Exploring new targets and chemical space with affinity selection-mass spectrometry
Prudent, Renaud, Annis, D Allen, Dandliker, Peter J, Ortholand, Jean-Yves, Roche, Didier
Published in Nature reviews. Chemistry (01.01.2021)
Published in Nature reviews. Chemistry (01.01.2021)
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Journal Article
A quantitative proteomic analysis of cofilin phosphorylation in myeloid cells and its modulation using the LIM kinase inhibitor Pyr1
Prudent, Renaud, Demoncheaux, Nathalie, Diemer, Hélène, Collin-Faure, Véronique, Kapur, Reuben, Paublant, Fabrice, Lafanechère, Laurence, Cianférani, Sarah, Rabilloud, Thierry
Published in PloS one (14.12.2018)
Published in PloS one (14.12.2018)
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Journal Article
Characterization of Signalling Pathways That Link Apoptosis and Autophagy to Cell Death Induced by Estrone Analogues Which Reversibly Depolymerize Microtubules
Mercier, Anne E, Prudent, Renaud, Pepper, Michael S, De Koning, Leanne, Nolte, Elsie, Peronne, Lauralie, Nel, Marcel, Lafanechère, Laurence, Joubert, Anna M
Published in Molecules (Basel, Switzerland) (29.01.2021)
Published in Molecules (Basel, Switzerland) (29.01.2021)
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Journal Article
A novel inhibitor of the mitochondrial respiratory complex I with uncoupling properties exerts potent antitumor activity
Al Assi, Alaa, Posty, Solène, Lamarche, Frédéric, Chebel, Amel, Guitton, Jérôme, Cottet-Rousselle, Cécile, Prudent, Renaud, Lafanechère, Laurence, Giraud, Stéphane, Dallemagne, Patrick, Suzanne, Peggy, Verney, Aurélie, Genestier, Laurent, Castets, Marie, Fontaine, Eric, Billaud, Marc, Cordier-Bussat, Martine
Published in Cell death & disease (02.05.2024)
Published in Cell death & disease (02.05.2024)
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Journal Article
Functional analysis of the BMP9 response of ALK1 mutants from HHT2 patients: a diagnostic tool for novel ACVRL1 mutations
Ricard, Nicolas, Bidart, Marie, Mallet, Christine, Lesca, Gaetan, Giraud, Sophie, Prudent, Renaud, Feige, Jean-Jacques, Bailly, Sabine
Published in Blood (02.09.2010)
Published in Blood (02.09.2010)
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Journal Article
Sulphamoylated 2-methoxyestradiol analogues induce apoptosis in adenocarcinoma cell lines
Visagie, Michelle, Theron, Anne, Mqoco, Thandi, Vieira, Warren, Prudent, Renaud, Martinez, Anne, Lafanechère, Laurence, Joubert, Annie
Published in PloS one (05.09.2013)
Published in PloS one (05.09.2013)
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Journal Article
Pharmacological Inhibition of LIM Kinase Stabilizes Microtubules and Inhibits Neoplastic Growth
PRUDENT, Renaud, VASSAL-STERMANN, Emilie, VALDAMERI, Glaucio, HONORE, Stéphane, ACI-SECHE, Samia, GRIERSON, David, ANTONIPILLAI, Juliana, RONG LI, DI PIETRO, Attilio, DUMONTET, Charles, BRAGUER, Diane, FLORENT, Jean-Claude, NGUYEN, Chi-Hung, KNAPP, Stefan, BERNARD, Ora, LAFANECHERE, Laurence, PILLET, Catherine, MARTINEZ, Anne, PRUNIER, Chloe, BARETTE, Caroline, SOLEILHAC, Emmanuelle, FILHOL, Odile, BEGHIN, Anne
Published in Cancer research (Chicago, Ill.) (01.09.2012)
Published in Cancer research (Chicago, Ill.) (01.09.2012)
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Journal Article
Preclinical Evaluation of a Novel Small Molecule Inhibitor of LIM Kinases (LIMK) CEL_Amide in Philadelphia-Chromosome Positive ( BCR::ABL+ ) Acute Lymphoblastic Leukemia (ALL)
Berrou, Jeannig, Dupont, Mélanie, Djamai, Hanane, Adicéam, Emilie, Parietti, Véronique, Kaci, Anna, Clappier, Emmanuelle, Cayuela, Jean-Michel, Baruchel, André, Paublant, Fabrice, Prudent, Renaud, Ghysdael, Jacques, Gardin, Claude, Dombret, Hervé, Braun, Thorsten
Published in Journal of clinical medicine (15.11.2022)
Published in Journal of clinical medicine (15.11.2022)
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Journal Article
Specific Targeting of Plant and Apicomplexa Parasite Tubulin through Differential Screening Using In Silico and Assay-Based Approaches
