Mice Lacking Dopamine D4 Receptors Are Supersensitive to Ethanol, Cocaine, and Methamphetamine
Rubinstein, Marcelo, Phillips, Tamara J., Bunzow, James R., Falzone, Tomás L., Dziewczapolski, Gustavo, Zhang, Ge, Fang, Yuan, Larson, Jennifer L., McDougall, John A., Chester, Julia A., Saez, Carmen, Pugsley, Thomas A., Gershanik, Oscar, Low, Malcolm J., Grandy, David K.
Published in Cell (19.09.1997)
Published in Cell (19.09.1997)
Get full text
Journal Article
3-Arylimino-2-indolones Are Potent and Selective Galanin GAL3 Receptor Antagonists
Konkel, Michael J, Lagu, Bharat, Boteju, Lakmal W, Jimenez, Hermogenes, Noble, Stewart, Walker, Mary W, Chandrasena, Gamini, Blackburn, Thomas P, Nikam, Sham S, Wright, Jon L, Kornberg, Brian E, Gregory, Tracy, Pugsley, Thomas A, Akunne, Hyacinth, Zoski, Kim, Wise, Lawrence D
Published in Journal of medicinal chemistry (29.06.2006)
Published in Journal of medicinal chemistry (29.06.2006)
Get full text
Journal Article
Synthesis and Pharmacological Evaluation of Thiopyran Analogues of the Dopamine D3 Receptor-Selective Agonist (4aR,10bR)-(+)-trans-3,4,4a,10b- Tetrahydro-4-n-propyl-2H,5H-[1]benzopyrano[4,3-b]-1,4-oxazin-9-ol (PD 128907)
van Vliet, L. Alexander, Rodenhuis, Nienke, Dijkstra, Durk, Wikström, Håkan, Pugsley, Thomas A, Serpa, Kevin A, Meltzer, Leonard T, Heffner, Thomas G, Wise, Lawrence D, Lajiness, Mary E, Huff, Rita M, Svensson, Kjell, Sundell, Staffan, Lundmark, Max
Published in Journal of medicinal chemistry (27.07.2000)
Published in Journal of medicinal chemistry (27.07.2000)
Get full text
Journal Article
Design, Synthesis, and Evaluation of Chromen-2-ones as Potent and Selective Human Dopamine D4 Antagonists
Kesten, Suzanne R, Heffner, Thomas G, Johnson, Stephen J, Pugsley, Thomas A, Wright, Jonathan L, Wise, Lawrence D
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
Get full text
Journal Article
Isoindolinone enantiomers having affinity for the dopamine D4 receptor
BELLIOTTI, T. R, BRINK, W. A, WISE, L. D, KESTEN, S. R, RUBIN, J. R, WUSTROW, D. J, ZOSKI, K. T, WHETZEL, S. Z, CORBIN, A. E, PUGSLEY, T. A, HEFFNER, T. G
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Get full text
Journal Article
Synthesis and dopamine agonist properties of (+)-trans-3,4,4a,10b-tetrahydro-4-propyl-2H,5H-[1]benzopyrano[4,3-b]-1,4-oxazin-9-ol and its enantiomers
DeWald, Horace A, Heffner, Thomas G, Jaen, Juan C, Lustgarten, David M, McPhail, Andrew T, Meltzer, Leonard T, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (01.01.1990)
Published in Journal of medicinal chemistry (01.01.1990)
Get full text
Journal Article
Further Characterization of Structural Requirements for Ligands at the Dopamine D2 and D3 Receptor: Exploring the Thiophene Moiety
Dijkstra, Durk, Rodenhuis, Nienke, Vermeulen, Erik S, Pugsley, Thomas A, Wise, Lawrence D, Wikström, Håkan V
Published in Journal of medicinal chemistry (04.07.2002)
Published in Journal of medicinal chemistry (04.07.2002)
Get full text
Journal Article
Chromeno[3,4-c]pyridin-5-ones: Selective Human Dopamine D4 Receptor Antagonists as Potential Antipsychotic Agents
Unangst, Paul C, Capiris, Thomas, Connor, David T, Heffner, Thomas G, MacKenzie, Robert G, Miller, Steven R, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (15.08.1997)
Published in Journal of medicinal chemistry (15.08.1997)
Get full text
Journal Article
4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties
Jaen, Juan C, Wise, Lawrence D, Caprathe, Bradley W, Tecle, Haile, Bergmeier, Stephen, Humblet, Christine C, Heffner, Thomas G, Meltzer, Leonard T, Pugsley, Thomas A
Published in Journal of medicinal chemistry (01.01.1990)
Published in Journal of medicinal chemistry (01.01.1990)
Get full text
Journal Article
Affinity for Dopamine D2, D3, and D4 Receptors of 2-Aminotetralins. Relevance of D2 Agonist Binding for Determination of Receptor Subtype Selectivity
