The selectivity of inhibitors of protein kinase CK2: an update
Pagano, Mario A, Bain, Jenny, Kazimierczuk, Zygmunt, Sarno, Stefania, Ruzzene, Maria, Di Maira, Giovanni, Elliott, Matthew, Orzeszko, Andrzej, Cozza, Giorgio, Meggio, Flavio, Pinna, Lorenzo A
Published in Biochemical journal (01.11.2008)
Published in Biochemical journal (01.11.2008)
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Quinalizarin as a potent, selective and cell-permeable inhibitor of protein kinase CK2
Cozza, Giorgio, Mazzorana, Marco, Papinutto, Elena, Bain, Jenny, Elliott, Matthew, di Maira, Giovanni, Gianoncelli, Alessandra, Pagano, Mario A, Sarno, Stefania, Ruzzene, Maria, Battistutta, Roberto, Meggio, Flavio, Moro, Stefano, Zagotto, Giuseppe, Pinna, Lorenzo A
Published in Biochemical journal (15.07.2009)
Published in Biochemical journal (15.07.2009)
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Detection of phospho-sites generated by protein kinase CK2 in CFTR: mechanistic aspects of Thr1471 phosphorylation
Venerando, Andrea, Franchin, Cinzia, Cant, Natasha, Cozza, Giorgio, Pagano, Mario A, Tosoni, Kendra, Al-Zahrani, Ateeq, Arrigoni, Giorgio, Ford, Robert C, Mehta, Anil, Pinna, Lorenzo A
Published in PloS one (18.09.2013)
Published in PloS one (18.09.2013)
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Optimization of Protein Kinase CK2 Inhibitors Derived from 4,5,6,7-Tetrabromobenzimidazole
Pagano, Mario A, Andrzejewska, Mariola, Ruzzene, Maria, Sarno, Stefania, Cesaro, Luca, Bain, Jenny, Elliott, Matthew, Meggio, Flavio, Kazimierczuk, Zygmunt, Pinna, Lorenzo A
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
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Identification of Ellagic Acid as Potent Inhibitor of Protein Kinase CK2: A Successful Example of a Virtual Screening Application
Cozza, Giorgio, Bonvini, Paolo, Zorzi, Elisa, Poletto, Giorgia, Pagano, Mario A., Sarno, Stefania, Donella-Deana, Arianna, Zagotto, Giuseppe, Rosolen, Angelo, Pinna, Lorenzo A., Meggio, Flavio, Moro, Stefano
Published in Journal of medicinal chemistry (20.04.2006)
Published in Journal of medicinal chemistry (20.04.2006)
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Tetrabromocinnamic Acid (TBCA) and Related Compounds Represent a New Class of Specific Protein Kinase CK2 Inhibitors
Pagano, Mario A., Poletto, Giorgia, Di Maira, Giovanni, Cozza, Giorgio, Ruzzene, Maria, Sarno, Stefania, Bain, Jenny, Elliott, Matthew, Moro, Stefano, Zagotto, Giuseppe, Meggio, Flavio, Pinna, Lorenzo A.
Published in Chembiochem : a European journal of chemical biology (02.01.2007)
Published in Chembiochem : a European journal of chemical biology (02.01.2007)
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Geldanamycin-induced Lyn dissociation from aberrant Hsp90-stabilized cytosolic complex is an early event in apoptotic mechanisms in B-chronic lymphocytic leukemia
Trentin, Livio, Frasson, Martina, Donella-Deana, Arianna, Frezzato, Federica, Pagano, Mario A., Tibaldi, Elena, Gattazzo, Cristina, Zambello, Renato, Semenzato, Gianpietro, Brunati, Anna M.
Published in Blood (01.12.2008)
Published in Blood (01.12.2008)
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Aurora-A site specificity: a study with synthetic peptide substrates
Ferrari, Stefano, Marin, Oriano, Pagano, Mario A, Meggio, Flavio, Hess, Daniel, El-Shemerly, Mahmoud, Krystyniak, Agnieszka, Pinna, Lorenzo A
Published in Biochemical journal (15.08.2005)
Published in Biochemical journal (15.08.2005)
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CFTR mutations altering CFTR fragmentation
Tosoni, Kendra, Stobbart, Michelle, Cassidy, Diane M, Venerando, Andrea, Pagano, Mario A, Luz, Simão, Amaral, Margarida D, Kunzelmann, Karl, Pinna, Lorenzo A, Farinha, Carlos M, Mehta, Anil
Published in Biochemical journal (01.01.2013)
Published in Biochemical journal (01.01.2013)
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An NBD Derivative of the Selective Rat Toxicant Norbormide as a New Probe for Living Cell Imaging
D'Amore, Claudio, Orso, Genny, Fusi, Fabio, Pagano, Mario A, Miotto, Giovanni, Forgiarini, Alessia, De Martin, Sara, Castellani, Giulia, Ribaudo, Giovanni, Rennison, David, Brimble, Margaret A, Hopkins, Brian, Ferrarese, Alessandro, Bova, Sergio
Published in Frontiers in pharmacology (23.09.2016)
Published in Frontiers in pharmacology (23.09.2016)
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Pancreatic and duodenal homeobox 1 (PDX1) phosphorylation at serine-269 is HIPK2-dependent and affects PDX1 subnuclear localization
An, Rong, da Silva Xavier, Gabriela, Semplici, Francesca, Vakhshouri, Saharnaz, Hao, Huai-Xiang, Rutter, Jared, Pagano, Mario A., Meggio, Flavio, Pinna, Lorenzo A., Rutter, Guy A.
