Substituted Aryl Benzylamines as Potent and Selective Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 3
Vicker, Nigel, Bailey, Helen V, Day, Joanna M, Mahon, Mary F, Smith, Andrew, Tutill, Helena J, Purohit, Atul, Potter, Barry V L
Published in Molecules (Basel, Switzerland) (26.11.2021)
Published in Molecules (Basel, Switzerland) (26.11.2021)
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Design and validation of specific inhibitors of 17β-hydroxysteroid dehydrogenases for therapeutic application in breast and prostate cancer, and in endometriosis
Day, Joanna M, Tutill, Helena J, Purohit, Atul, Reed, Michael J
Published in Endocrine-related cancer (01.09.2008)
Published in Endocrine-related cancer (01.09.2008)
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Journal Article
Lung isolation, one-lung ventilation and hypoxaemia during lung isolation
Purohit, Atul, Bhargava, Suresh, Mangal, Vandana, Parashar, Vinod Kumar
Published in Indian journal of anaesthesia (01.09.2015)
Published in Indian journal of anaesthesia (01.09.2015)
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Journal Article
Phase I Study of STX 64 (667 Coumate) in Breast Cancer Patients: The First Study of a Steroid Sulfatase Inhibitor
STANWAY, Susannah J, PUROHIT, Atul, ELLIOTT, Moira, POTTER, Barry V. L, REED, Michael J, COOMBES, R. Charles, WOO, L. W. Lawrence, SUFI, Saulat, VIGUSHIN, David, WARD, Rebecca, WILSON, Richard H, STANCZYK, Frank Z, DOBBS, Nicola, KULINSKAYA, Elena
Published in Clinical cancer research (01.03.2006)
Published in Clinical cancer research (01.03.2006)
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STX140, but not paclitaxel, inhibits mammary tumour initiation and progression in C3(1)/SV40 T/t-antigen transgenic mice
Meyer-Losic, Florence, Newman, Simon P, Day, Joanna M, Reed, Michael J, Kasprzyk, Philip G, Purohit, Atul, Foster, Paul A
Published in PloS one (06.12.2013)
Published in PloS one (06.12.2013)
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Aromatase and Dual Aromatase-Steroid Sulfatase Inhibitors from the Letrozole and Vorozole Templates
Wood, Paul M., Woo, L. W. Lawrence, Thomas, Mark P., Mahon, Mary F., Purohit, Atul, Potter, Barry V. L.
Published in ChemMedChem (01.08.2011)
Published in ChemMedChem (01.08.2011)
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Structure-Activity Relationship for the First-in-Class Clinical Steroid Sulfatase Inhibitor Irosustat (STX64, BN83495)
Woo, L. W. Lawrence, Ganeshapillai, Dharshini, Thomas, Mark P., Sutcliffe, Oliver B., Malini, Bindu, Mahon, Mary F., Purohit, Atul, Potter, Barry V. L.
Published in ChemMedChem (04.11.2011)
Published in ChemMedChem (04.11.2011)
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C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
Ganeshapillai, Dharshini, Woo, L. W. Lawrence, Thomas, Mark P, Purohit, Atul, Potter, Barry V. L
Published in ACS omega (30.09.2018)
Published in ACS omega (30.09.2018)
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2-Substituted Estradiol Bis-sulfamates, Multitargeted Antitumor Agents: Synthesis, In Vitro SAR, Protein Crystallography, and In Vivo Activity
Leese, Mathew P, Leblond, Bertrand, Smith, Andrew, Newman, Simon P, Di Fiore, Anna, De Simone, Giuseppina, Supuran, Claudiu T, Purohit, Atul, Reed, Michael J, Potter, Barry V. L
Published in Journal of medicinal chemistry (28.12.2006)
Published in Journal of medicinal chemistry (28.12.2006)
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The Development of Steroid Sulfatase Inhibitors for Hormone-Dependent Cancer Therapy
Day, Joanna M., Purohit, Atul, Tutill, Helena J., Foster, Paul A., Woo, L. W. Lawrence, Potter, Barry V. L., Reed, Michael J.
Published in Annals of the New York Academy of Sciences (01.02.2009)
Published in Annals of the New York Academy of Sciences (01.02.2009)
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Synthesis, Anti-tubulin and Antiproliferative SAR of Steroidomimetic Dihydroisoquinolinones
Leese, Mathew P., Jourdan, Fabrice L., Major, Meriel R., Dohle, Wolfgang, Thomas, Mark P., Hamel, Ernest, Ferrandis, Eric, Mahon, Mary F., Newman, Simon P., Purohit, Atul, Potter, Barry V. L.
Published in ChemMedChem (01.04.2014)
Published in ChemMedChem (01.04.2014)
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Recent developments of steroid sulfatase inhibitors as anti-cancer agents
Foster, Paul A, Reed, Michael J, Purohit, Atul
Published in Anti-cancer agents in medicinal chemistry (01.10.2008)
Published in Anti-cancer agents in medicinal chemistry (01.10.2008)
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Journal Article
STX140 Is Efficacious In vitro and In vivo in Taxane-Resistant Breast Carcinoma Cells
NEWMAN, Simon P, FOSTER, Paul A, REED, Michael J, PUROHIT, Atul, STENGEL, Chloe, DAY, Joanna M, HO, Yaik T, JUDDE, Jean-Gabriel, LASSALLE, Myriam, PREVOST, Gregoire, LEESE, Mathew P, POTTER, Barry V. L
Published in Clinical cancer research (15.01.2008)
Published in Clinical cancer research (15.01.2008)
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A New Therapeutic Strategy against Hormone-Dependent Breast Cancer: The Preclinical Development of a Dual Aromatase and Sulfatase Inhibitor
FOSTER, Paul A, CHANDER, Surinder K, PUROHIT, Atul, NEWMAN, Simon P, WOO, L. W. Lawrence, SUTCLIFFE, Oliver B, BUBERT, Christian, DUJIN ZHOU, SHIUAN CHEN, POTTER, Barry V. L, REED, Michael J
Published in Clinical cancer research (15.10.2008)
Published in Clinical cancer research (15.10.2008)
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