Discovery of a Clinical Stage Multi-Kinase Inhibitor Sodium (E)-2-{2-Methoxy-5-[(2′,4′,6′-trimethoxystyrylsulfonyl)methyl]phenylamino}acetate (ON 01910.Na): Synthesis, Structure–Activity Relationship, and Biological Activity
Reddy, M. V. Ramana, Venkatapuram, Padmavathi, Mallireddigari, Muralidhar R, Pallela, Venkat R, Cosenza, Stephen C, Robell, Kimberly A, Akula, Balaiah, Hoffman, Benjamin S, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (22.09.2011)
Published in Journal of medicinal chemistry (22.09.2011)
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Journal Article
Design, synthesis, and biological evaluation of 1-(4-sulfamylphenyl)-3-trifluoromethyl-5-indolyl pyrazolines as cyclooxygenase-2 (COX-2) and lipoxygenase (LOX) inhibitors
Reddy, M.V. Ramana, Billa, Vinay K., Pallela, Venkat R., Mallireddigari, Muralidhar R., Boominathan, Rengasamy, Gabriel, Jerome L., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Changes in behavior and brain acetylcholinesterase activity in mosquito fish, Gambusia affinis in response to the sub-lethal exposure to chlorpyrifos
Rao, J Venkateswara, Begum, Ghousia, Pallela, R, Usman, P K, Rao, R Nageswara
Published in International journal of environmental research and public health (01.12.2005)
Published in International journal of environmental research and public health (01.12.2005)
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Optimized conditions for callus induction, plant regeneration and alkaloids accumulation in stem and shoot tip explants of Phyla nodiflora
Ahmed, A.B.A., Pallela, R., Rao, A.S., Rao, M.V., Mat Taha, R.
Published in Spanish journal of agricultural research : SJAR (01.12.2011)
Published in Spanish journal of agricultural research : SJAR (01.12.2011)
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Discovery of 8‑Cyclopentyl-2-[4-(4-methyl-piperazin-1-yl)-phenylamino]-7-oxo-7,8-dihydro-pyrido[2,3‑d]pyrimidine-6-carbonitrile (7x) as a Potent Inhibitor of Cyclin-Dependent Kinase 4 (CDK4) and AMPK-Related Kinase 5 (ARK5)
Reddy, M. V. Ramana, Akula, Balireddy, Cosenza, Stephen C, Athuluridivakar, Saikrishna, Mallireddigari, Muralidhar R, Pallela, Venkat R, Billa, Vinay K, Subbaiah, D. R. C. Venkata, Bharathi, E. Vijaya, Vasquez-Del Carpio, Rodrigo, Padgaonkar, Amol, Baker, Stacey J, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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(Z)-1-Aryl-3-arylamino-2-propen-1-ones, Highly Active Stimulators of Tubulin Polymerization: Synthesis, Structure–Activity Relationship (SAR), Tubulin Polymerization, and Cell Growth Inhibition Studies
Reddy, M. V. Ramana, Akula, Balaiah, Cosenza, Stephen C, Lee, Clement M, Mallireddigari, Muralidhar R, Pallela, Venkat R, Subbaiah, D. R. C. Venkata, Udofa, Andrew, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2)
Reddy, M.V. Ramana, Akula, Balireddy, Jatiani, Shashidhar, Vasquez-Del Carpio, Rodrigo, Billa, Vinay K., Mallireddigari, Muralidhar R., Cosenza, Stephen C., Venkata Subbaiah, D.R.C., Bharathi, E. Vijaya, Pallela, Venkat R., Ramkumar, Poornima, Jain, Rinku, Aggarwal, Aneel K., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Design, synthesis, and biological evaluation of ( E)- and ( Z)-styryl-2-acetoxyphenyl sulfides and sulfones as cyclooxygenase-2 inhibitors
Reddy, M.V. Ramana, Mallireddigari, Muralidhar Reddy, Pallela, Venkat R., Venkatapuram, Padmavathi, Boominathan, Rengasamy, Bell, Stanley C., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (01.03.2005)
Published in Bioorganic & medicinal chemistry (01.03.2005)
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Journal Article
Design, Synthesis, and Biological Evaluation of (E)‑N‑Aryl-2-arylethenesulfonamide Analogues as Potent and Orally Bioavailable Microtubule-Targeted Anticancer Agents
