On the Bioactive Conformation of NAN-190 (1) and MP3022 (2), 5-HT1A Receptor Antagonists
Paluchowska, Maria H, Mokrosz, Maria J, Bojarski, Andrzej, Wesołowska, Anna, Borycz, Jolanta, Charakchieva-Minol, Sijka, Chojnacka-Wójcik, Ewa
Published in Journal of medicinal chemistry (02.12.1999)
Published in Journal of medicinal chemistry (02.12.1999)
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Spacer conformation in biologically active molecules. Part 2. Structure and conformation of 4-[2-(diphenylmethylamino)ethyl]-1-(2-methoxyphenyl) piperazine and its diphenylmethoxy analog—potential 5-HT1A receptor ligands
Karolak-Wojciechowska, J., Fruziński, A., Czylkowski, R., Paluchowska, M.H., Mokrosz, M.J.
Published in Journal of molecular structure (10.09.2003)
Published in Journal of molecular structure (10.09.2003)
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STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF CENTRAL-NERVOUS-SYSTEM AGENTS .13. 4-[3-(BENZOTRIAZOL-1-YL)PROPYL]-1-(2-METHOXYPHENYL)PIPERAZINE, A NEW PUTATIVE 5-HT1A RECEPTOR ANTAGONIST, AND ITS ANALOGS
MOKROSZ, JL, PALUCHOWSKA, MH, CHOJNACKAWOJCIK, E, FILIP, M, CHARAKCHIEVAMINOL, S, DERENWESOLEK, A, MOKROSZ, MJ
Published in Journal of medicinal chemistry (19.08.1994)
Published in Journal of medicinal chemistry (19.08.1994)
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Structure-activity relationship studies of CNS agents, XIX: Quantitative analysis of the alkyl chain effects on the 5-HT1A and 5-HT2 receptor affinities of 4-alkyl-1-arylpiperazines and their analogs
Mokrosz, J L, Mokrosz, M J, Charakchieva-Minol, S, Paluchowska, M H, Bojarski, A J, Duszyńska, B
Published in Archiv der Pharmazie (Weinheim) (1995)
Published in Archiv der Pharmazie (Weinheim) (1995)
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Structure-activity relationship studies of CNS agents. XII. 1-[4-(4-aryl-1-piperazinyl)butyl]-3,4-dihydro-2(1H)-quinolinones: new 5-HT1A, 5-HT2 and D2 ligands with a potential antipsychotic activity
Mokrosz, J L, Chojnacka-Wójcik, E, Dereń-Wesołek, A, Kłodzińska, A, Maćkowiak, M, Bielecka, Z, Paluchowska, M H
Published in Drug design and discovery (01.04.1994)
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Published in Drug design and discovery (01.04.1994)
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Substitution mode of the amide fragment in some new N-[omega-[4-(2-methoxyphenyl)piperazin-1-yl]alkyl]pyrid-2(1H)-ones and their 5-HT1A/5-HT2A activity
Paluchowska, M H, Bugno, R, Charakchieva-Minol, S, Bojarski, A J, Wesołowska, A
Published in Polish journal of pharmacology (01.07.2001)
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Published in Polish journal of pharmacology (01.07.2001)
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Effect of the amide fragment on 5-HT1A receptor activity of some analogs of MP 3022
Paluchowska, M H, Charakchieva-Minol, S, Tatarczyńska, E, Kłodzińska, A
Published in Polish journal of pharmacology (01.09.1999)
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Published in Polish journal of pharmacology (01.09.1999)
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Effect of linking bridge modifications on the 5-HT1A receptor activity of some 4-(omega-benzotriazol-1-yl)alkyl-1-(2-methoxy-phenyl)piperazines
Paluchowska, M H, Kłodzińska, A, Tatarczyńska, E, Szaro, A, Chojnacka-Wójcik, E
Published in Polish journal of pharmacology (01.07.1998)
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Published in Polish journal of pharmacology (01.07.1998)
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Structures and conformations of 1-aryl-1,4-dihydro-3(2 H )-isoquinolinones
Karolak-Wojciechowska, J., Czylkowski, R., Karczmarzyk, Z., Paluchowska, M.H., Rys, B., Szneler, E., Mokrosz, M.J.
