Synthesis and multiparametric evaluation of thiadiazoles and oxadiazoles as diacylglycerol acyltransferase type 1 inhibitors
Mougenot, Patrick, Namane, Claudie, Fett, Eykmar, Goumy, Florence, Dadji-Faïhun, Rommel, Langot, Gwladys, Monseau, Catherine, Onofri, Bénédicte, Pacquet, François, Pascal, Cécile, Crespin, Olivier, Ben-Hassine, Majdi, Ragot, Jean-Luc, Van-Pham, Thao, Philippo, Christophe, Chatelain-Egger, Florence, Péron, Philippe, Le Bail, Jean-Christophe, Guillot, Etienne, Chamiot-Clerc, Philippe, Chabanaud, Marie-Aude, Pruniaux, Marie-Pierre, Ménegotto, Jérôme, Schmidt, Friedemann, Venier, Olivier, Viviani, Fabrice, Nicolai, Eric
Published in Bioorganic & medicinal chemistry letters (01.01.2016)
Published in Bioorganic & medicinal chemistry letters (01.01.2016)
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Thiadiazoles as new inhibitors of diacylglycerol acyltransferase type 1
Mougenot, Patrick, Namane, Claudie, Fett, Eykmar, Camy, Florence, Dadji-Faïhun, Rommel, Langot, Gwladys, Monseau, Catherine, Onofri, Bénédicte, Pacquet, François, Pascal, Cécile, Crespin, Olivier, Ben-Hassine, Majdi, Ragot, Jean-Luc, Van-Pham, Thao, Philippo, Christophe, Chatelain-Egger, Florence, Péron, Philippe, Le Bail, Jean-Christophe, Guillot, Etienne, Chamiot-Clerc, Philippe, Chabanaud, Marie-Aude, Pruniaux, Marie-Pierre, Schmidt, Friedemann, Venier, Olivier, Nicolaï, Eric, Viviani, Fabrice
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Discovery of SAR184841, a potent and long-lasting inhibitor of 11β-hydroxysteroid dehydrogenase type 1, active in a physiopathological animal model of T2D
Venier, Olivier, Pascal, Cécile, Braun, Alain, Namane, Claudie, Mougenot, Patrick, Crespin, Olivier, Pacquet, François, Mougenot, Cécile, Monseau, Catherine, Onofri, Bénédicte, Dadji-Faïhun, Rommel, Leger, Céline, Ben-Hassine, Majdi, Van-Pham, Thao, Ragot, Jean-Luc, Philippo, Christophe, Farjot, Géraldine, Noah, Lionel, Maniani, Karima, Boutarfa, Asma, Nicolaï, Eric, Guillot, Etienne, Pruniaux, Marie-Pierre, Güssregen, Stefan, Engel, Christian, Coutant, Anne-Laure, de Miguel, Beatriz, Castro, Antonio
Published in Bioorganic & medicinal chemistry letters (15.04.2013)
Published in Bioorganic & medicinal chemistry letters (15.04.2013)
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Pyrrolidine-pyrazole ureas as potent and selective inhibitors of 11β-hydroxysteroid-dehydrogenase type 1
Venier, Olivier, Pascal, Cécile, Braun, Alain, Namane, Claudie, Mougenot, Patrick, Crespin, Olivier, Pacquet, François, Mougenot, Cécile, Monseau, Catherine, Onofri, Bénédicte, Dadji-Faïhun, Rommel, Leger, Céline, Ben-Hassine, Majdi, Van-Pham, Thao, Ragot, Jean-Luc, Philippo, Christophe, Güssregen, Stefan, Engel, Christian, Farjot, Géraldine, Noah, Lionel, Maniani, Karima, Nicolaï, Eric
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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Biokinetic data and models for occupational intake of lanthanoids
Leggett, Rich, Ansoborlo, Eric, Bailey, Michael, Gregoratto, Demetrio, Paquet, Francois, Taylor, David
Published in International journal of radiation biology (01.11.2014)
Published in International journal of radiation biology (01.11.2014)
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METHODS OF MAKING TOLEBRUTINIB
CABOS, Claude, VIGNE, Sylvie, CHARAUDEAU, Alexis, BORIE, Cyril, BENELLI, Christophe, JANSSENS, Laurence, BAILLY, Frédéric, SALLÉ, Laurent, RODIER, Fabien, SODO, Alfred, PACQUET, François, BOSCH, Michaël
Year of Publication 21.12.2023
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Year of Publication 21.12.2023
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ICRP Publication 137: Occupational Intakes of Radionuclides: Part 3
Pacquet, Francois, Bailey, Michael, Leggett, Richard Wayne, Lipsztein, Joyce, Marsh, James, Fell, Tim, Smith, Tracy, Nosske, Dietmar, Eckerman, Keith, Berkovskii, Vladimir, Blanchardon, Eric, Bolch, Wes, Harrison, John
Year of Publication 01.12.2017
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Year of Publication 01.12.2017
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Dissociated Nonsteroidal Glucocorticoid Receptor Modulators; Discovery of the Agonist Trigger in a Tetrahydronaphthalene−Benzoxazine Series