Soleilhac, Emmanuelle, Brillet-Guéguen, Loraine, Roussel, Véronique, Prudent, Renaud, Touquet, Bastien, Dass, Sheena, Aci-Sèche, Samia, Kasam, Vinod, Barette, Caroline, Imberty, Anne, Breton, Vincent, Vantard, Marylin, Horvath, Dragos, Botté, Cyrille, Tardieux, Isabelle, Roy, Sylvaine, Maréchal, Eric, Lafanechère, Laurence
Published in International journal of molecular sciences (09.10.2018)
Published in International journal of molecular sciences (09.10.2018)
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Journal Article
New potent dual inhibitors of CK2 and Pim kinases: discovery and structural insights
López-Ramos, Miriam, Prudent, Renaud, Moucadel, Virginie, Sautel, Céline F, Barette, Caroline, Lafanechère, Laurence, Mouawad, Liliane, Grierson, David, Schmidt, Frédéric, Florent, Jean-Claude, Filippakopoulos, Panagis, Bullock, Alex N, Knapp, Stefan, Reiser, Jean-Baptiste, Cochet, Claude
Published in The FASEB journal (01.09.2010)
Published in The FASEB journal (01.09.2010)
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Journal Article
Two Antagonistic Microtubule Targeting Drugs Act Synergistically to Kill Cancer Cells
Peronne, Lauralie, Denarier, Eric, Rai, Ankit, Prudent, Renaud, Vernet, Audrey, Suzanne, Peggy, Ramirez-Rios, Sacnicté, Michallet, Sophie, Guidetti, Mélanie, Vollaire, Julien, Lucena-Agell, Daniel, Ribba, Anne-Sophie, Josserand, Véronique, Coll, Jean-Luc, Dallemagne, Patrick, Díaz, J. Fernando, Oliva, María Ángela, Sadoul, Karin, Akhmanova, Anna, Andrieux, Annie, Lafanechère, Laurence
Published in Cancers (01.08.2020)
Published in Cancers (01.08.2020)
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Journal Article
Functional Analysis of Protein Kinase CK2 of the Human Malaria Parasite Plasmodium falciparum
Holland, Zoë, Prudent, Renaud, Reiser, Jean-Baptiste, Cochet, Claude, Doerig, Christian
Published in Eukaryotic Cell (01.03.2009)
Published in Eukaryotic Cell (01.03.2009)
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Journal Article
Antitumoral activity of allosteric inhibitors of protein kinase CK2
Moucadel, Virginie, Prudent, Renaud, Sautel, Céline F, Teillet, Florence, Barette, Caroline, Lafanechere, Laurence, Receveur-Brechot, Veronique, Cochet, Claude
Published in Oncotarget (01.12.2011)
Published in Oncotarget (01.12.2011)
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Journal Article
Novel synthetic pharmacophores inducing a stabilization of cellular microtubules
Martinez, Anne, Soleilhac, Emmanuelle, Barette, Caroline, Prudent, Renaud, Gozzi, Gustavo J, Vassal-Stermann, Emilie, Pillet, Catherine, Di Pietro, Attilio, Fauvarque, Marie-Odile, Lafanechere, Laurence
Published in Current cancer drug targets (01.01.2015)
Published in Current cancer drug targets (01.01.2015)
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Journal Article
Expanding the chemical diversity of CK2 inhibitors
Prudent, Renaud, Moucadel, Virginie, López-Ramos, Miriam, Aci, Samia, Laudet, Beatrice, Mouawad, Liliane, Barette, Caroline, Einhorn, Jacques, Einhorn, Cathy, Denis, Jean-Noel, Bisson, Gilles, Schmidt, Frédéric, Roy, Sylvaine, Lafanechere, Laurence, Florent, Jean-Claude, Cochet, Claude
Published in Molecular and cellular biochemistry (01.09.2008)
Published in Molecular and cellular biochemistry (01.09.2008)
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Journal Article
Affinity selection mass spectrometry speeding drug discovery
Prudent, Renaud, Lemoine, Hugues, Walsh, Jarrod, Roche, Didier
Published in Drug discovery today (01.11.2023)
Published in Drug discovery today (01.11.2023)
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Journal Article
LIM kinases: cofilin and beyond
Prunier, Chloé, Prudent, Renaud, Kapur, Reuben, Sadoul, Karin, Lafanechère, Laurence
Published in Oncotarget (20.06.2017)
Published in Oncotarget (20.06.2017)
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Journal Article
Identification of Polyoxometalates as Nanomolar Noncompetitive Inhibitors of Protein Kinase CK2
Prudent, Renaud, Moucadel, Virginie, Laudet, Béatrice, Barette, Caroline, Lafanechère, Laurence, Hasenknopf, Bernold, Li, Joaquim, Bareyt, Sébastian, Lacôte, Emmanuel, Thorimbert, Serge, Malacria, Max, Gouzerh, Pierre, Cochet, Claude
Published in Chemistry & biology (21.07.2008)
Published in Chemistry & biology (21.07.2008)
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