Site recognition and substrate screens for PKN family proteins
Collazos, Alejandra, Michael, Nicholas, Whelan, Richard D H, Kelly, Gavin, Mellor, Harry, Pang, Leon C H, Totty, Nick, Parker, Peter J
Published in Biochemical journal (15.09.2011)
Published in Biochemical journal (15.09.2011)
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Identification of a novel orally bioavailable ERK5 inhibitor with selectivity over p38α and BRD4
Myers, Stephanie M., Miller, Duncan C., Molyneux, Lauren, Arasta, Mercedes, Bawn, Ruth H., Blackburn, Timothy J., Cook, Simon J., Edwards, Noel, Endicott, Jane A., Golding, Bernard T., Griffin, Roger J., Hammonds, Tim, Hardcastle, Ian R., Harnor, Suzannah J., Heptinstall, Amy B., Lochhead, Pamela A., Martin, Mathew P., Martin, Nick C., Newell, David R., Owen, Paul J., Pang, Leon C., Reuillon, Tristan, Rigoreau, Laurent J.M., Thomas, Huw D., Tucker, Julie A., Wang, Lan-Zhen, Wong, Ai-Ching, Noble, Martin E.M., Wedge, Stephen R., Cano, Celine
Published in European journal of medicinal chemistry (15.09.2019)
Published in European journal of medicinal chemistry (15.09.2019)
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Co-crystal structures of inhibitors with MRCKβ, a key regulator of tumor cell invasion
Heikkila, Timo, Wheatley, Edward, Crighton, Diane, Schroder, Ewald, Boakes, Alexandra, Kaye, Sarah J, Mezna, Mokdad, Pang, Leon, Rushbrooke, Mathew, Turnbull, Andrew, Olson, Michael F
Published in PloS one (20.09.2011)
Published in PloS one (20.09.2011)
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Discovery of potent inhibitors of the lyso phospholipase autotaxin
Shah, Pritom, Cheasty, Anne, Foxton, Caroline, Raynham, Tony, Farooq, Muddasar, Gutierrez, Irene Farre, Lejeune, Aurore, Pritchard, Michelle, Turnbull, Andrew, Pang, Leon, Owen, Paul, Boyd, Susan, Stowell, Alexandra, Jordan, Allan, Hamilton, Niall M., Hitchin, James R., Stockley, Martin, MacDonald, Ellen, Quesada, Mar Jimenez, Trivier, Elisabeth, Skeete, Jana, Ovaa, Huib, Moolenaar, Wouter H., Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
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Journal Article
Discovery of potent inhibitors of the lysophospholipase autotaxin
Shah, Pritom, Cheasty, Anne, Foxton, Caroline, Raynham, Tony, Farooq, Muddasar, Gutierrez, Irene Farre, Lejeune, Aurore, Pritchard, Michelle, Turnbull, Andrew, Pang, Leon, Owen, Paul, Boyd, Susan, Stowell, Alexandra, Jordan, Allan, Hamilton, Niall M., Hitchin, James R., Stockley, Martin, MacDonald, Ellen, Quesada, Mar Jimenez, Trivier, Elisabeth, Skeete, Jana, Ovaa, Huib, Moolenaar, Wouter H., Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (15.11.2016)
Published in Bioorganic & medicinal chemistry letters (15.11.2016)
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Abstract LB-99: Identification and characterization of small molecule thieno[3,2-d]pyrimidine inhibitors of Protein Kinase C iota (PKCι)
Soudy, Christelle, Stanway, Emma, Patel, Bhavisha, Barton, Caroline, Barnard, Michelle, Pang, Leon, Owen, Paul, Turnbull, Andrew, Ruggeri, Bruce A., Dorsey, Bruce D., Ator, Mark A., Ott, Greg R., Linch, Mark, Riou, Philippe, Parker, Peter J., Kjaer, Sven, Dillon, Christian, McDonald, Neil Q., Roffey, Jon
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Co-Crystal Structures of Inhibitors with MRCK[beta], a Key Regulator of Tumor Cell Invasion
Heikkila, Timo, Wheatley, Edward, Crighton, Diane, Schroder, Ewald, Boakes, Alexandra, Kaye, Sarah J, Mezna, Mokdad, Pang, Leon, Rushbrooke, Mathew, Turnbull, Andrew, Olson, Michael F
Published in PloS one (20.09.2011)
Published in PloS one (20.09.2011)
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Journal Article