Monohydrazone Based G‑Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells
Amato, Jussara, Miglietta, Giulia, Morigi, Rita, Iaccarino, Nunzia, Locatelli, Alessandra, Leoni, Alberto, Novellino, Ettore, Pagano, Bruno, Capranico, Giovanni, Randazzo, Antonio
Published in Journal of medicinal chemistry (26.03.2020)
Published in Journal of medicinal chemistry (26.03.2020)
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Journal Article
HMGB1 binds to the KRAS promoter G-quadruplex: a new player in oncogene transcriptional regulation?
Amato, Jussara, Madanayake, Thushara W, Iaccarino, Nunzia, Novellino, Ettore, Randazzo, Antonio, Hurley, Laurence H, Pagano, Bruno
Published in Chemical communications (Cambridge, England) (01.01.2018)
Published in Chemical communications (Cambridge, England) (01.01.2018)
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On the binding of naphthalene diimides to a human telomeric G-quadruplex multimer model
Pirota, Valentina, Platella, Chiara, Musumeci, Domenica, Benassi, Alessandra, Amato, Jussara, Pagano, Bruno, Colombo, Giorgio, Freccero, Mauro, Doria, Filippo, Montesarchio, Daniela
Published in International journal of biological macromolecules (01.01.2021)
Published in International journal of biological macromolecules (01.01.2021)
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Journal Article
Ligand binding to G-quadruplex DNA: new insights from ultraviolet resonance Raman spectroscopy
Di Fonzo, Silvia, Amato, Jussara, D'Aria, Federica, Caterino, Marco, D'Amico, Francesco, Gessini, Alessandro, Brady, John W, Cesàro, Attilio, Pagano, Bruno, Giancola, Concetta
Published in Physical chemistry chemical physics : PCCP (15.04.2020)
Published in Physical chemistry chemical physics : PCCP (15.04.2020)
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Journal Article
Binding of Harmine Derivatives to DNA: A Spectroscopic Investigation
Pagano, Bruno, Caterino, Marco, Filosa, Rosanna, Giancola, Concetta
Published in Molecules (Basel, Switzerland) (27.10.2017)
Published in Molecules (Basel, Switzerland) (27.10.2017)
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Journal Article
Controlled Pore Glass-based oligonucleotide affinity support: towards High Throughput Screening methods for the identification of conformation-selective G-quadruplex ligands
Platella, Chiara, Musumeci, Domenica, Arciello, Angela, Doria, Filippo, Freccero, Mauro, Randazzo, Antonio, Amato, Jussara, Pagano, Bruno, Montesarchio, Daniela
Published in Analytica chimica acta (07.11.2018)
Published in Analytica chimica acta (07.11.2018)
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Journal Article
Studying the effect of crowding and dehydration on DNA G-quadruplexes
Petraccone, Luigi, Pagano, Bruno, Giancola, Concetta
Published in Methods (San Diego, Calif.) (01.05.2012)
Published in Methods (San Diego, Calif.) (01.05.2012)
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Journal Article
Assessing the influence of pH and cationic strength on i-motif DNA structure
Iaccarino, Nunzia, Di Porzio, Anna, Amato, Jussara, Pagano, Bruno, Brancaccio, Diego, Novellino, Ettore, Leardi, Riccardo, Randazzo, Antonio
Published in Analytical and bioanalytical chemistry (01.11.2019)
Published in Analytical and bioanalytical chemistry (01.11.2019)
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Journal Article
Targeting of Telomeric Repeat-Containing RNA G-Quadruplexes: From Screening to Biophysical and Biological Characterization of a New Hit Compound
Marzano, Simona, Pagano, Bruno, Iaccarino, Nunzia, Di Porzio, Anna, De Tito, Stefano, Vertecchi, Eleonora, Salvati, Erica, Randazzo, Antonio, Amato, Jussara
Published in International journal of molecular sciences (24.09.2021)
Published in International journal of molecular sciences (24.09.2021)
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Journal Article
Toward the Development of Specific G‑Quadruplex Binders: Synthesis, Biophysical, and Biological Studies of New Hydrazone Derivatives
Amato, Jussara, Morigi, Rita, Pagano, Bruno, Pagano, Alessia, Ohnmacht, Stephan, De Magis, Alessio, Tiang, Yee-Peng, Capranico, Giovanni, Locatelli, Alessandra, Graziadio, Alessandra, Leoni, Alberto, Rambaldi, Mirella, Novellino, Ettore, Neidle, Stephen, Randazzo, Antonio
Published in Journal of medicinal chemistry (23.06.2016)
Published in Journal of medicinal chemistry (23.06.2016)
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Applications of isothermal titration calorimetry in biophysical studies of G-quadruplexes
Pagano, Bruno, Mattia, Carlo Andrea, Giancola, Concetta
Published in International Journal of Molecular Sciences (02.07.2009)
Published in International Journal of Molecular Sciences (02.07.2009)
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Book Review
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition
Nocentini, Alessio, Di Porzio, Anna, Bonardi, Alessandro, Bazzicalupi, Carla, Petreni, Andrea, Biver, Tarita, Bua, Silvia, Marzano, Simona, Amato, Jussara, Pagano, Bruno, Iaccarino, Nunzia, De Tito, Stefano, Amente, Stefano, Supuran, Claudiu T., Randazzo, Antonio, Gratteri, Paola
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2024)
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2024)
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Toward G-Quadruplex-Based Anticancer Agents: Biophysical and Biological Studies of Novel AS1411 Derivatives
Ogloblina, Anna M, Iaccarino, Nunzia, Capasso, Domenica, Di Gaetano, Sonia, Garzarella, Emanuele U, Dolinnaya, Nina G, Yakubovskaya, Marianna G, Pagano, Bruno, Amato, Jussara, Randazzo, Antonio
Published in International journal of molecular sciences (21.10.2020)
Published in International journal of molecular sciences (21.10.2020)
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Journal Article
Synthesis and Characterization of Bis-Triazolyl-Pyridine Derivatives as Noncanonical DNA-Interacting Compounds
Di Porzio, Anna, Galli, Ubaldina, Amato, Jussara, Zizza, Pasquale, Iachettini, Sara, Iaccarino, Nunzia, Marzano, Simona, Santoro, Federica, Brancaccio, Diego, Carotenuto, Alfonso, De Tito, Stefano, Biroccio, Annamaria, Pagano, Bruno, Tron, Gian Cesare, Randazzo, Antonio
Published in International journal of molecular sciences (04.11.2021)
Published in International journal of molecular sciences (04.11.2021)
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Journal Article
Structural and Conformational Requisites in DNA Quadruplex Groove Binding: Another Piece to the Puzzle
Cosconati, Sandro, Marinelli, Luciana, Trotta, Roberta, Virno, Ada, De Tito, Stefano, Romagnoli, Romeo, Pagano, Bruno, Limongelli, Vittorio, Giancola, Concetta, Baraldi, Pier Giovanni, Mayol, Luciano, Novellino, Ettore, Randazzo, Antonio
Published in Journal of the American Chemical Society (12.05.2010)
Published in Journal of the American Chemical Society (12.05.2010)
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