Polar Radical Pair Pathway To Assemble the Pyrimidinone Core of the HIV Integrase Inhibitor Raltegravir Potassium
Pye, Philip J, Zhong, Yong-Li, Jones, Gavin O, Reamer, Robert A, Houk, Kendall N, Askin, David
Published in Angewandte Chemie (International ed.) (19.05.2008)
Published in Angewandte Chemie (International ed.) (19.05.2008)
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Development of a Second-Generation, Highly Efficient Manufacturing Route for the HIV Integrase Inhibitor Raltegravir Potassium
Humphrey, Guy R, Pye, Philip J, Zhong, Yong-Li, Angelaud, Remy, Askin, David, Belyk, Kevin M, Maligres, Peter E, Mancheno, Danny E, Miller, Ross A, Reamer, Robert A, Weissman, Steven A
Published in Organic process research & development (21.01.2011)
Published in Organic process research & development (21.01.2011)
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A New Planar Chiral Bisphosphine Ligand for Asymmetric Catalysis: Highly Enantioselective Hydrogenations under Mild Conditions
Pye, Philip J, Rossen, Kai, Reamer, Robert A, Tsou, Nancy N, Volante, R. P, Reider, Paul J
Published in Journal of the American Chemical Society (02.07.1997)
Published in Journal of the American Chemical Society (02.07.1997)
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Efficient Synthesis of NK1 Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation
Brands, Karel M. J, Payack, Joseph F, Rosen, Jonathan D, Nelson, Todd D, Candelario, Alexander, Huffman, Mark A, Zhao, Matthew M, Li, Jing, Craig, Bridgette, Song, Zhiguo J, Tschaen, David M, Hansen, Karl, Devine, Paul N, Pye, Philip J, Rossen, Kai, Dormer, Peter G, Reamer, Robert A, Welch, Christopher J, Mathre, David J, Tsou, Nancy N, McNamara, James M, Reider, Paul J
Published in Journal of the American Chemical Society (26.02.2003)
Published in Journal of the American Chemical Society (26.02.2003)
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Kinetic Resolution of rac-4,12-Dibromo[2.2]paracyclophane in a Palladium [2.2]PHANEPHOS Catalyzed Amination
Rossen, Kai, Pye, Philip J, Maliakal, Ashok, Volante, R. P
Published in Journal of organic chemistry (19.09.1997)
Published in Journal of organic chemistry (19.09.1997)
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Serendipitous discovery of a pH-dependant atropisomer bond rotation: Toward a write-protectable chiral molecular switch?
Welch, Christopher J., Biba, Mirlinda, Pye, Philip, Angelaud, Remy, Egbertson, Melissa
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.11.2008)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.11.2008)
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Development of practical syntheses of potent non-nucleoside reverse transcriptase inhibitors
Kuethe, Jeffrey T., Zhong, Yong-Li, Alam, Mahbub, Alorati, Anthony D., Beutner, Gregory L., Cai, Dongwei, Fleitz, Fred J., Gibb, Andrew D., Kassim, Amude, Linn, Kathleen, Mancheno, Danny, Marcune, Benjamin, Pye, Philip J., Scott, Jeremy P., Tellers, David M., Xiang, Bangping, Yasuda, Nobuyoshi, Yin, Jingjun, Davies, Ian W.
Published in Tetrahedron (27.06.2009)
Published in Tetrahedron (27.06.2009)
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Conference Proceeding
Crystallization-Induced Diastereoselection: Asymmetric Synthesis of Substance P Inhibitors
Pye, Philip J., Rossen, Kai, Weissman, Steven A., Maliakal, Ashok, Reamer, Robert A., Ball, Richard, Tsou, Nancy N., Volante, R. P., Reider, Paul J.
Published in Chemistry : a European journal (15.03.2002)
Published in Chemistry : a European journal (15.03.2002)
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A Practical Synthesis of a COX-2-Specific Inhibitor
Davies, Ian W, Marcoux, Jean-Francois, Corley, Edward G, Journet, Michel, Cai, Dong-Wei, Palucki, Michael, Wu, Jimmy, Larsen, Robert D, Rossen, Kai, Pye, Philip J, DiMichele, Lisa, Dormer, Peter, Reider, Paul J
Published in Journal of organic chemistry (15.12.2000)
Published in Journal of organic chemistry (15.12.2000)
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Efficient and Practical Synthesis of a Potent Anti-MRSA β-Methylcarbapenem Containing a Releasable Side Chain
Humphrey, Guy R, Miller, Ross A, Pye, Philip J, Rossen, Kai, Reamer, Robert A, Maliakal, Ashok, Ceglia, Scott S, Grabowski, Edward J. J, Volante, R. P, Reider, Paul J
Published in Journal of the American Chemical Society (15.12.1999)
Published in Journal of the American Chemical Society (15.12.1999)
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Taxane diterpenes 2: Synthesis of the 7-deoxy ABC taxane skeleton, and reactions of the A-ring
Magnus, Philip, Booth, John, Diorazio, Louis, Donohoe, Timothy, Lynch, Vince, Magnus, Nicholas, Mendoza, José, Pye, Philip, Tarrant, James
Published in Tetrahedron (04.11.1996)
Published in Tetrahedron (04.11.1996)
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LEFORT LAURENT, VERZIJL GERARDUS KAREL MARIA, SU JINXIONG, KAPTEIN BERNARDUS, HORVATH ANDRAS, PYE PHILIP JAMES, YUAN YUANYUAN
Year of Publication 28.01.2022
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Year of Publication 28.01.2022
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BTK 억제제 제조를 위한 방법 및 중간체
WANG SHUO, WAGSCHAL SIMON ALBERT, SU JINXIONG, HORVATH ANDRAS, CHEN CHENG YI, PYE PHILIP JAMES, YUAN YUANYUAN
Year of Publication 28.01.2022
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Year of Publication 28.01.2022
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SYNTHESIS OF A BRUTON'S TYROSINE KINASE INHIBITOR
CHEN WEI, BENHAIM CYRIL, HORVATH ANDRAS, SMYTH MARK S, GOLDMAN ERICK, VERNER ERIK J, PYE PHILIP
Year of Publication 12.09.2017
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Year of Publication 12.09.2017
Patent
Serendipitous discovery of a pH-dependant atropisomer bond rotation : Toward a write-protectable chiral molecular switch?: Enantioseparations
WELCH, Christopher J, BIBA, Mirlinda, PYE, Philip, ANGELAUD, Remy, EGBERTSON, Melissa
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (2008)
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Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (2008)
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