemMedChem (07.01.2020)
Published in ChemMedChem (07.01.2020)
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A novel small-molecule MRCK inhibitor blocks cancer cell invasion
Unbekandt, Mathieu, Croft, Daniel R, Crighton, Diane, Mezna, Mokdad, McArthur, Duncan, McConnell, Patricia, Schüttelkopf, Alexander W, Belshaw, Simone, Pannifer, Andrew, Sime, Mairi, Bower, Justin, Drysdale, Martin, Olson, Michael F
Published in Cell communication and signaling (05.10.2014)
Published in Cell communication and signaling (05.10.2014)
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THE IDENTIFICATION AND CHARACTERISATION OF SMALL-MOLECULE HUMAN ABAD INHIBITORS AS THERAPEUTICS IN ALZHEIMER’S DISEASE
Aitken, Laura, Baillie, Gemma, Sethi, Ritika, Robinson, John S., Rajamanickam, Muralikrishnan, Pannifer, Andrew, Morrison, Angus, Jones, Philip S., Smith, Terry K., McElroy, Stuart P., Gunn-Moore, Frank J.
Published in Alzheimer's & dementia (01.07.2017)
Published in Alzheimer's & dementia (01.07.2017)
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