van Vliet, L. Alexander, Tepper, Pieter G, Dijkstra, Durk, Damsma, Geert, Wikström, Håkan, Pugsley, Thomas A, Akunne, Hyacinth C, Heffner, Thomas G, Glase, Shelly A, Wise, Lawrence D
Published in Journal of medicinal chemistry (11.10.1996)
Published in Journal of medicinal chemistry (11.10.1996)
Get full text
Journal Article
The discovery of PD 89211 and related compounds: Selective dopamine D4 receptor antagonists
Pugsley, Thomas A, Shih, Yu Hsin, Whetzel, Steven Z, Zoski, Kim, Van Leeuwen, Don, Akunne, Hyacinth, Mackenzie, R, Heffner, Thomas G, Wustrow, David, Wise, Lawrence D
Published in Progress in neuro-psychopharmacology & biological psychiatry (01.02.2002)
Published in Progress in neuro-psychopharmacology & biological psychiatry (01.02.2002)
Get full text
Journal Article
Thiazoloindans and Thiazolobenzopyrans: A Novel Class of Orally Active Central Dopamine (Partial) Agonists
van Vliet, L. Alexander, Rodenhuis, Nienke, Wikström, Håkan, Pugsley, Thomas A, Serpa, Kevin A, Meltzer, Leonard T, Heffner, Thomas G, Wise, Lawrence D, Lajiness, Mary E, Huff, Rita M, Svensson, Kjell, Haenen, Guido R. M. M, Bast, Aalt
Published in Journal of medicinal chemistry (21.09.2000)
Published in Journal of medicinal chemistry (21.09.2000)
Get full text
Journal Article
Synthesis and potential antipsychotic activity of 1H-imidazo[1,2-c]pyrazolo[3,4-e]pyrimidines
DeWald, Horace A, Beeson, Nicholas W, Hershenson, Fred M, Wise, Lawrence D, Downs, David A, Heffner, Thomas G, Coughenour, Linda L, Pugsley, Thomas A
Published in Journal of medicinal chemistry (01.02.1988)
Published in Journal of medicinal chemistry (01.02.1988)
Get full text
Journal Article
A rapid filtration assay for soluble receptors using polyethylenimine-treated filters
Bruns, Robert F., Lawson-Wendling, Karen, Pugsley, Thomas A.
Published in Analytical biochemistry (01.07.1983)
Published in Analytical biochemistry (01.07.1983)
Get full text
Journal Article
A Series of 6- and 7-Piperazinyl- and -Piperidinylmethylbenzoxazinones with Dopamine D4 Antagonist Activity: Discovery of a Potential Atypical Antipsychotic Agent
Belliotti, Thomas R, Wustrow, David J, Brink, Wouter A, Zoski, Kim T, Shih, Yu-Hsin, Whetzel, Steven Z, Georgic, Lynn M, Corbin, Ann E, Akunne, Hyacinth C, Heffner, Thomas G, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (16.12.1999)
Published in Journal of medicinal chemistry (16.12.1999)
Get full text
Journal Article
A New Type of Prodrug of Catecholamines: An Opportunity To Improve the Treatment of Parkinson's Disease
Venhuis, Bastiaan J, Rodenhuis, Nienke, Wikström, Håkan V, Wustrow, David, Meltzer, Leonard T, Wise, Lawrence D, Johnson, Stephen J, Pugsley, Thomas A, Sundell, Staffan, Dijkstra, Durk
Published in Journal of medicinal chemistry (29.08.2002)
Published in Journal of medicinal chemistry (29.08.2002)
Get full text
Journal Article
Substituted [(4-Phenylpiperazinyl)- methyl]benzamides: Selective Dopamine D4 Agonists
Glase, Shelly A, Akunne, Hyacinth C, Georgic, Lynn M, Heffner, Thomas G, MacKenzie, Robert G, Manley, Peter J, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (06.06.1997)
Published in Journal of medicinal chemistry (06.06.1997)
Get full text
Journal Article
Discovery of selective dopamine D4 receptor antagonists: 1-Aryloxy-3-(4-aryloxypiperidinyl)-2-propanols
Wright, Jon L., Gregory, Tracy F., Heffner, Thomas G., MacKenzie, Robert G., Pugsley, Thomas A., Meulen, Seth Vander, Wise, Lawrence D.
Published in Bioorganic & medicinal chemistry letters (03.06.1997)
Published in Bioorganic & medicinal chemistry letters (03.06.1997)
Get full text
Journal Article
(Aryloxy)alkylamines as Selective Human Dopamine D4 Receptor Antagonists: Potential Antipsychotic Agents
Unangst, Paul C, Capiris, Thomas, Connor, David T, Doubleday, Robert, Heffner, Thomas G, MacKenzie, Robert G, Miller, Steven R, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (05.12.1997)
Published in Journal of medicinal chemistry (05.12.1997)
Get full text
Journal Article