Barker, Mike, Clackers, Margaret, Copley, Royston, Demaine, Derek A, Humphreys, Davina, Inglis, Graham G. A, Johnston, Michael J, Jones, Haydn T, Haase, Michael V, House, David, Loiseau, Richard, Nisbet, Lesley, Pacquet, Francois, Skone, Philip A, Shanahan, Stephen E, Tape, Dan, Vinader, Victoria M, Washington, Melanie, Uings, Iain, Upton, Richard, McLay, Iain M, Macdonald, Simon J. F
Published in Journal of medicinal chemistry (13.07.2006)
Published in Journal of medicinal chemistry (13.07.2006)
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Discovery of SAR184841, a potent and long-lasting inhibitor of 11[beta]-hydroxysteroid dehydrogenase type 1, active in a physiopathological animal model of T2D
Venier, Olivier, Pascal, Cecile, Braun, Alain, Namane, Claudie, Mougenot, Patrick, Crespin, Olivier, Pacquet, Francois, Mougenot, Cecile, Monseau, Catherine, Onofri, Benedicte, Dadji-Faiehun, Rommel, Leger, Celine, Ben-Hassine, Majdi, Van-Pham, Thao, Ragot, Jean-Luc, Philippo, Christophe, Farjot, Geraldine, Noah, Lionel, Maniani, Karima, Boutarfa, Asma, Nicolaie, Eric, Guillot, Etienne, Pruniaux, Marie-Pierre, Guessregen, Stefan, Engel, Christian, Coutant, Anne-Laure, de Miguel, Beatriz, Castro, Antonio
Published in Bioorganic & medicinal chemistry letters (15.04.2013)
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Published in Bioorganic & medicinal chemistry letters (15.04.2013)
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TETRAHYDROQUINOXALINE UREA DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF
PACQUET, FRANÇOIS, NICOLAI, ERIC, NAMANE, CLAUDIE, PASCAL, CÉCILE, VENIER, OLIVIER
Year of Publication 19.11.2014
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Year of Publication 19.11.2014
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Design and Synthesis of New Nonsteroidal Glucocorticoid Modulators through Application of an “Agreement Docking” Method
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Published in Journal of medicinal chemistry (14.07.2005)
Published in Journal of medicinal chemistry (14.07.2005)
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Assessment and interpretation of internal doses: uncertainty and variability
Paquet, F., Bailey, M.R., Leggett, R.W., Harrison, J.D.
Published in Annals of the ICRP (01.06.2016)
Published in Annals of the ICRP (01.06.2016)
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مشتقات اليوريا التيتراهيدروكوينوكساليني ، إعدادها وتطبيقها في العلاج
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Year of Publication 01.02.2011
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Year of Publication 01.02.2011
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Methods of making tolebrutinib
BOSCH, MICHAEL, SODO, ALFRED, BAILLY, FREDERIC, BENELLI, CHRISTOPHE, RODIER, FABIEN, SALLE, LAURENT, JANSSENS, LAURENCE, BORIE, CYRIL, CABOS, CLAUDE, VIGNE, SYLVIE, CHARAUDEAU, ALEXIS, PACQUET, FRANCOIS
Year of Publication 01.03.2024
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Year of Publication 01.03.2024
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Tetrahydroquinoxaline urea derivatives as modulators of 11beta-hydroxysteroid dehydrogenase type 1
NAMANE CLAUDIE, NICOLAI ERIC, PASCAL CECILE, PACQUET FRANCOIS, VENIER OLIVIER
Year of Publication 10.09.2013
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Year of Publication 10.09.2013
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DERIVES D'UREE DE TETRAHYDROQUINOXALINE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
NAMANE CLAUDIE, NICOLAI ERIC, PASCAL CECILE, PACQUET FRANCOIS, VENIER OLIVIER
Year of Publication 05.04.2013
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Year of Publication 05.04.2013
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TETRAHYDROQUINOXALINE UREA DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF
NICOLAI, ERIC, PASCAL, CECILE, NAMANE, CLAUDIE, PACQUET, FRANCOIS, VENIER, OLIVIER
Year of Publication 06.06.2012
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Year of Publication 06.06.2012
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