Induction of apoptosis and cell cycle arrest by CP-358,774, an inhibitor of epidermal growth factor receptor tyrosine kinase
MOYER, J. D, BARBACCI, E. G, NEVEU, M, POLLACK, V. A, PUSTILNIK, L. R, REYNOLDS, M. M, SLOAN, D, THELEMAN, A, MILLER, P, IWATA, K. K, ARNOLD, L, BOMAN, B, CUNNINGHAM, A, DIORIO, C, DOTY, J, MORIN, M. J, MOYER, M. P
Published in Cancer research (Chicago, Ill.) (01.11.1997)
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Published in Cancer research (Chicago, Ill.) (01.11.1997)
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Inhibition of Epidermal Growth Factor Receptor-Associated Tyrosine Phosphorylation in Human Carcinomas with CP-358,774: Dynamics of Receptor Inhibition In Situ and Antitumor Effects in Athymic Mice
Pollack, V A, Savage, D M, Baker, D A, Tsaparikos, K E, Sloan, D E, Moyer, J D, Barbacci, E G, Pustilnik, L R, Smolarek, T A, Davis, J A, Vaidya, M P, Arnold, L D, Doty, J L, Iwata, K K, Morin, M J
Published in The Journal of pharmacology and experimental therapeutics (01.11.1999)
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Published in The Journal of pharmacology and experimental therapeutics (01.11.1999)
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Anilinoquinazoline Inhibitors of Fructose 1,6-Bisphosphatase Bind at a Novel Allosteric Site: Synthesis, In Vitro Characterization, and X-ray Crystallography
Wright, Stephen W, Carlo, Anthony A, Carty, Maynard D, Danley, Dennis E, Hageman, David L, Karam, George A, Levy, Carolyn B, Mansour, Mahmoud N, Mathiowetz, Alan M, McClure, Lester D, Nestor, McPherson, R. Kirk, Pandit, Jayvardhan, Pustilnik, Leslie R, Schulte, Gayle K, Soeller, Walter C, Treadway, Judith L, Wang, Ing-Kae, Bauer, Paul H
Published in Journal of medicinal chemistry (29.08.2002)
Published in Journal of medicinal chemistry (29.08.2002)
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The biological and biochemical effects of CP-654577, a selective erbB2 kinase inhibitor, on human breast cancer cells
BARBACCI, E. Gabriella, PUSTILNIK, Leslie R, KATH, John C, ZHENGYU LIU, MOYER, James D, ROSSI, Ann Marie K, EMERSON, Erling, MILLER, Penny E, BOSCOE, Brian P, COX, Eric D, IWATA, Kenneth K, JANI, Jitesh P, PROVONCHA, Kathleen
Published in Cancer research (Chicago, Ill.) (01.08.2003)
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Published in Cancer research (Chicago, Ill.) (01.08.2003)
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INHIBITION OF THE ONCOGENE PRODUCT P185(ERBB-2) IN-VITRO AND IN-VIVO BY GELDANAMYCIN AND DIHYDROGELDANAMYCIN DERIVATIVES
SCHNUR, RC, CORMAN, ML, GALLASCHUN, RJ, COOPER, BA, DEE, MF, DOTY, JL, MUZZI, ML, MOYER, JD, DIORIO, CI, BARBACCI, EG, MILLER, PE, OBRIEN, AT, MORIN, MJ, FOSTER, BA, POLLACK, VA, SAVAGE, DM, SLOAN, DE, PUSTILNIK, LR, MOYER, MP
Published in Journal of medicinal chemistry (15.09.1995)
Published in Journal of medicinal chemistry (15.09.1995)
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Achieving selectivity between highly homologous tyrosine kinases: a novel selective erbB2 inhibitor
Bhattacharya, Samit K., Cox, Eric D., Kath, John C., Mathiowetz, Alan M., Morris, Joel, Moyer, James D., Pustilnik, Leslie R., Rafidi, Kris, Richter, Daniel T., Su, Chunyan, Wessel, Matthew D.
Published in Biochemical and biophysical research communications (25.07.2003)
Published in Biochemical and biophysical research communications (25.07.2003)
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ERBB-2 ONCOGENE INHIBITION BY GELDANAMYCIN DERIVATIVES - SYNTHESIS, MECHANISM OF ACTION, AND STRUCTURE-ACTIVITY-RELATIONSHIPS
SCHNUR, RC, CORMAN, ML, GALLASCHUN, RJ, COOPER, BA, DEE, MF, DOTY, JL, MUZZI, ML, DIORIO, CI, BARBACCI, EG, MILLER, PE, POLLACK, VA, SAVAGE, DM, SLOAN, DE, PUSTILNIK, LR, MOYER, JD, MOYER, MP
Published in Journal of medicinal chemistry (15.09.1995)
Published in Journal of medicinal chemistry (15.09.1995)
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