Published in Biochemical and biophysical research communications (20.08.2010)
Published in Biochemical and biophysical research communications (20.08.2010)
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Biochemical and three-dimensional-structural study of the specific inhibition of protein kinase CK2 by [5-oxo-5,6-dihydroindolo-(1,2-a)quinazolin-7-yl]acetic acid (IQA)
Sarno, Stefania, de Moliner, Erika, Ruzzene, Maria, Pagano, Mario A, Battistutta, Roberto, Bain, Jenny, Fabbro, Doriano, Schoepfer, Joseph, Elliott, Matthew, Furet, Pascal, Meggio, Flavio, Zanotti, Giuseppe, Pinna, Lorenzo A
Published in Biochemical journal (15.09.2003)
Published in Biochemical journal (15.09.2003)
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Lyn-mediated mitochondrial tyrosine phosphorylation is required to preserve mitochondrial integrity in early liver regeneration
Gringeri, Enrico, Carraro, Amedeo, Tibaldi, Elena, D'Amico, Francesco E, Mancon, Mario, Toninello, Antonio, Pagano, Mario A, Vio, Claudia, Cillo, Umberto, Brunati, Anna M
Published in Biochemical journal (15.01.2010)
Published in Biochemical journal (15.01.2010)
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A Noncanonical Sequence Phosphorylated by Casein Kinase 1 in β-Catenin May Play a Role in Casein Kinase 1 Targeting of Important Signaling Proteins
Marin, Oriano, Bustos, Victor H., Cesaro, Luca, Meggio, Flavio, Pagano, Mario A., Antonelli, Marcelo, Allende, Catherine C., Pinna, Lorenzo A., Allende, Jorge E.
Published in Proceedings of the National Academy of Sciences - PNAS (02.09.2003)
Published in Proceedings of the National Academy of Sciences - PNAS (02.09.2003)
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Inhibition of Protein Kinase CK2 by Condensed Polyphenolic Derivatives. An in Vitro and in Vivo Study
Meggio, Flavio, Pagano, Mario A, Moro, Stefano, Zagotto, Giuseppe, Ruzzene, Maria, Sarno, Stefania, Cozza, Giorgio, Bain, Jenny, Elliott, Matthew, Deana, Arianna Donella, Brunati, Anna Maria, Pinna, Lorenzo A
Published in Biochemistry (Easton) (12.10.2004)
Published in Biochemistry (Easton) (12.10.2004)
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A Modified KESTREL Search Reveals a Basophilic Substrate Consensus for the Saccharomyces cerevisiae Npr1 Protein Kinase
Gander, Stefan, Martin, Dietmar, Hauri, Simon, Moes, Suzette, Poletto, Giorgia, Pagano, Mario A, Marin, Oriano, Meggio, Flavio, Jenoe, Paul
Published in Journal of proteome research (06.11.2009)
Published in Journal of proteome research (06.11.2009)
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Cystic fibrosis transmembrane regulator fragments with the Phe508 deletion exert a dual allosteric control over the master kinase CK2
Pagano, Mario A, Marin, Oriano, Cozza, Giorgio, Sarno, Stefania, Meggio, Flavio, Treharne, Kate J, Mehta, Anil, Pinna, Lorenzo A
Published in Biochemical journal (27.01.2010)
Published in Biochemical journal (27.01.2010)
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2-Dimethylamino-4,5,6,7-tetrabromo-1H-benzimidazole: a novel powerful and selective inhibitor of protein kinase CK2
Pagano, Mario A, Meggio, Flavio, Ruzzene, Maria, Andrzejewska, Mariola, Kazimierczuk, Zygmunt, Pinna, Lorenzo A
Published in Biochemical and biophysical research communications (03.09.2004)
Published in Biochemical and biophysical research communications (03.09.2004)
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Structural features underlying the selectivity of the kinase inhibitors NBC and dNBC: role of a nitro group that discriminates between CK2 and DYRK1A
Sarno, Stefania, Mazzorana, Marco, Traynor, Ryan, Ruzzene, Maria, Cozza, Giorgio, Pagano, Mario A., Meggio, Flavio, Zagotto, Giuseppe, Battistutta, Roberto, Pinna, Lorenzo A.
Published in Cellular and molecular life sciences : CMLS (01.02.2012)
Published in Cellular and molecular life sciences : CMLS (01.02.2012)
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Label-free fluorescence detection of kinase activity using a gold nanoparticle based indicator displacement assay
Pezzato, Cristian, Zaramella, Davide, Martinelli, Massimiliano, Pieters, Grégory, Pagano, Mario A, Prins, Leonard J
Published in Organic & biomolecular chemistry (28.01.2015)
Published in Organic & biomolecular chemistry (28.01.2015)
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