Published in Journal of molecular structure (28.06.2002)
Published in Journal of molecular structure (28.06.2002)
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Structure-intrinsic activity relationship studies in the group of 1-imido/amido substituted 4-(4-arylpiperazin-1-yl) cyclohexane derivatives; new, potent 5-HT1A receptor agents with anxiolytic-like activity
BOJARSKI, Andrzej J, PALUCHOWSKA, Maria H, DUSZYNSKA, Beata, BUGNO, Ryszard, KŁODZINSKA, Aleksandra, TATARCZYNSKA, Ewa, CHOJNACKA-WOJCIK, Ewa
Published in Bioorganic & medicinal chemistry (01.03.2006)
Published in Bioorganic & medicinal chemistry (01.03.2006)
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Active conformation of some arylpiperazine postsynaptic 5-HT1A receptor antagonists
Paluchowska, MH, Bojarski, AJ, Charakchieva-Minol, S, Wesolowska, A
Published in European journal of medicinal chemistry (01.04.2002)
Published in European journal of medicinal chemistry (01.04.2002)
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Pharmacological characterization of MP349, a novel 5-HT1A-receptor antagonist with anxiolytic-like activity, in mice and rats
Wesołowska, Anna, Paluchowska, Maria H, Gołembiowska, Krystyna, Chojnacka-Wójcik, Ewa
Published in Journal of pharmacy and pharmacology (01.04.2003)
Published in Journal of pharmacy and pharmacology (01.04.2003)
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Crystal and Molecular Structure of 4-[ω-(Benzotriazolyl)alkyl]-1-(2-methoxyphenyl)piperazines with a Different Pharmacological Activity
Karolak-Wojciechowska, Janina, Fruziński, Andrzej, Bojarski, Andrzej J., Paluchowska, Maria H., Mokrosz, Maria J.
Published in Archiv der Pharmazie (Weinheim) (01.10.1998)
Published in Archiv der Pharmazie (Weinheim) (01.10.1998)
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Structure-activity relationship studies of CNS agents, Part 32: Effect of structural modifications in 1-arylpiperazine derivatives on alpha(1) -adrenoreceptor affinity
Mokrosz, M J, Paluchowska, M H, Charakchieva-Minol, S, Bień, A
Published in Archiv der Pharmazie (Weinheim) (01.06.1997)
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Published in Archiv der Pharmazie (Weinheim) (01.06.1997)
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Structure-activity relationship studies of CNS agents, XV: N-[omega-(4-aryl-1-piperazinyl)alkyl]-2-oxo-1,2,3,4-tetrahydroquinoline s and -4-oxo-1,2,3,4-tetrahydropyrazino[1,2-a]indoles: new, highly potent 5-HT1A ligands
Mokrosz, J L, Duszyńska, B, Paluchowska, M H
Published in Archiv der Pharmazie (Weinheim) (01.08.1994)
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Published in Archiv der Pharmazie (Weinheim) (01.08.1994)
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Structure-activity relationship studies of central nervous system agents. XIII: 4-[3-(Benzotriazol-1-yl)propyl]-1-(2-methoxyphenyl)piperazine, a new putative 5-HT1A receptor antagonist, and its analogs
MOKROSZ, J. L, PALUCHOWSKA, M. H, CHOJNACKA-WOJCIK, E, FILIP, M, CHARAKCHIEVA-MINOL, S, DEREN-WESOLEK, A, MOKROSZ, M. J
Published in Journal of medicinal chemistry (1994)
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Published in Journal of medicinal chemistry (1994)
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Structure-activity relationship studies of CNS agents, Part 22. A search for new trazodone-like antidepressants: synthesis and preliminary receptor binding studies
Mokrosz, J L, Duszynska, B, Paluchowska, M H, Charakchieva-Minol, S, Mokrosz, M J
Published in Archiv der Pharmazie (Weinheim) (1995)
Published in Archiv der Pharmazie (Weinheim) (1995)
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