Reddy, M. V. Ramana, Mallireddigari, Muralidhar R, Pallela, Venkat R, Cosenza, Stephen C, Billa, Vinay K, Akula, Balaiah, Subbaiah, D. R. C. Venkata, Bharathi, E. Vijaya, Padgaonkar, Amol, Lv, Hua, Gallo, James M, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (11.07.2013)
Published in Journal of medicinal chemistry (11.07.2013)
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Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910·Na (Rigosertib®), a phase III clinical stage anti-cancer agent
Pallela, Venkat R, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Akula, Balaiah, Subbaiah, D R C Venkata, Reddy, E Premkumar, Reddy, M V Ramana
Published in Organic & biomolecular chemistry (28.03.2013)
Published in Organic & biomolecular chemistry (28.03.2013)
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Journal Article
Design, Synthesis, and Biological Evaluation of (E)-Styrylbenzylsulfones as Novel Anticancer Agents
Reddy, M. V. Ramana, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Pallela, Venkat R, Iqbal, Nabisa M, Robell, Kimberly A, Kang, Anthony D, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (10.01.2008)
Published in Journal of medicinal chemistry (10.01.2008)
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Journal Article
Radiolabeled somatostatin analogs in prostate cancer
Thakur, M.L., Kolan, H., Li, J., Wiaderkiewicz, R., Pallela, V.R., Duggaraju, R., Schally, A.V.
Published in Nuclear medicine and biology (1997)
Published in Nuclear medicine and biology (1997)
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Chitosan–amylopectin/hydroxyapatite and chitosan–chondroitin sulphate/hydroxyapatite composite scaffolds for bone tissue engineering
Venkatesan, Jayachandran, Pallela, Ramjee, Bhatnagar, Ira, Kim, Se-Kwon
Published in International journal of biological macromolecules (01.12.2012)
Published in International journal of biological macromolecules (01.12.2012)
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Anti-photoaging and photoprotective compounds derived from marine organisms
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Book Review
Design, synthesis and evaluation of ( E)-α-benzylthio chalcones as novel inhibitors of BCR-ABL kinase
Reddy, M.V. Ramana, Pallela, Venkat R., Cosenza, Stephen C., Mallireddigari, Muralidhar R., Patti, Revathi, Bonagura, Marie, Truongcao, May, Akula, Balaiah, Jatiani, Shashidhar S., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (15.03.2010)
Published in Bioorganic & medicinal chemistry (15.03.2010)
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Journal Article
A receptor-specific peptide for imaging infection and inflammation
Rao, P S, Pallela, V R, Vassileva-Belnikolovska, D, Jungkind, D, Thakur, M L
Published in Nuclear medicine communications (01.11.2000)
Published in Nuclear medicine communications (01.11.2000)
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Journal Article
Imaging Thromboembolism with Tc-99m–Labeled Thrombospondin Receptor Analogs TP-1201 and TP-1300
Pallela, V.R., Thakur, M.L., Consigny, P.M., Rao, P.S., Vasileva-Belnikolavska, D., Shi, R.
Published in Thrombosis research (15.02.1999)
Published in Thrombosis research (15.02.1999)
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Journal Article
99mTc-Labeled Vasoactive Intestinal Peptide Receptor Agonist: Functional Studies
Pallela, Venkat R, Thakur, Mathew L, Chakder, Sushanta, Rattan, Satish
Published in The Journal of nuclear medicine (1978) (01.02.1999)
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Published in The Journal of nuclear medicine (1978) (01.02.1999)
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