Miramides A–D: Identification of Detoxin-like Depsipeptides after Heterologous Expression of a Hybrid NRPS-PKS Gene Cluster from Streptomyces mirabilis Lu17588
Paulus, Constanze, Myronovskyi, Maksym, Zapp, Josef, Rodríguez Estévez, Marta, Lopatniuk, Maria, Rosenkränzer, Birgit, Palusczak, Anja, Luzhetskyy, Andriy
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Published in Microorganisms (Basel) (30.08.2022)
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2- and 3-[(Aryl)(azolyl)methyl]indoles as Potential Non-steroidal Aromatase Inhibitors
Lézé, Marie-Pierre, Borgne, Marc Le, Marchand, Pascal, Loquet, Denis, Kogler, Manuela, Baut, Guillaume Le, Palusczak, Anja, Hartmann, Rolf W.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2004)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2004)
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Loseolamycins: A Group of New Bioactive Alkylresorcinols Produced after Heterologous Expression of a Type III PKS from Micromonospora endolithica
Lasch, Constanze, Gummerlich, Nils, Myronovskyi, Maksym, Palusczak, Anja, Zapp, Josef, Luzhetskyy, Andriy
Published in Molecules (Basel, Switzerland) (09.10.2020)
Published in Molecules (Basel, Switzerland) (09.10.2020)
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Miramides A–D: Identification of Detoxin-like Depsipeptides after Heterologous Expression of a Hybrid NRPS-PKS Gene Cluster from IStreptomyces mirabilis/I Lu17588
Paulus, Constanze, Myronovskyi, Maksym, Zapp, Josef, Rodríguez Estévez, Marta, Lopatniuk, Maria, Rosenkränzer, Birgit, Palusczak, Anja, Luzhetskyy, Andriy
Published in Microorganisms (Basel) (01.08.2022)
Published in Microorganisms (Basel) (01.08.2022)
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Synthesis and biological evaluation of 5-[(aryl)(1H-imidazol-l-yl)methyl]-1H-indoles : Potent and selective aromatase inhibitors
LEZE, Marie-Pierre, LE BORGNE, Marc, PINSON, Patricia, PALUSCZAK, Anja, DUFLOS, Muriel, LE BAUT, Guillaume, HARTMANN, Rolf W
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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A New Class of Nonsteroidal Aromatase Inhibitors: Design and Synthesis of Chromone and Xanthone Derivatives and Inhibition of the P450 Enzymes Aromatase and 17α-Hydroxylase/C17,20-Lyase
Recanatini, Maurizio, Bisi, Alessandra, Cavalli, Andrea, Belluti, Federica, Gobbi, Silvia, Rampa, Angela, Valenti, Piero, Palzer, Martina, Palusczak, Anja, Hartmann, Rolf W
Published in Journal of medicinal chemistry (01.03.2001)
Published in Journal of medicinal chemistry (01.03.2001)
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Synthesis and Evaluation of 17-Aliphatic Heterocycle-Substituted Steroidal Inhibitors of 17α-Hydroxylase/C17−20-Lyase (P450 17)
Hartmann, Rolf W, Hector, Markus, Wachall, Bertil G, Palusczak, Anja, Palzer, Martina, Huch, Volker, Veith, Michael
Published in Journal of medicinal chemistry (16.11.2000)
Published in Journal of medicinal chemistry (16.11.2000)
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Synthesis and biological evaluation of 5-[(aryl)(1 H-imidazol-1-yl)methyl]-1 H-indoles: Potent and selective aromatase inhibitors
Lézé, Marie-Pierre, Le Borgne, Marc, Pinson, Patricia, Palusczak, Anja, Duflos, Muriel, Le Baut, Guillaume, Hartmann, Rolf W.
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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CYP 17 and CYP 19 Inhibitors. Evaluation of Fluorine Effects on the Inhibiting Activity of Regioselectively Fluorinated 1-(Naphthalen-2-ylmethyl)imidazoles
Hartmann, Rolf W., Palusczak, Anja, Lacan, Fabrice, Ricci, Giacomo, Ruzziconi, Renzo
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2004)
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2004)
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Synthesis and Evaluation of a Dimer of 2-(4-Pyridylmethyl)-1-Indanone as a Novel Nonsteroidal Aromatase Inhibitor
Gupta, Ranju, Jindal, Dharam Paul, Jit, Birinder, Narang, Gaurav, Palusczak, Anja, Hartmann, Rolf W.
Published in Archiv der Pharmazie (Weinheim) (01.07.2004)
Published in Archiv der Pharmazie (Weinheim) (01.07.2004)
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Synthesis and study of some new N-substituted imide derivatives as potential anticancer agents
Jindal, Dharam Paul, Bedi, Vikas, Jit, Birinder, Karkra, Nalin, Guleria, Sheetal, Bansal, Ranju, Palusczak, Anja, Hartmann, Rolf W.
Published in Farmaco (Società chimica italiana : 1989) (01.04.2005)
Published in Farmaco (Società chimica italiana : 1989) (01.04.2005)
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Pharmacophore Modeling and in Silico Screening for New P450 19 (Aromatase) Inhibitors
Schuster, Daniela, Laggner, Christian, Steindl, Theodora M., Palusczak, Anja, Hartmann, Rolf W., Langer, Thierry
Published in ChemInform (01.08.2006)
Published in ChemInform (01.08.2006)
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Synthesis and Study of Some New N-Substituted Imide Derivatives as Potential Anticancer Agents
Jindal, Dharam Paul, Bedi, Vikas, Jit, Birinder, Karkra, Nalin, Guleria, Sheetal, Bansal, Ranju, Palusczak, Anja, Hartmann, Rolf W.
Published in ChemInform (06.09.2005)
Published in ChemInform (06.09.2005)
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