Discovery and Structure-Based Design of Potent Covalent PPARγ Inverse-Agonists BAY-4931 and BAY-0069
Orsi, Douglas L., Pook, Elisabeth, Bräuer, Nico, Friberg, Anders, Lienau, Philip, Lemke, Christopher T., Stellfeld, Timo, Brüggemeier, Ulf, Pütter, Vera, Meyer, Hanna, Baco, Maria, Tang, Stephanie, Cherniack, Andrew D., Westlake, Lindsay, Bender, Samantha A., Kocak, Mustafa, Strathdee, Craig A., Meyerson, Matthew, Eis, Knut, Goldstein, Jonathan T.
Published in Journal of medicinal chemistry (10.11.2022)
Published in Journal of medicinal chemistry (10.11.2022)
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The Solution Structure of the N-Terminal Domain of E3L Shows a Tyrosine Conformation That May Explain Its Reduced Affinity to Z-DNA in vitro
Kahmann, Jan D., Wecking, Diana A., Putter, Vera, Lowenhaupt, Ky, Kim, Yang-Gyun, Schmieder, Peter, Oschkinat, Hartmut, Rich, Alexander, Schade, Markus
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Published in Proceedings of the National Academy of Sciences - PNAS (02.03.2004)
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Inhibition of BUB1 Kinase by BAY 1816032 Sensitizes Tumor Cells toward Taxanes, ATR, and PARP Inhibitors In Vitro and In Vivo
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Discovery and Characterization of the Potent and Highly Selective 1,7-Naphthyridine-Based Inhibitors BAY-091 and BAY-297 of the Kinase PIP4K2A
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Published in Journal of medicinal chemistry (11.11.2021)
Published in Journal of medicinal chemistry (11.11.2021)
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Correction to “Discovery and Structure-Based Design of Potent Covalent PPARγ Inverse-Agonists BAY-4931 and BAY-0069”
Orsi, Douglas L., Pook, Elisabeth, Bräuer, Nico, Friberg, Anders, Lienau, Philip, Lemke, Christopher T., Stellfeld, Timo, Brüggemeier, Ulf, Pütter, Vera, Meyer, Hanna, Baco, Maria, Tang, Stephanie, Cherniack, Andrew D., Westlake, Lindsay, Bender, Samantha A., Kocak, Mustafa, Strathdee, Craig A., Meyerson, Matthew, Eis, Knut, Goldstein, Jonathan T.
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Published in Journal of medicinal chemistry (12.01.2023)
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Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains
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Published in Journal of medicinal chemistry (11.05.2017)
Published in Journal of medicinal chemistry (11.05.2017)
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Expression and Characterization of Relaxin Family Peptide Receptor 1 Variants
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Published in Frontiers in pharmacology (28.01.2022)
Published in Frontiers in pharmacology (28.01.2022)
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Dual targeting of the androgen receptor and PI3K/AKT/mTOR pathways in prostate cancer models improves antitumor efficacy and promotes cell apoptosis
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Structural Evidence for Isoform-Selective Allosteric Inhibition of Lactate Dehydrogenase A
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Interaction and Assembly of Murine Pre-replicative Complex Proteins in Yeast and Mouse Cells
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Published in Journal of molecular biology (14.03.2003)
Published in Journal of molecular biology (14.03.2003)
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Surface‐mutagenesis strategies to enable structural biology crystallization platforms
Schaefer, Martina, Pütter, Vera, Hilpmann, André, Egner, Ursula, Holton, Simon James, Hillig, Roman Christian
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Published in Acta crystallographica. Section D, Biological crystallography. (01.09.2024)
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The RESOLUTE consortium: unlocking SLC transporters for drug discovery
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Published in Nature reviews. Drug discovery (01.07.2020)
Published in Nature reviews. Drug discovery (01.07.2020)
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Discovery and characterization of orally bioavailable 4-chloro-6-fluoroisophthalamides as covalent PPARG inverse-agonists
Orsi, Douglas L., Ferrara, Steven J., Siegel, Stephan, Friberg, Anders, Bouché, Léa, Pook, Elisabeth, Lienau, Philip, Bluck, Joseph P., Lemke, Christopher T., Akcay, Gizem, Stellfeld, Timo, Meyer, Hanna, Pütter, Vera, Holton, Simon J., Korr, Daniel, Jerchel-Furau, Isabel, Pantelidou, Constantia, Strathdee, Craig A., Meyerson, Matthew, Eis, Knut, Goldstein, Jonathan T.
Published in Bioorganic & medicinal chemistry (15.01.2023)
Published in Bioorganic & medicinal chemistry (15.01.2023)
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ACYL SULFONAMIDES FOR TREATING CANCER
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Year of Publication 29.10.2020
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Year of Publication 29.10.2020
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Structure of wild-type Plk-1 kinase domain in complex with a selective DARPin
Bandeiras, Tiago M., Hillig, Roman Christian, Matias, Pedro M., Eberspaecher, Uwe, Fanghänel, Jörg, Thomaz, Mónica, Miranda, Sandra, Crusius, Kerstin, Pütter, Vera, Amstutz, Patrick, Gulotti-Georgieva, Maya, Binz, H. Kaspar, Holz, Caterina, Schmitz, Arndt A. P., Lang, Christine, Donner, Peter, Egner, Ursula, Carrondo, Maria A., Müller-Tiemann, Beate
Published in Acta crystallographica. Section D, Biological crystallography. (01.04.2008)
Published in Acta crystallographica. Section D, Biological crystallography. (01.04.2008)
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SUBSTITUTED BENZYLINDAZOLES FOR USE AS BUB1 KINASE INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISEASES
MENGEL Anne, PREUSSE Cornelia, HITCHCOCK Marion, FANGHANEL Jorg, GNOTH Mark Jean, BRIEM Hans, SCHULZE Volker, PRECHTL Stefan, LIENAU Philip, SIEMEISTER Gerhard, PUTTER Vera, FERNANDEZ-MONTALVAN Amaury Ernesto, EIS Knut, WENGNER Antje Margret, HOLTON Simon
Year of Publication 29.06.2018
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Year of Publication 29.06.2018
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Substituted benzylindazoles for use as Bub1 kinase inhibitors in the treatment of hyperproliferative diseases
Schulze, Volker, Preusse, Cornelia, Briem, Hans, Mengel, Anne, Fanghanel, Jorg, Putter, Vera, Holton, Simon, Siemeister, Gerhard, Gnoth, Mark Jean, Lienau, Philip, Hitchcock, Marion, Wengner, Antje Margret, Prechtl, Stefan, Eis, Knut, Fernandez-Montalvan, Amaury Ernesto
Year of Publication 15.06.2017
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Year of Publication 15.06.2017
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