The evolution of amidine-based brain penetrant BACE1 inhibitors
Oehlrich, Daniel, Prokopcova, Hana, Gijsen, Harrie J.M.
Published in Bioorganic & medicinal chemistry letters (01.05.2014)
Published in Bioorganic & medicinal chemistry letters (01.05.2014)
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C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp(3) C-H Activation
Prokopcova, Hana, Bergman, Sheba D., Aelvoet, Karel, Smout, Veerle, Herrebout, Wouter, Van der Veken, Benjamin, Meerpoel, Lieven, Maes, Bert U. W.
Published in Chemistry : a European journal (22.11.2010)
Published in Chemistry : a European journal (22.11.2010)
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Structure-Activity Relationships and Molecular Docking of Novel Dihydropyrimidine-Based Mitotic Eg5 Inhibitors
Prokopcová, Hana, Dallinger, Doris, Uray, Georg, Kaan, Hung Yi Kristal, Ulaganathan, Venkatasubramanian, Kozielski, Frank, Laggner, Christian, Kappe, C. Oliver
Published in ChemMedChem (04.10.2010)
Published in ChemMedChem (04.10.2010)
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4-Cyano-6,7-dimethoxycarbostyrils with Solvent- and pH-Independent High Fluorescence Quantum Yields and Emission Maxima
Ahvale, Appasaheb B., Prokopcová, Hana, Šefčovičová, Jana, Steinschifter, Waltraud, Täubl, Anna E., Uray, Georg, Stadlbauer, Wolfgang
Published in European Journal of Organic Chemistry (01.01.2008)
Published in European Journal of Organic Chemistry (01.01.2008)
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Structural Basis for Inhibition of Eg5 by Dihydropyrimidines: Stereoselectivity of Antimitotic Inhibitors Enastron, Dimethylenastron and Fluorastrol
Kaan, Hung Yi Kristal, Ulaganathan, Venkatasubramanian, Rath, Oliver, Prokopcová, Hana, Dallinger, Doris, Kappe, C. Oliver, Kozielski, Frank
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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Ruthenium‐Catalyzed Reductive Arylation of N‐(2‐Pyridinyl)amides with Isopropanol and Arylboronate Esters
Ronson, Thomas O., Renders, Evelien, Van Steijvoort, Ben F., Wang, Xubin, Wybon, Clarence C. D., Prokopcová, Hana, Meerpoel, Lieven, Maes, Bert U. W.
Published in Angewandte Chemie International Edition (08.01.2019)
Published in Angewandte Chemie International Edition (08.01.2019)
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Journal Article
The Role of the Alcohol and Carboxylic Acid in Directed Ruthenium-Catalyzed C(sp3)H α-Alkylation of Cyclic Amines
Bergman, Sheba D., Storr, Thomas E., Prokopcová, Hana, Aelvoet, Karel, Diels, Gaston, Meerpoel, Lieven, Maes, Bert U. W.
Published in Chemistry : a European journal (13.08.2012)
Published in Chemistry : a European journal (13.08.2012)
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A Bayesian Approach to Kinetic Modeling of Accelerated Stability Studies and Shelf Life Determination
Chau, Joris, Altan, Stan, Burggraeve, Anneleen, Coppenolle, Hans, Kifle, Yimer Wasihun, Prokopcova, Hana, Van Daele, Timothy, Sterckx, Hans
Published in AAPS PharmSciTech (30.11.2023)
Published in AAPS PharmSciTech (30.11.2023)
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Microwave-assisted one-pot diboration/Suzuki cross-couplings. A rapid route to tetrasubstituted alkenes
Prokopcová, Hana, Ramírez, Jesús, Fernández, Elena, Kappe, C. Oliver
Published in Tetrahedron letters (11.08.2008)
Published in Tetrahedron letters (11.08.2008)
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Journal Article
1,4-Oxazine β‑Secretase 1 (BACE1) Inhibitors: From Hit Generation to Orally Bioavailable Brain Penetrant Leads
Rombouts, Frederik J. R, Tresadern, Gary, Delgado, Oscar, Martínez-Lamenca, Carolina, Van Gool, Michiel, García-Molina, Aránzazu, Alonso de Diego, Sergio A, Oehlrich, Daniel, Prokopcova, Hana, Alonso, José Manuel, Austin, Nigel, Borghys, Herman, Van Brandt, Sven, Surkyn, Michel, De Cleyn, Michel, Vos, Ann, Alexander, Richard, Macdonald, Gregor, Moechars, Dieder, Gijsen, Harrie, Trabanco, Andrés A
Published in Journal of medicinal chemistry (22.10.2015)
Published in Journal of medicinal chemistry (22.10.2015)
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Journal Article
Optimization of 1,4-Oxazine β‑Secretase 1 (BACE1) Inhibitors Toward a Clinical Candidate
Gijsen, Harrie J. M, Alonso de Diego, Sergio A, De Cleyn, Michel, García-Molina, Aránzazu, Macdonald, Gregor J, Martínez-Lamenca, Carolina, Oehlrich, Daniel, Prokopcova, Hana, Rombouts, Frederik J. R, Surkyn, Michel, Trabanco, Andrés A, Van Brandt, Sven, Van den Bossche, Dries, Van Gool, Michiel, Austin, Nigel, Borghys, Herman, Dhuyvetter, Deborah, Moechars, Diederik
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
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Journal Article
Evaluation of a Series of β‑Secretase 1 Inhibitors Containing Novel Heteroaryl-Fused-Piperazine Amidine Warheads
Oehlrich, Daniel, Peschiulli, Aldo, Tresadern, Gary, Van Gool, Michiel, Vega, Juan Antonio, De Lucas, Ana Isabel, Alonso de Diego, Sergio A, Prokopcova, Hana, Austin, Nigel, Van Brandt, Sven, Surkyn, Michel, De Cleyn, Michel, Vos, Ann, Rombouts, Frederik J. R, Macdonald, Gregor, Moechars, Dieder, Gijsen, Harrie J. M, Trabanco, Andrés A
Published in ACS medicinal chemistry letters (08.08.2019)
Published in ACS medicinal chemistry letters (08.08.2019)
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Journal Article
C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp3 CH Activation
Prokopcová, Hana, Bergman, Sheba D., Aelvoet, Karel, Smout, Veerle, Herrebout, Wouter, Van der Veken, Benjamin, Meerpoel, Lieven, Maes, Bert U. W.
Published in Chemistry : a European journal (22.11.2010)
Published in Chemistry : a European journal (22.11.2010)
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Journal Article
Correction to Optimization of 1,4-Oxazine β‑Secretase 1 (BACE1) Inhibitors Toward a Clinical Candidate
Gijsen, Harrie J. M, Alonso de Diego, Sergio A, De Cleyn, Michel, García-Molina, Aránzazu, Macdonald, Gregor J, Martinez-Lamenca, Carolina, Oehlrich, Daniel, Prokopcova, Hana, Rombouts, Frederik J. R, Surkyn, Michel, Trabanco, Andrés A, Van Brandt, Sven, Van den Bossche, Dries, Van Gool, Michiel, Austin, Nigel, Borghys, Herman, Dhuyvetter, Deborah, Urmaliya, Vijay, Teisman, Ard, Moechars, Diederik
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
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Journal Article