2-Difluoromethyloestrone 3- O-sulphamate, a highly potent steroid sulphatase inhibitor
Reed, Julie E, Lawrence Woo, L.W, Robinson, James J, Leblond, Bertrand, Leese, Mathew P, Purohit, Atul, Reed, Michael J, Potter, Barry V.L
Published in Biochemical and biophysical research communications (23.04.2004)
Published in Biochemical and biophysical research communications (23.04.2004)
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Journal Article
Inhibition of MDA-MB-231 cell cycle progression and cell proliferation by C-2-substituted oestradiolmono- andbis-3-O-sulphamates
Raobaikady, Bindumalini, Reed, Michael J., Leese, Mathew P., Potter, Barry V.L., Purohit, Atul
Published in International journal of cancer (20.10.2005)
Published in International journal of cancer (20.10.2005)
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Journal Article
Development of hormone-dependent prostate cancer models for the evaluation of inhibitors of 17beta-hydroxysteroid dehydrogenase type 3
Day, Joanna M, Tutill, Helena J, Foster, Paul A, Bailey, Helen V, Heaton, Wesley B, Sharland, Christopher M, Vicker, Nigel, Potter, Barry V L, Purohit, Atul, Reed, Michael J
Published in Molecular and cellular endocrinology (25.03.2009)
Published in Molecular and cellular endocrinology (25.03.2009)
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Journal Article
The design of novel 17beta-hydroxysteroid dehydrogenase type 3 inhibitors
Vicker, Nigel, Sharland, Christopher M, Heaton, Wesley B, Gonzalez, Ana M Ramos, Bailey, Helen V, Smith, Andrew, Springall, Jeremy S, Day, Joanna M, Tutill, Helena J, Reed, Michael J, Purohit, Atul, Potter, Barry V L
Published in Molecular and cellular endocrinology (25.03.2009)
Published in Molecular and cellular endocrinology (25.03.2009)
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Journal Article
Cytokines in human breast cyst fluid
Parish, David C., Ghilchik, Margaret W., Day, Joanna M., Eaton, James, Purohit, Atul, Reed, Michael J.
Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
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Journal Article
Novel non-steroidal inhibitors of human 11beta-hydroxysteroid dehydrogenase type 1
Vicker, Nigel, Su, Xiangdong, Ganeshapillai, Dharshini, Smith, Andrew, Purohit, Atul, Reed, Michael J, Potter, Barry V L
Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
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Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
Journal Article
Inhibition of human and rat 11beta-hydroxysteroid dehydrogenase type 1 by 18beta-glycyrrhetinic acid derivatives
Su, Xiangdong, Vicker, Nigel, Lawrence, Harshani, Smith, Andrew, Purohit, Atul, Reed, Michael J, Potter, Barry V L
Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
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Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
Journal Article
Differential effects of estrone and estrone-3-O-sulfamate derivatives on mitotic arrest, apoptosis, and microtubule assembly in human breast cancer cells
MACCARTHY-MORROGH, Lucy, TOWNSEND, Paul A, PUROHIT, Atul, HEJAZ, Hatem A. M, POTTER, Barry V. L, REED, Michael J, PACKHAM, Graham
Published in Cancer research (Chicago, Ill.) (01.10.2000)
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Published in Cancer research (Chicago, Ill.) (01.10.2000)
Journal Article
Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity
Jackson, Toby, Woo, L W Lawrence, Trusselle, Melanie N, Chander, Surinder K, Purohit, Atul, Reed, Michael J, Potter, Barry V L
Published in Organic & biomolecular chemistry (21.10.2007)
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Published in Organic & biomolecular chemistry (21.10.2007)
Journal Article
Inhibition of MCF-7 breast cancer cell proliferation and in vivo steroid sulphatase activity by 2-methoxyoestradiol-bis-sulphamate
Raobaikady, Bindumalini, Purohit, Atul, Chander, Surinder K., Woo, L.W.Lawrence, Leese, Mathew P., Potter, Barry V.L., Reed, Michael J.
Published in Journal of steroid biochemistry and molecular biology (01.02.2003)
Published in Journal of steroid biochemistry and molecular biology (01.02.2003)
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Journal Article
Conference Proceeding
Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential
Howarth, Nicola M, Purohit, Atul, Reed, Michael J, Potter, Barry V. L
Published in Journal of medicinal chemistry (01.01.1994)
Published in Journal of medicinal chemistry (01.01.1994)
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Journal Article
Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II
Vicker, Nigel, Ho, Yaikat, Robinson, James, Woo, Lawrence L.W., Purohit, Atul, Reed, Michael J., Potter, Barry V.L.
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
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Journal Article
Lack of aromatisation of the 3-keto-4-ene metabolite of tibolone to an estrogenic derivative
Raobaikady, Bindumalini, Parsons, Michael F.C., Reed, Michael J., Purohit, Atul
Published in Steroids (01.07.2006)
Published in Steroids (01.07.2006)
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Journal Article
INHIBITORS OF 17BETA-HYDROXYSTEROID DEHYDROGENASE
BAILEY HELEN VICTORIA, DAY JOANNA MARY, POTTER BARRY VICTOR LLOYD, PUROHIT ATUL, VICKER NIGEL, HEATON WESLEY
Year of Publication 10.09.2010
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Year of Publication 10.09.2010
Patent
Benzothiazole derivatives as novel inhibitors of human 11beta-hydroxysteroid dehydrogenase type 1
Su, Xiangdong, Vicker, Nigel, Ganeshapillai, Dharshini, Smith, Andrew, Purohit, Atul, Reed, Michael J, Potter, Barry V L
Published in Molecular and cellular endocrinology (27.03.2006)
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Published in Molecular and cellular endocrinology (27.03.2006)
Journal Article
Novel D-ring modified steroid derivatives as potent, non-estrogenic, steroid sulfatase inhibitors with in vivo activity
Fischer, Delphine S., Chander, Surinder K., Woo, L.W.Lawrence, Fenton, Janine C., Purohit, Atul, Reed, Michael J., Potter, Barry V.L.
Published in Journal of steroid biochemistry and molecular biology (01.02.2003)
Published in Journal of steroid biochemistry and molecular biology (01.02.2003)
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Journal Article
Conference Proceeding