novel, small molecule inhibitor of Hsc70/Hsp70 potentiates Hsp90 inhibitor induced apoptosis in HCT116 colon carcinoma cells
Massey, Andrew J, Williamson, Douglas S, Browne, Helen, Murray, James B, Dokurno, Pawel, Shaw, Terry, Macias, Alba T, Daniels, Zoe, Geoffroy, Stephanie, Dopson, Melanie, Lavan, Paul, Matassova, Natalia, Francis, Geraint L, Graham, Christopher J, Parsons, Rachel, Wang, Yikang, Padfield, Antony, Comer, Mike, Drysdale, Martin J, Wood, Mike
Published in Cancer chemotherapy and pharmacology (01.08.2010)
Published in Cancer chemotherapy and pharmacology (01.08.2010)
Get full text
Journal Article
Combining Hit Identification Strategies: Fragment-Based and in Silico Approaches to Orally Active 2-Aminothieno[2,3-d]pyrimidine Inhibitors of the Hsp90 Molecular Chaperone
Brough, Paul A, Barril, Xavier, Borgognoni, Jenifer, Chene, Patrick, Davies, Nicholas G. M, Davis, Ben, Drysdale, Martin J, Dymock, Brian, Eccles, Suzanne A, Garcia-Echeverria, Carlos, Fromont, Christophe, Hayes, Angela, Hubbard, Roderick E, Jordan, Allan M, Jensen, Michael Rugaard, Massey, Andrew, Merrett, Angela, Padfield, Antony, Parsons, Rachel, Radimerski, Thomas, Raynaud, Florence I, Robertson, Alan, Roughley, Stephen D, Schoepfer, Joseph, Simmonite, Heather, Sharp, Swee Y, Surgenor, Allan, Valenti, Melanie, Walls, Steven, Webb, Paul, Wood, Mike, Workman, Paul, Wright, Lisa
Published in Journal of medicinal chemistry (13.08.2009)
Published in Journal of medicinal chemistry (13.08.2009)
Get full text
Journal Article
Antagonists of the Human A2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-d]pyrimidines
Gillespie, Roger J, Bamford, Samantha J, Botting, Ruth, Comer, Mike, Denny, Sarah, Gaur, Suneel, Griffin, Michael, Jordan, Allan M, Knight, Anthony R, Lerpiniere, Joanne, Leonardi, Stefania, Lightowler, Sean, McAteer, Steven, Merrett, Angela, Misra, Anil, Padfield, Antony, Reece, Mark, Saadi, Mona, Selwood, Daniel L, Stratton, Gemma C, Surry, Dominic, Todd, Richard, Tong, Xin, Ruston, Vicki, Upton, Rebecca, Weiss, Scott M
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
Get full text
Journal Article
Antagonists of the Human A(2A) Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-d]pyrimidines
Gillespie, Roger J., Bamford, Samantha J., Botting, Ruth, Comer, Mike, Denny, Sarah, Gaur, Suneel, Griffin, Michael, Jordan, Allan M., Knight, Anthony R., Lerpiniere, Joanne, Leonardi, Stefania, Lightowler, Sean, McAteer, Steven, Merrett, Angela, Misra, Anil, Padfield, Antony, Reece, Mark, Saadi, Mona, Selwood, Daniel L., Stratton, Gemma C., Surry, Dominic, Todd, Richard, Tong, Xin, Ruston, Vicki, Upton, Rebecca, Weiss, Scott M.
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
Get full text
Journal Article
Antagonists of the Human A 2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5- d ]pyrimidines
Gillespie, Roger J., Bamford, Samantha J., Botting, Ruth, Comer, Mike, Denny, Sarah, Gaur, Suneel, Griffin, Michael, Jordan, Allan M., Knight, Anthony R., Lerpiniere, Joanne, Leonardi, Stefania, Lightowler, Sean, McAteer, Steven, Merrett, Angela, Misra, Anil, Padfield, Antony, Reece, Mark, Saadi, Mona, Selwood, Daniel L., Stratton, Gemma C., Surry, Dominic, Todd, Richard, Tong, Xin, Ruston, Vicki, Upton, Rebecca, Weiss, Scott M.
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
Get full text
Journal Article