Structure-based design of potent and selective inhibitors of collagenase-3 (MMP-13)
Kim, Soong-Hoon, Pudzianowski, Andrew T., Leavitt, Kenneth J., Barbosa, Joseph, McDonnell, Patricia A., Metzler, William J., Rankin, Bruce M., Liu, Richard, Vaccaro, Wayne, Pitts, William
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Synthesis and SAR of pyrrolotriazine-4-one based Eg5 inhibitors
Kim, Kyoung Soon, Lu, Songfeng, Cornelius, Lyndon A., Lombardo, Louis J., Borzilleri, Robert M., Schroeder, Gretchen M., Sheng, Christopher, Rovnyak, George, Crews, Donald, Schmidt, Robert J., Williams, David K., Bhide, Rajeev S., Traeger, Sarah C., McDonnell, Patricia A., Mueller, Luciano, Sheriff, Steven, Newitt, John A., Pudzianowski, Andrew T., Yang, Zheng, Wild, Robert, Lee, Frances Y., Batorsky, Roberta, Ryder, James S., Ortega-Nanos, Marie, Shen, Henry, Gottardis, Marco, Roussell, Deborah L.
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
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Aroylguanidine-based factor Xa inhibitors: The discovery of BMS-344577
Shi, Yan, Li, Chi, O’Connor, Stephen P., Zhang, Jing, Shi, Mengxiao, Bisaha, Sharon N., Wang, Ying, Sitkoff, Doree, Pudzianowski, Andrew T., Huang, Christine, Klei, Herbert E., Kish, Kevin, Yanchunas, Joseph, Liu, Eddie C.-K., Hartl, Karen S., Seiler, Steve M., Steinbacher, Thomas E., Schumacher, William A., Atwal, Karnail S., Stein, Philip D.
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
Cyanoguanidine-based lactam derivatives as a novel class of orally bioavailable factor Xa inhibitors
Shi, Yan, Zhang, Jing, Shi, Mengxiao, O’Connor, Stephen P., Bisaha, Sharon N., Li, Chi, Sitkoff, Doree, Pudzianowski, Andrew T., Chong, Saeho, Klei, Herbert E., Kish, Kevin, Yanchunas, Joseph, Liu, Eddie C.-K., Hartl, Karen S., Seiler, Steve M., Steinbacher, Thomas E., Schumacher, William A., Atwal, Karnail S., Stein, Philip D.
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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Journal Article
Ketene aminal-based lactam derivatives as a novel class of orally active FXa inhibitors
Shi, Yan, Zhang, Jing, Stein, Philip D., Shi, Mengxiao, O’Connor, Stephen P., Bisaha, Sharon N., Li, Chi, Atwal, Karnail S., Bisacchi, Gregory S., Sitkoff, Doree, Pudzianowski, Andrew T., Liu, Eddie C., Hartl, Karen S., Seiler, Steven M., Youssef, Sonia, Steinbacher, Thomas E., Schumacher, William A., Rendina, Alan R., Bozarth, Jeffrey M., Peterson, Tara L., Zhang, Ge, Zahler, Robert
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
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Quantum-chemical studies of model cytochrome P450 hydrocarbon oxidation mechanisms. 1. A MINDO/3 study of hydroxylation and epoxidation pathways for methane and ethylene
Pudzianowski, Andrew T, Loew, Gilda H
Published in Journal of the American Chemical Society (01.08.1980)
Published in Journal of the American Chemical Society (01.08.1980)
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Benzodiazepine-based selective inhibitors of mitochondrial F1F0 ATP hydrolase
HAMANN, Lawrence G, DING, Charles Z, MILLER, Arthur V, MADSEN, Cort S, WANG, Paulina, STEIN, Philip D, PUDZIANOWSKI, Andrew T, GREEN, David W, MONSHIZADEGAN, Hossain, ATWAL, Karnail S
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
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Hydrogen abstractions from methyl groups by atomic oxygen. Kinetic isotope effects calculated from MNDO/UHF results and an assessment of their applicability to monooxygenase-dependent hydroxylations
Pudzianowski, Andrew T, Loew, Gilda H
Published in Journal of physical chemistry (1952) (01.03.1983)
Published in Journal of physical chemistry (1952) (01.03.1983)
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Erratum to “Ketene aminal-based lactam derivatives as a novel class of orally active FXa inhibitors” [Bioorg. Med. Chem. Lett. 15 (2005) 5453–5458]
Shi, Yan, Zhang, Jing, Stein, Philip D., Shi, Mengxiao, O’Connor, Stephen P., Bisaha, Sharon N., Li, Chi, Atwal, Karnail S., Bisacchi, Gregory S., Sitkoff, Doree, Pudzianowski, Andrew T., Liu, Eddie C., Hartl, Karen S., Seiler, Steven M., Youssef, Sonia, Steinbacher, Thomas E., Schumacher, William A., Rendina, Alan R., Bozarth, Jeffrey M., Peterson, Tara L., Zhang, Ge, Zahler, Robert
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Journal Article
Benzodiazepine-based selective inhibitors of mitochondrial F 1 F 0 ATP hydrolase
Hamann, Lawrence G., Ding, Charles Z., Miller, Arthur V., Madsen, Cort S., Wang, Paulina, Stein, Philip D., Pudzianowski, Andrew T., Green, David W., Monshizadegan, Hossain, Atwal, Karnail S.
Published in Bioorganic & medicinal chemistry letters (01.02.2004)
Published in Bioorganic & medicinal chemistry letters (01.02.2004)
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Radiation chemistry of glassy alkaline ice systems from a structural viewpoint
Pudzianowski, Andrew T, Schwartz, Robert N
Published in Journal of physical chemistry (1952) (01.01.1979)
Published in Journal of physical chemistry (1952) (01.01.1979)
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Aromatic isosteres as conformational probes for an isoprenyl subunit: application to inhibitors of squalene synthase
Biller, Scott A., Abt, Jeffrey W., Pudzianowski, Andrew T., Rich, Lois C., Slusarchyk, Dorothy A., Ciosek, Carl.P.
Published in Bioorganic & medicinal chemistry letters (01.04.1993)
Published in Bioorganic & medicinal chemistry letters (01.04.1993)
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